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Found 14 Enz. Inhib. hit(s) with Target = 'Elongation of very long chain fatty acids protein 3'
TargetElongation of very long chain fatty acids protein 3(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50250164(6,6-dimethyl-3-(5-methyl-3-oxo-2-phenyl-2,3-dihydr...)
Affinity DataIC50: >10nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299971(4-Fluoro-N-{[(+)-(4S)-2-oxo-6-(1H-pyrazol-5-yl)-4-...)
Affinity DataIC50:  19nMAssay Description:Inhibition of mouse ELOVL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249844(3-[2-(4-isopropylphenyl)-5-methyl-3-oxo-2,3-dihydr...)
Affinity DataIC50:  59nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50299971(4-Fluoro-N-{[(+)-(4S)-2-oxo-6-(1H-pyrazol-5-yl)-4-...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human ELOVL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249892(6,6-dimethyl-3-{5-methyl-3-oxo-2-[4-(trifluorometh...)
Affinity DataIC50:  194nMAssay Description:Inhibition of mouse ELOVL3 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249791(3-[2-(4-chlorophenyl)-5-methyl-3-oxo-2,3-dihydro-1...)
Affinity DataIC50:  221nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249892(6,6-dimethyl-3-{5-methyl-3-oxo-2-[4-(trifluorometh...)
Affinity DataIC50:  337nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249891(3-[2-(4-methyllphenyl)-5-methyl-3-oxo-2,3-dihydro-...)
Affinity DataIC50:  375nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249815(3-[2-(4-methoxyphenyl)-5-methyl-3-oxo-2,3-dihydro-...)
Affinity DataIC50:  503nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50:  717nMAssay Description:Inhibition of C-terminal V5-epitope-tagged mouse ELOVL3 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50293789(3-endo-(Pyridin-2-ylsulfonyl)-N-[4-(trifluoromethy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse ELOVL3 expressed in Pichia pastoris SND1168More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50249843(3-[2-(4-cyanophenyl)-5-methyl-3-oxo-2,3-dihydro-1H...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human ELOVL3 expressed in african green monkey COS7 cells assessed as stearoyl-CoA elongationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50298968((1R*,4S*,6R*)-(+/-)-2-[(1-Methyl-1H-imidazol-4-yl)...)
Affinity DataIC50:  1.51E+3nMAssay Description:Inhibition of C-terminal V5-epitope-tagged human ELOVL3 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElongation of very long chain fatty acids protein 3(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50293789(3-endo-(Pyridin-2-ylsulfonyl)-N-[4-(trifluoromethy...)
Affinity DataIC50:  6.94E+3nMAssay Description:Inhibition of human ELOVL3 expressed in Pichia pastoris SND1168More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed