BDBM50176263 3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenol::CHEMBL1400::O-DESMETHYL TRAMADOL::Ultracet::rel-3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenol
SMILES CN(C)C[C@H]1CCCC[C@]1(O)c1cccc(O)c1
InChI Key InChIKey=UWJUQVWARXYRCG-HIFRSBDPSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50176263
TargetMu-type opioid receptor(Homo sapiens (Human))
Rensselaer Polytechnic Institute
Curated by ChEMBL
Rensselaer Polytechnic Institute
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at human MOR expressed in CHO cell membranes after 60 mins by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Rensselaer Polytechnic Institute
Curated by ChEMBL
Rensselaer Polytechnic Institute
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation after 1 hr by HTRF ...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Rensselaer Polytechnic Institute
Curated by ChEMBL
Rensselaer Polytechnic Institute
Curated by ChEMBL
Affinity DataEC50: 245nMAssay Description:Inhibition of Trypanosoma cruzi recombinant triosephosphate isomerase after 2 hrsMore data for this Ligand-Target Pair
Affinity DataEC50: 245nMAssay Description:Agonist activity at rat mu opioid receptor expressed in CHO cells incubated for 1 hr by [35S]GTPgammaS binding based liquid scintillation counting me...More data for this Ligand-Target Pair