Compile Data Set for Download or QSAR
Report error Found 240 Enz. Inhib. hit(s) with Target = 'Serine protease 1/Trypsin-2'
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50131780BDBM50131780((1-Benzhydryl-2-{2-[(5-carbamimidoyl-thiophen-2-yl...)
Affinity DataKi:  0.300nMAssay Description:In vitro inhibition constant (Ki) against human trypsin was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172845BDBM50172845((2-{2-[2-(5-Chloro-2-[1,2,4]triazol-1-yl-benzyl)-o...)
Affinity DataKi:  0.700nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172841BDBM50172841((2-{2-[2-(5-Chloro-2-[1,2,4]triazol-1-yl-benzyl)-o...)
Affinity DataKi:  1.30nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172829BDBM50172829([2-(5-Chloro-2-[1,2,4]triazol-1-yl-benzyl)-oxazolo...)
Affinity DataKi:  1.5nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172831BDBM50172831([2-(5-Chloro-2-[1,2,4]triazol-1-yl-benzyl)-oxazolo...)
Affinity DataKi:  1.5nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172832BDBM50172832(2-(2-{2-[2-(5-Chloro-2-[1,2,4]triazol-1-yl-benzyl)...)
Affinity DataKi:  1.60nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172826BDBM50172826([2-(5-Chloro-2-[1,2,4]triazol-1-yl-benzyl)-oxazolo...)
Affinity DataKi:  1.60nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172830BDBM50172830([2-(5-Chloro-2-[1,2,4]triazol-1-yl-benzyl)-oxazolo...)
Affinity DataKi:  2.90nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096100BDBM50096100(2-(3-Carbamimidoyl-phenyl)-5-trifluoromethyl-2H-py...)
Affinity DataKi:  3.40nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096111BDBM50096111(2-(3-Carbamimidoyl-phenyl)-5-trifluoromethyl-2H-py...)
Affinity DataKi:  3.90nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096097BDBM50096097(2-(3-Carbamimidoyl-phenyl)-5-trifluoromethyl-2H-py...)
Affinity DataKi:  4nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096110BDBM50096110(2-(3-Carbamimidoyl-phenyl)-5-trifluoromethyl-2H-py...)
Affinity DataKi:  4.30nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096099BDBM50096099(2-(3-Carbamimidoyl-phenyl)-5-methyl-2H-pyrazole-3-...)
Affinity DataKi:  4.60nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172847BDBM50172847([2-(5-Chloro-2-[1,2,4]triazol-1-yl-benzyl)-oxazolo...)
Affinity DataKi:  6.90nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096090BDBM50096090(5-Butyl-2-(3-carbamimidoyl-phenyl)-2H-pyrazole-3-c...)
Affinity DataKi:  11nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096091BDBM50096091(2-(3-Carbamimidoyl-phenyl)-5-methyl-2H-pyrazole-3-...)
Affinity DataKi:  13nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096085BDBM50096085(2-(3-Carbamimidoyl-phenyl)-5-methyl-2H-pyrazole-3-...)
Affinity DataKi:  15nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096095BDBM50096095(2-(3-Carbamimidoyl-phenyl)-2H-pyrazole-3-carboxyli...)
Affinity DataKi:  15nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 12751BDBM12751(CHEMBL152854 | 1-(3-carbamimidoylphenyl)-3-methyl-...)
Affinity DataKi:  16nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172853BDBM50172853([2-(3-Chloro-benzyl)-oxazolo[4,5-c]pyridin-4-yl]-(...)
Affinity DataKi:  16nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172853BDBM50172853([2-(3-Chloro-benzyl)-oxazolo[4,5-c]pyridin-4-yl]-(...)
Affinity DataKi:  16nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096098BDBM50096098(2-(3-Carbamimidoyl-phenyl)-5-methyl-2H-pyrazole-3-...)
Affinity DataKi:  17nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172835BDBM50172835((2,2-Difluoro-2-piperidin-2-yl-ethyl)-[2-(2-tetraz...)
