Compile Data Set for Download or QSAR
Report error Found 1131 Enz. Inhib. hit(s) with Target = 'Bcl-2-related protein A1'
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50210070(CHEMBL3883565)
Affinity DataKi: <0.100nMAssay Description:Inhibition of FITC-betaA-DIIRNIARHLAQVGDSMRSI-NH2 binding to recombinant human Bcl2A1 (1 to 152 residues) BH3 binding site expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetBcl-2-related protein A1 [1-149](Human)
University of California Riverside

LigandPNGBDBM218795(130E7 | Ac-λIAQELRRIGDEFNAYYARR-NH2)
Affinity DataKd:  2.60nMpH: 7.4 T: 2°CAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558852(CHEMBL4747465)
Affinity DataIC50: 6.5nMAssay Description:Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558851(CHEMBL4782684)
Affinity DataIC50: 6.60nMAssay Description:Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1 [1-149](Human)
University of California Riverside

LigandPNGBDBM218788(hNOXA | Ac-CATQLRRFGDKLNFRQKLLN-NH2)
Affinity DataIC50: 7.5nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50210070(CHEMBL3883565)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of FITC-betaA-DIIRNIARHLAQVGDSMRSI-NH2 binding to recombinant human Bcl2A1 (1 to 152 residues) BH3 binding site expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetBcl-2-related protein A1 [1-149](Human)
University of California Riverside

LigandPNGBDBM218795(130E7 | Ac-λIAQELRRIGDEFNAYYARR-NH2)
Affinity DataIC50: 8.70nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558851(CHEMBL4782684)
Affinity DataKi:  10nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM32274(cid_1002249 | SMR000115103 | 2,5-dichloro-3-(4-met...)
Affinity DataEC50:  10nMpH: 7.4 T: 2°CAssay Description:The multiplex is constructed by using beads for each protein target that have been labeled with varying intensities of red color, so that each assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2009
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558856(CHEMBL4791348)
Affinity DataIC50: 13nMAssay Description:Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1 [1-149](Human)
University of California Riverside

LigandPNGBDBM218796(130D11 | Ac-λAQELR(Xi)IGD(Xi+4)FNAYYARR-NH2)
Affinity DataIC50: 13.9nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558854(CHEMBL4755711)
Affinity DataIC50: 14nMAssay Description:Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1 [1-149](Human)
University of California Riverside

LigandPNGBDBM218791(hNOXAs | Ac-CATQLRRFGDKLN-NH2)
Affinity DataIC50: 15nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50587033(CHEMBL5075478)
Affinity DataIC50: 18nMAssay Description:Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM333146(US10196404, Example 1 | Compound I | US10196404, E...)
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal His6-tagged Bfl-1 (1 to 151 residues) (unknown origin) expressed in Escherichia coli using Fluor 647-labeled BAK peptide WIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM33133(SMR000225370 | MLS000702137 | cid_15945005 | 3-(4-...)
Affinity DataEC50:  20nMpH: 7.4 T: 2°CAssay Description:The multiplex is constructed by using beads for each protein target that have been labeled with varying intensities of red color, so that each assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2009
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558857(CHEMBL4752520)
Affinity DataIC50: 20nMAssay Description:Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50648874(CHEMBL5613766)
Affinity DataIC50: 22nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50610581(CHEMBL5281728)
Affinity DataEC50:  23nMAssay Description:Displacement of fluorescent-labeled BID-BH3 peptide from His-tagged BFL-1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558853(CHEMBL4465826)
Affinity DataIC50: 31nMAssay Description:Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558852(CHEMBL4747465)
Affinity DataKi:  31nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50210069(CHEMBL3884841)
Affinity DataKi:  32nMAssay Description:Inhibition of FITC-betaA-DIIRNIARHLAQVGDSMRSI-NH2 binding to recombinant human Bcl2A1 (1 to 152 residues) BH3 binding site expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM33066(cid_1002248 | 2,5-dichloro-3-[2-(dimethylamino)-5-...)
Affinity DataEC50:  40nMpH: 7.4 T: 2°CAssay Description:The multiplex is constructed by using beads for each protein target that have been labeled with varying intensities of red color, so that each assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2009
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558857(CHEMBL4752520)
Affinity DataKi:  47nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM33134(cid_15945006 | SMR000225371 | MLS000702136 | 5-(4-...)
Affinity DataEC50:  50nMpH: 7.4 T: 2°CAssay Description:The multiplex is constructed by using beads for each protein target that have been labeled with varying intensities of red color, so that each assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2009
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558855(CHEMBL4740212)
Affinity DataIC50: 55nMAssay Description:Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50648872(CHEMBL5613621)
Affinity DataIC50: 63nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM33102(N-ethyl-N-(1-hydroxy-3,4-dioxo-2-naphthalenyl)prop...)
Affinity DataEC50:  80nMpH: 7.4 T: 2°CAssay Description:The multiplex is constructed by using beads for each protein target that have been labeled with varying intensities of red color, so that each assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2009
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM33080(SMR000131460 | MLS000521051 | cid_9550553 | 2-[[7-...)
Affinity DataEC50:  80nMpH: 7.4 T: 2°CAssay Description:The multiplex is constructed by using beads for each protein target that have been labeled with varying intensities of red color, so that each assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2009
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM33097(MLS000521052 | cid_11957209 | 3-[[7-(1,3-benzothia...)
Affinity DataEC50:  80nMpH: 7.4 T: 2°CAssay Description:The multiplex is constructed by using beads for each protein target that have been labeled with varying intensities of red color, so that each assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2009
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558854(CHEMBL4755711)
Affinity DataKi:  82nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1 [1-149](Human)
University of California Riverside

