BDBM50030196 CHEMBL3354065
SMILES CCCCC1CCN(CCCN2C(=O)CCc3ccccc23)CC1
InChI Key InChIKey=PHMGZAICAOYEAF-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50030196
Affinity DataEC50: 263nMAssay Description:Positive modulatory activity at human M1 receptor expressed in HEK293T cells assessed as effect on xanomeline-induced response by BRET based Gq prote...More data for this Ligand-Target Pair
Affinity DataEC50: 191nMAssay Description:Positive modulatory activity at human M1 receptor expressed in HEK293T cells assessed as effect on carbachol-induced response by BRET based Gq protei...More data for this Ligand-Target Pair
Affinity DataEC50: 832nMAssay Description:Agonist activity at human M1 receptor expressed in HEK293T cells by BRET based beta-arrestin engagement assayMore data for this Ligand-Target Pair
Affinity DataEC50: 102nMAssay Description:Agonist activity at human M1 receptor expressed in HEK293T cells by BRET based Gq protein activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Positive modulatory activity at human M1 receptor expressed in HEK293T cells assessed as effect on xanomeline-induced response by BRET based Gq prote...More data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Positive modulatory activity at human M1 receptor expressed in HEK293T cells assessed as effect on carbachol-induced response by BRET based Gq protei...More data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Agonist activity at human M1 receptor expressed in HEK293T cells by BRET based Gq protein engagement assayMore data for this Ligand-Target Pair
Affinity DataEC50: 275nMAssay Description:Agonist activity at human M4 receptor expressed in HEK293T cells by BRET based Gq protein activation assayMore data for this Ligand-Target Pair