Affinity DataKi:  17nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096105BDBM50096105(2-(3-Carbamimidoyl-phenyl)-5-trifluoromethyl-2H-py...)
Affinity DataKi:  20nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50087533BDBM50087533(CHEMBL140072 | CHEMBL153611 | 3-(3-Carbamimidoyl-p...)
Affinity DataKi:  21nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172848BDBM50172848((2-Piperidin-2-yl-ethyl)-[2-(2-tetrazol-1-yl-benzy...)
Affinity DataKi:  23nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096102BDBM50096102(4-Bromo-1-(3-carbamimidoyl-phenyl)-1H-pyrrole-2-ca...)
Affinity DataKi:  32nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172827BDBM50172827([2-(3-Chloro-benzyl)-oxazolo[4,5-c]pyridin-4-yl]-(...)
Affinity DataKi:  44nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096094BDBM50096094(2-(3-Carbamimidoyl-phenyl)-5-methyl-2H-pyrazole-3-...)
Affinity DataKi:  49nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112086BDBM50112086(CHEMBL48361 | 3-({2-[(4-Carbamimidoyl-phenylamino)...)
Affinity DataKi:  50.3nMAssay Description:Inhibitory constant (Ki) was determined against human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096104BDBM50096104(2-(3-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  53nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096084BDBM50096084(1-(3-Carbamimidoyl-phenyl)-1H-pyrrole-2-carboxylic...)
Affinity DataKi:  56nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096108BDBM50096108(2-(3-Carbamimidoyl-phenyl)-5-trifluoromethyl-2H-py...)
Affinity DataKi:  59nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096101BDBM50096101(2-(3-Carbamimidoyl-phenyl)-5-methyl-2H-pyrazole-3-...)
Affinity DataKi:  59nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 12657BDBM12657(CHEMBL559015 | 1-[3-(Aminomethyl)phenyl]-N-[3-fluo...)
Affinity DataKi:  60nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50068493BDBM50068493((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  80nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50172843BDBM50172843((2,2-Difluoro-2-piperidin-2-yl-ethyl)-[2-(2-[1,2,4...)
Affinity DataKi:  86nMAssay Description:Inhibitory constant against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096103BDBM50096103(2-(3-Carbamimidoyl-phenyl)-5-methyl-2H-pyrazole-3-...)
Affinity DataKi:  87nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096113BDBM50096113(2-(3-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  100nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096088BDBM50096088(2-(3-Carbamimidoyl-phenyl)-5-methyl-2H-pyrazole-3-...)
Affinity DataKi:  100nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096086BDBM50096086(2-(3-Aminomethyl-phenyl)-5-methyl-2H-pyrazole-3-ca...)
Affinity DataKi:  120nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096089BDBM50096089(2-(3-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  120nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102780BDBM50102780(3-{5-[AMINO(IMINIO)METHYL]-1H-INDOL-2-YL}-1,1'-BIP...)
Affinity DataKi:  130nMAssay Description:The compound was tested for inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096093BDBM50096093(2-(3-Aminomethyl-phenyl)-5-methyl-2H-pyrazole-3-ca...)
Affinity DataKi:  130nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096112BDBM50096112(2-(3-Carbamimidoyl-phenyl)-5-methyl-2H-pyrazole-3-...)
Affinity DataKi:  150nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50068490BDBM50068490([4-(1-Carbamimidoyl-piperidin-4-yloxy)-phenyl]-(2-...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50068487BDBM50068487([4-(1-Carbamimidoyl-piperidin-4-yloxy)-phenyl]-(2-...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50068501BDBM50068501((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50068485BDBM50068485((2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-7-...)
Affinity DataKi:  200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2012
Entry Details Article
PubMed
TargetSerine protease 1/Trypsin-2(Human)
Lg Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096109BDBM50096109(2-(3-Aminomethyl-phenyl)-5-methyl-2H-pyrazole-3-ca...)
Affinity DataKi:  220nMAssay Description:In vitro activity against human trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
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