Compile Data Set for Download or QSAR
Report error Found 562 Enz. Inhib. hit(s) with Target = 'KiSS-1 receptor'
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50082078BDBM50082078(CHEMBL3422411)
Affinity DataEC50:  0.00600nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50508242BDBM50508242(CHEMBL4539775)
Affinity DataEC50:  0.0220nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392485BDBM50392485(CHEMBL2152055)
Affinity DataEC50:  0.0230nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50508234BDBM50508234(CHEMBL4533110)
Affinity DataEC50:  0.0240nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045514BDBM50045514(CHEMBL3315315)
Affinity DataKi:  0.0260nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045510BDBM50045510(CHEMBL3314227)
Affinity DataKi:  0.0270nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045500BDBM50045500(CHEMBL3314217)
Affinity DataKi:  0.0280nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50508221BDBM50508221(CHEMBL4462883)
Affinity DataEC50:  0.0280nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392490BDBM50392490(CHEMBL2152060)
Affinity DataEC50:  0.0290nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442965BDBM50442965(CHEMBL3086282)
Affinity DataKi:  0.0320nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442966BDBM50442966(CHEMBL3087927)
Affinity DataKi:  0.0330nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045509BDBM50045509(CHEMBL3314226)
Affinity DataKi:  0.0340nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045513BDBM50045513(Kisspeptin-10)
Affinity DataKi:  0.0350nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045507BDBM50045507(CHEMBL3314224)
Affinity DataKi:  0.0360nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045499BDBM50045499(CHEMBL3314216)
Affinity DataKi:  0.0360nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045498BDBM50045498(CHEMBL3314215)
Affinity DataKi:  0.0370nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50508225BDBM50508225(CHEMBL4528114)
Affinity DataEC50:  0.0370nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045512BDBM50045512(CHEMBL3314229)
Affinity DataKi:  0.0380nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 26349BDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataKi:  0.0390nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392486BDBM50392486(CHEMBL2152056)
Affinity DataEC50:  0.0390nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045506BDBM50045506(CHEMBL3314223)
Affinity DataKi:  0.0390nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442968BDBM50442968(CHEMBL3087793)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392402BDBM50392402(CHEMBL2151643)
Affinity DataEC50:  0.0410nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKiSS-1 receptor(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442967BDBM50442967(CHEMBL3087925)
Affinity DataKi:  0.0420nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442966BDBM50442966(CHEMBL3087927)
Affinity DataKi:  0.0430nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442964BDBM50442964(CHEMBL3085809)
Affinity DataKi:  0.0440nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442968BDBM50442968(CHEMBL3087793)
Affinity DataKi:  0.0450nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392401BDBM50392401(CHEMBL2151642)
Affinity DataKi:  0.0460nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 26349BDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataEC50:  0.0490nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392405BDBM50392405(CHEMBL2151646)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKiSS-1 receptor(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442965BDBM50442965(CHEMBL3086282)
Affinity DataKi:  0.0510nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392405BDBM50392405(CHEMBL2151646)
Affinity DataKi:  0.0510nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045517BDBM50045517(CHEMBL3314209)
Affinity DataKi:  0.0520nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442963BDBM50442963(CHEMBL3085804)
Affinity DataKi:  0.0520nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442962BDBM50442962(CHEMBL3087929)
Affinity DataKi:  0.0550nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 26349BDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataKi:  0.0570nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442964BDBM50442964(CHEMBL3085809)
Affinity DataEC50:  0.0570nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50508241BDBM50508241(CHEMBL4451244)
Affinity DataEC50:  0.0580nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetKiSS-1 receptor(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442964BDBM50442964(CHEMBL3085809)
Affinity DataKi:  0.0590nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442967BDBM50442967(CHEMBL3087925)
Affinity DataKi:  0.0620nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045513BDBM50045513(Kisspeptin-10)
Affinity DataKi:  0.0620nMAssay Description:Displacement of [125I]-Kp-10 from human Kiss1 receptor by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 26349BDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataEC50:  0.0650nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392401BDBM50392401(CHEMBL2151642)
Affinity DataEC50:  0.0650nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442982BDBM50442982(CHEMBL3086283)
Affinity DataKi:  0.0650nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392488BDBM50392488(CHEMBL2152058)
Affinity DataEC50:  0.0650nMAssay Description:Agonist activity at human OT7T175 assessed as increase in intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetKiSS-1 receptor(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392405BDBM50392405(CHEMBL2151646)
Affinity DataKi:  0.0680nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50508220BDBM50508220(CHEMBL4541289)
Affinity DataEC50:  0.0680nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetKiSS-1 receptor(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045507BDBM50045507(CHEMBL3314224)
Affinity DataKi:  0.0690nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Human)
Umr7247

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50082074BDBM50082074(CHEMBL3422408)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/1/2016
Entry Details Article
PubMed
TargetKiSS-1 receptor(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50442963BDBM50442963(CHEMBL3085804)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
Displayed 1 to 50 (of 562 total ) | Next | Last >>
Jump to: