Compile Data Set for Download or QSAR
Report error Found 242 Enz. Inhib. hit(s) with Target = 'Transcription activator BRG1 [1448-1575]'
TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394450BDBM394450(US10308614, Example 51 | 2-(6-amino-5-(8-(5-)
Affinity DataIC50: 3.40nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394468BDBM394468(US10308614, Example 69 | 2-(6-amino-5-(8-)
Affinity DataIC50: 3.90nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394474BDBM394474(US10308614, Example 75 | 2-(6-amino-5-(8-(5-)
Affinity DataIC50: 4nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394469BDBM394469(US10308614, Example 70 | 2-(6-amino-5-(8-(pyridin-)
Affinity DataIC50: 4.10nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394462BDBM394462(US10308614, Example 63 | 2-(6-amino-5-(8-phenyl-3,...)
Affinity DataIC50: 4.30nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394446BDBM394446(US10308614, Example 47 | 2-(6-amino-5-(8-(2-)
Affinity DataIC50: 4.5nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394470BDBM394470(US10308614, Example 71 | 2-(6-amino-5-(8-)
Affinity DataIC50: 5nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394589BDBM394589(US10308614, Example 192 | 2-(6-amino-5-(1-(1-)
Affinity DataIC50: 6.30nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394476BDBM394476(US10308614, Example 77 | 2-(6-amino-5-(8-(thiazol-)
Affinity DataIC50: 6.5nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394585BDBM394585(US10308614, Example 188 | 2-(6-amino-5-(1-(1-)
Affinity DataIC50: 6.60nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394475BDBM394475(US10308614, Example 76 | 2-(6-amino-5-(8-(4-)
Affinity DataIC50: 6.70nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394427BDBM394427(US10308614, Example 28 | US10308614, Example 84 | ...)
Affinity DataIC50: 8.40nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394528BDBM394528(US10308614, Example 129 | 1-(4-(3-amino-6-(2-)
Affinity DataIC50: 10.4nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394449BDBM394449(US10308614, Example 50 | 2-(6-amino-5-(8-)
Affinity DataIC50: 10.6nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394473BDBM394473(US10308614, Example 74 | 2-(6-amino-5-((1R,4R)-5-)
Affinity DataIC50: 10.6nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394485BDBM394485(US10308614, Example 85 | Enantiomer 1 and Enantiom...)
Affinity DataIC50: 11nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394441BDBM394441(US10308614, Example 42 | 1-(3-amino-6-(2-)
Affinity DataIC50: 11.3nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394461BDBM394461(US10308614, Example 62 | (4-(3-amino-6-(2-)
Affinity DataIC50: 11.7nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394595BDBM394595(US10308614, Example 198 | 2-(6-amino-5-(trans-2-ph...)
Affinity DataIC50: 12.1nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394575BDBM394575(US10308614, Example 178 | 2-(6-amino-5-(2-)
Affinity DataIC50: 12.2nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394537BDBM394537(US10308614, Example 138 | (4-(3-amino-6-(2-)
Affinity DataIC50: 12.6nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394584BDBM394584(US10308614, Example 187 | 2-(6-amino-5-(1-methyl-)
Affinity DataIC50: 12.8nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394605BDBM394605(US10308614, Example 209 | 2-(6-amino-5-cyclohexylp...)
Affinity DataIC50: 14.5nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394571BDBM394571(US10308614, Example 174 | 2-(6-amino-5-)
Affinity DataIC50: 14.8nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394458BDBM394458(US10308614, Example 59 | 1-(3-amino-6-(2-)
Affinity DataIC50: 15.8nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394427BDBM394427(US10308614, Example 28 | US10308614, Example 84 | ...)
Affinity DataIC50: 17.2nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394580BDBM394580(US10308614, Example 183 | 2-(6-amino-5-((1-)
Affinity DataIC50: 17.2nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394424BDBM394424(US10308614, Example 25 | 2-(6-amino-5-(4-methyl-)
Affinity DataIC50: 17.6nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394508BDBM394508(US10308614, Example 109 | 2-(6-amino-5-(3-methyl-)
Affinity DataIC50: 17.6nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394587BDBM394587(US10308614, Example 190 | 2-(6-amino-5-)
Affinity DataIC50: 17.6nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394456BDBM394456(US10308614, Example 57 | 2-(6-amino-5-(3-)
Affinity DataIC50: 17.7nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394492BDBM394492(US10308614, Example 92 | (S)-2-(6-amino-5-(3-methy...)
Affinity DataIC50: 18.5nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394621BDBM394621(US10308614, Example 225 | 2-(6-amino-5-((1,4-trans...)
Affinity DataIC50: 19nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394481BDBM394481(US10308614, Example 81 | Enantiomer 1 and Enantiom...)
Affinity DataIC50: 19.1nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394442BDBM394442(US10308614, Example 43 | 2-(6-amino-5-(8-)
Affinity DataIC50: 19.3nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394510BDBM394510(US10308614, Example 111 | 2-(6-amino-5-(4-)
Affinity DataIC50: 19.7nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394525BDBM394525(US10308614, Example 126 | (3-(3-amino-6-(2-)
Affinity DataIC50: 20.3nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394619BDBM394619(US10308614, Example 223 | 2-(6-amino-5-(1-benzyl-1...)
Affinity DataIC50: 20.5nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394542BDBM394542(US10308614, Example 143 | (4-(3-amino-6-(2-)
Affinity DataIC50: 20.6nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394430BDBM394430(US10308614, Example 31 | 1-(3-amino-6-(2-)
Affinity DataIC50: 20.8nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394414BDBM394414(US10308614, Example 15 | 2-(6-amino-5-(4-(1-)
Affinity DataIC50: 20.9nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394622BDBM394622(US10308614, Example 226 | 2-(6-amino-5-((1,4-trans...)
Affinity DataIC50: 20.9nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394399BDBM394399(US10308614, Example 1 | tert-butyl 4-(3-amino-6-(2...)
Affinity DataIC50: 21.4nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394592BDBM394592(US10308614, Example 195 | (2R)-2-[4-[3-amino- 6-(2...)
Affinity DataIC50: 21.7nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394509BDBM394509(US10308614, Example 110 | 2-(6-amino-5-(4-)
Affinity DataIC50: 21.9nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394586BDBM394586(US10308614, Example 189 | 2-(6-amino-5-(4-)
Affinity DataIC50: 22.2nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394520BDBM394520(US10308614, Example 121 | 3-(3-amino-6-(2-hydroxyp...)
Affinity DataIC50: 22.5nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394493BDBM394493(US10308614, Example 93 | (R)-2-(6-amino-5- (3-meth...)
Affinity DataIC50: 23.8nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394606BDBM394606(US10308614, Example 210 | 2-(6-amino-5-)
Affinity DataIC50: 23.9nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetTranscription activator BRG1 [1448-1575](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 394591BDBM394591(US10308614, Example 194 | 2-(4-(3-amino-6-(2-)
Affinity DataIC50: 24.7nMAssay Description:His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvprgsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNAQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

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