Compile Data Set for Download or QSAR
Report error Found 2815 Enz. Inhib. hit(s) with Target = 'Beta-1 adrenergic receptor'
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404791BDBM50404791(CHEMBL31025)
Affinity DataKd:  0.00000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404774BDBM50404774(CHEMBL31857)
Affinity DataKd:  0.00000100nMAssay Description:In vivo inhibition of Beta-1 adrenergic receptor in guinea pig right atria after 40 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404790BDBM50404790(CHEMBL13284)
Affinity DataKd:  0.00000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 40 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404790BDBM50404790(CHEMBL13284)
Affinity DataKd:  0.00000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404793BDBM50404793(CHEMBL31638)
Affinity DataKd:  0.0000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404763BDBM50404763(CHEMBL283289)
Affinity DataKd:  0.0000100nMAssay Description:In vivo inhibition of Beta-1 adrenergic receptor in guinea pig right atria after 40 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404796BDBM50404796(Brevibloc | ESMOLOL)
Affinity DataKd:  0.00100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404796BDBM50404796(Brevibloc | ESMOLOL)
Affinity DataKd:  0.00100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 40 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404804BDBM50404804(CHEMBL13365)
Affinity DataKd:  0.00100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 40 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 25761BDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50379086BDBM50379086(CHEMBL2012522 | CHEMBL2012521 | LY-377604)
Affinity DataKi:  0.0230nMAssay Description:Displacement of [125I]Iodocyanopindolol from human adrenergic beta1 receptor expressed in insect sf9 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413482BDBM50413482(CHEMBL443435)
Affinity DataEC50:  0.0398nMAssay Description:Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422862BDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor S190A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422862BDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor W134A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422862BDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat wild type beta-1 adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50568740BDBM50568740(CHEMBL4860528)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50601567BDBM50601567(CHEMBL5206565)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50601551BDBM50601551(CHEMBL5207281)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50601574BDBM50601574(CHEMBL5201074)
Affinity DataKd:  0.0750nMAssay Description:Displacement of [3H]CGP12177 from human beta-1 adrenergic receptor stably expressed in HEK293T cell membrane incubated for 2 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422862BDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0794nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356F mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 25392BDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.0840nMAssay Description:Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 25392BDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.0840nMAssay Description:Agonistic activity was assessed by measuring cAMP accumulation in CHO cell lines expressing cloned human Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 25392BDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.0840nMAssay Description:Agonist activity at human cloned adrenergic beta-1 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 25392BDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.0840nMAssay Description:Agonist activity at human beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 25392BDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  0.0840nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50027663BDBM50027663(Carazolol | 1-(9H-carbazol-4-yloxy)-3-(isopropylam...)
Affinity DataKi:  0.0900nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50318983BDBM50318983(2-((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)pip...)
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404789BDBM50404789(CHEMBL30622)
Affinity DataKd:  0.100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 85818BDBM85818(Fluorocarazolol,(S) | Fluorocarazolol,(R))
Affinity DataKi:  0.114nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50126071BDBM50126071((R)-1-((R)-3-Chloro-phenyl)-2-[2-(7-methoxy-1H-ind...)
Affinity DataEC50:  0.130nMAssay Description:Agonistic activity against human Beta-1 adrenergic receptor by measuring cAMP accumulation in CHO cells expressing beta3-ARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50126076BDBM50126076((R)-1-(3-Chloro-phenyl)-2-[2-(7-methoxy-1H-indol-3...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at Homo sapiens (human) beta1 adrenoreceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81885BDBM81885(CAS_52560-77-7 | 2-(3-tert-Butylamino-2-hydroxypro...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50167072BDBM50167072(CHEMBL3799125)
Affinity DataKi:  0.210nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50098668BDBM50098668(4-(3-tert-Butylamino-2-hydroxy-propoxy)-1,3-dihydr...)
Affinity DataKi:  0.25nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422862BDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.316nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 86453BDBM86453(NSC_3083544 | CAS_73573-87-2 | Formoterol)
Affinity DataEC50:  0.316nMAssay Description:Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 25746BDBM25746(cid_2685 | 2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-meth...)
Affinity DataKd:  0.331nMAssay Description:Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 25748BDBM25748(ICI 89,406 | 3-(2-{[3-(2-cyanophenoxy)-2-hydroxypr...)
Affinity DataKd:  0.331nMAssay Description:Antagonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292219BDBM50292219((2S)-1-(tert-butylamino)-3-[(4-morpholin-4-yl-1,2,...)
Affinity DataKd:  0.363nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50241366BDBM50241366((S)-1-(isopropylamino)-3-(m-tolyloxy)propan-2-ol (...)
Affinity DataKd:  0.380nMAssay Description:Binding affinity to beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 85818BDBM85818(Fluorocarazolol,(S) | Fluorocarazolol,(R))
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50526681BDBM50526681(CHEMBL4537221)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50019443BDBM50019443(LB-46 | 1-(1H-Indol-4-yloxy)-3-isopropylamino-prop...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity at human adrenergic beta-1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50328336BDBM50328336(3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-...)
Affinity DataEC50:  0.570nMAssay Description:Agonist activity at human recombinant adrenergic beta-1 receptor expressed in CHO cells assessed as cyclic AMP formation by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50299900BDBM50299900(5-hydroxy-8-(1-hydroxy-2-(2-methyl-1-o-tolylpropan...)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at human adrenergic beta 1 expressed in CHO-K1 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50578620BDBM50578620(CHEMBL4868585)
Affinity DataEC50:  0.603nMAssay Description:Agonist activity at human beta1 adrenoreceptor overexpressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 25747BDBM25747(4-[3-(tert-butylamino)-2-hydroxypropoxy]-2,3-dihyd...)
Affinity DataKd:  0.620nMpH: 7.4 T: 2°CAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2008
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019443BDBM50019443(LB-46 | 1-(1H-Indol-4-yloxy)-3-isopropylamino-prop...)
Affinity DataKi:  0.660nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25761BDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKi:  0.690nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413485BDBM50413485(CHEMBL483200 | CHEMBL446840)
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
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