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Found 2 Enz. Inhib. hit(s) with Target = 'Sodium- and chloride-dependent GABA transporter 1' and Ligand = 'BDBM50591809'
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Isf College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50591809(CHEMBL5203365)
Affinity DataKi:  79nMAssay Description:Binding affinity to mouse GAT-1 expressed in human HEK293 cells assessed as inhibition constant in presence of NO711 marker by competitive binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Isf College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50591809(CHEMBL5203365)
Affinity DataIC50:  166nMAssay Description:Inhibition of mouse GAT-1 expressed in human HEK293 cells assessed as inhibition of [3H]GABA uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed