BDBM50591809 CHEMBL5203365
SMILES OC(=O)[C@@H]1CCCN(C1)\C=C\C=C\c1ccccc1-c1ccccc1-c1ccccc1
InChI Key InChIKey=PVPUJGNLADUCLH-PNPAXDADSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50591809
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Isf College Of Pharmacy
Curated by ChEMBL
Isf College Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Binding affinity to mouse GAT-1 expressed in human HEK293 cells assessed as inhibition constant in presence of NO711 marker by competitive binding as...More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Isf College Of Pharmacy
Curated by ChEMBL
Isf College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 166nMAssay Description:Inhibition of mouse GAT-1 expressed in human HEK293 cells assessed as inhibition of [3H]GABA uptakeMore data for this Ligand-Target Pair