BDBM50246759 CHEMBL4098772
SMILES Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOc2cc3nccc(Nc4ccc5scnc5c4)c3cc2S(=O)(=O)C(C)(C)C)C(C)(C)C)cc1
InChI Key InChIKey=RIEGJNXDHULIKM-GPPJZCFZSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50246759
Targetvon Hippel-Lindau disease tumor suppressor(Homo sapiens (Human))
Shaoxing University
Curated by ChEMBL
Shaoxing University
Curated by ChEMBL
Affinity DataIC50: 656nMAssay Description:Binding affinity to VHL in human THP-1 cellsMore data for this Ligand-Target Pair
Targetvon Hippel-Lindau disease tumor suppressor(Homo sapiens (Human))
Shaoxing University
Curated by ChEMBL
Shaoxing University
Curated by ChEMBL
Affinity DataKd: 500nMAssay Description:Binding affinity to VHL (unknown origin) assessed as reduction of HIF1alpha derived peptide binding to VHL complex by competitive binding fluorescenc...More data for this Ligand-Target Pair