LigandPNGBDBM218789(homo_hNOXA | Ac-hCATQLRRFGDKLNFRQKLLN-NH2)
Affinity DataIC50: 83nMAssay Description:One hundred microliters of a 600 ng/mL solution of biotin-BID (Biotin-lc-EDIIRNIARHLAQVGDSMDR-NH2, where lc indicates a hydrocarbon chain of six meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511123(CHEMBL4522193)
Affinity DataKi:  84nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511124(CHEMBL4533559)
Affinity DataKi:  100nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511138(CHEMBL4576854)
Affinity DataKi:  100nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511138(CHEMBL4576854)
Affinity DataKi:  100nMAssay Description:Displacement of fluorescent-labeled BID-BH3 peptide from His-tagged human BFL-1 (1 to 151 residues) expressed in Escherichia coli BL21 (DE3) assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50210069(CHEMBL3884841)
Affinity DataIC50: 110nMAssay Description:Inhibition of FITC-betaA-DIIRNIARHLAQVGDSMRSI-NH2 binding to recombinant human Bcl2A1 (1 to 152 residues) BH3 binding site expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM33098(MLS000520993 | cid_11957260 | 2-[[7-(1,3-benzothia...)
Affinity DataEC50:  120nMpH: 7.4 T: 2°CAssay Description:The multiplex is constructed by using beads for each protein target that have been labeled with varying intensities of red color, so that each assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2009
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50330250(5,5'-Dibenzyl-6,6',7,7'-tetrahydroxy-3,3'-dimethyl...)
Affinity DataIC50: 122nMAssay Description:Inhibition of FITC-labeled Bim BH3 binding to GST-tagged Bcl2A1 (unknown origin) preincubated for 2 mins followed by FITC-Bim-BH3 addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2020
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50330250(5,5'-Dibenzyl-6,6',7,7'-tetrahydroxy-3,3'-dimethyl...)
Affinity DataIC50: 122nMAssay Description:Inhibition of Bfl-1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM33180(MLS000674027 | 3-[[7-[(5-methyl-1,3,4-thiadiazol-2...)
Affinity DataEC50:  130nMpH: 7.4 T: 2°CAssay Description:The multiplex is constructed by using beads for each protein target that have been labeled with varying intensities of red color, so that each assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2009
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558856(CHEMBL4791348)
Affinity DataKi:  133nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511136(CHEMBL4558313)
Affinity DataKi:  150nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50511125(CHEMBL4462138)
Affinity DataKi:  170nMAssay Description:Inhibition of N-terminal His6-tagged human Bfl-1 (1 to 151 residues), expressed in Escherichia coli Rosetta2 DE3 by fluorescent labeled FAM-Bid pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM33097(MLS000521052 | cid_11957209 | 3-[[7-(1,3-benzothia...)
Affinity DataEC50:  170nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH 1X01 MH079850-01 HTS to identify small molecule regulators of Bcl-2 family protein int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558855(CHEMBL4740212)
Affinity DataKi:  175nMAssay Description:Covalent binding affinity to human Bcl2A1 by FBid based FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50366237(GAMBOGIC ACID)
Affinity DataIC50: 176nMAssay Description:Inhibition of recombinant Bfl-1 (1-152) (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM33107(2-chloro-3-{[4-(diethylamino)phenyl]amino}naphthoq...)
Affinity DataEC50:  180nMpH: 7.4 T: 2°CAssay Description:The multiplex is constructed by using beads for each protein target that have been labeled with varying intensities of red color, so that each assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2009
Entry Details
PCBioAssay
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM39156(CHEMBL1272100 | MLS-0090874.0001 | 3-chloro-1-(3,4...)
Affinity DataIC50: 240nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetBcl-2-related protein A1(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50313364((2S,3R,4R,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylphen...)
Affinity DataIC50: 250nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
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