Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with Target = 'Elongation of very long chain fatty acids protein 3'
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50250164BDBM50250164(6,6-dimethyl-3-(5-methyl-3-oxo-2-phenyl-2,3-dihydr...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Mouse)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50299971BDBM50299971(4-Fluoro-N-{[(+)-(4S)-2-oxo-6-(1H-pyrazol-5-yl)-4-...)
Affinity DataIC50: 19nMAssay Description:Inhibition of mouse ELOVL3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249844BDBM50249844(3-[2-(4-isopropylphenyl)-5-methyl-3-oxo-2,3-dihydr...)
Affinity DataIC50: 59nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50299971BDBM50299971(4-Fluoro-N-{[(+)-(4S)-2-oxo-6-(1H-pyrazol-5-yl)-4-...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human ELOVL3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Mouse)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249892BDBM50249892(6,6-dimethyl-3-{5-methyl-3-oxo-2-[4-(trifluorometh...)
Affinity DataIC50: 194nMAssay Description:Inhibition of mouse ELOVL3 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249791BDBM50249791(3-[2-(4-chlorophenyl)-5-methyl-3-oxo-2,3-dihydro-1...)
Affinity DataIC50: 221nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249892BDBM50249892(6,6-dimethyl-3-{5-methyl-3-oxo-2-[4-(trifluorometh...)
Affinity DataIC50: 337nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249891BDBM50249891(3-[2-(4-methyllphenyl)-5-methyl-3-oxo-2,3-dihydro-...)
Affinity DataIC50: 375nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249815BDBM50249815(3-[2-(4-methoxyphenyl)-5-methyl-3-oxo-2,3-dihydro-...)
Affinity DataIC50: 503nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Mouse)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50298968BDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 717nMAssay Description:Inhibition of C-terminal V5-epitope-tagged mouse ELOVL3 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Mouse)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293789BDBM50293789(3-endo-(Pyridin-2-ylsulfonyl)-N-[4-(trifluoromethy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse ELOVL3 expressed in Pichia pastoris SND1168More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249843BDBM50249843(3-[2-(4-cyanophenyl)-5-methyl-3-oxo-2,3-dihydro-1H...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50298968BDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL3 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetElongation of very long chain fatty acids protein 3(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293789BDBM50293789(3-endo-(Pyridin-2-ylsulfonyl)-N-[4-(trifluoromethy...)
Affinity DataIC50: 6.94E+3nMAssay Description:Inhibition of human ELOVL3 expressed in Pichia pastoris SND1168More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed