973 SMILES Strings for Guanylate cyclase soluble subunit alpha-1

Compound Name
SMILES String
C(c1cncnc1)n1nc(cc1-c1ccon1)-c1ncccn1
CC(=C)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(=O)NCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(=O)NNC(=O)C1(C)C(=O)Nc2nc(nc(N)c12)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(=O)NS(=O)(=O)C1CCN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(=O)NS(=O)(=O)CCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(=O)Nc1cnc(nc1N)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
CC(=O)OC(C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)c1ccccc1
CC(=O)OCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(=O)OCC(=O)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(=O)O[C@@H](C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F |r|
CC(=O)c1cc(nn1Cc1ccccc1F)-c1ncc(F)c(NC(CO)CO)n1
CC(=O)c1cc(nn1Cc1ccccc1F)-c1ncc(F)c(NCC(O)(C(F)(F)F)C(F)(F)F)n1
CC(=O)c1cc(nn1Cc1ccccc1F)-c1ncc(F)c(O)n1
CC(C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)S(C)(=O)=O
CC(C(=O)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)S(C)(=O)=O
CC(C(C1CC1)c1ccc(Cl)c(NC(=O)C([C@@H](C)C(F)(F)F)c2ccc(Cl)cc2)c1)C(O)=O |r|
CC(C)(C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)S(C)(=O)=O
CC(C)(C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)c1ccccc1
CC(C)(C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)n1cncn1
CC(C)(C(=O)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)S(C)(=O)=O
CC(C)(C(O)=O)n1cc(nn1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12
CC(C)(C(O)=O)n1cc(nn1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12
CC(C)(C)C(=O)Nc1cnc(nc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)C(=O)Nc1cnc(nc1N)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
CC(C)(C)CC(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)CCCn1nc(-c2nc3NC(=O)[C@](C)(c3c(N)n2)c2ccc(CCC(O)=O)cc2)c2ccc(Cl)cc12 |r|
CC(C)(C)CCn1nc(-c2nc3NC(=O)C(C)(c4nc(CC(C)(C)C(O)=O)co4)c3c(N)n2)c2ccc(Cl)cc12
CC(C)(C)CCn1nc(-c2nc3NC(=O)[C@](C)(c3c(N)n2)c2ccc(CCC(O)=O)cc2)c2cccnc12 |r|
CC(C)(C)NC(=O)c1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)OC(=O)N1CC(O)(CNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)C1
CC(C)(C)OC(=O)N1CCN(C(C1)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)OC(=O)NC1CCN(C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)OC(=O)NCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)OC(=O)NCCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)OC(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)OC(=O)Nc1cnc(nc1N)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
CC(C)(C)OC(=O)n1c2cnc(nc2[nH]c1=O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)S(=O)(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)S(=O)Nc1cnc(nc1NS(=O)C(C)(C)C)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C)c1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(C=C)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(CC(O)=O)c1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12 |r|
CC(C)(CCc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2cc(Cl)ccc12)C(O)=O
CC(C)(CCc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2cc(F)ccc12)C(O)=O
CC(C)(CCc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(CCc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(F)ccc12)C(O)=O
CC(C)(CCc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ccccc12)C(O)=O
CC(C)(CCc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)C(O)=O
CC(C)(CCc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ncccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(CCc1csc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2cc(F)ccc12)C(O)=O
CC(C)(CCc1csc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(CCc1csc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ccccc12)C(O)=O
CC(C)(CCl)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(CO)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(Cc1ccc(cc1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1ccc(cc1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)C(O)=O
CC(C)(Cc1ccc(cc1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1ccc(cc1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2ncccc12)C(O)=O
CC(C)(Cc1ccc(nc1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1cccc(c1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1cccc(c1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCC2)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCC2)c2ncccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCC2)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCC2)c2cc(F)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCC2)c2ccccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCC2)c2ncccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCO2)c2cc(F)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCO2)c2ccccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCO2)c2ncccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2c(F)ccc(F)c2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2c(F)cccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccc(F)cc2)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccc(F)cc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2cc(F)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2ccccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2ncccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2F)c2cc(F)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1nn[nH]n1
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ccccc12)c1nn[nH]n1
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ncccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C2CC2)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1coc(n1)C1(C2CC2)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(F)ccc12)C(O)=O
CC(C)(Cc1csc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncc(F)cc12)C(O)=O
CC(C)(Cc1csc(n1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)F)c2ncc(F)cc12)C(O)=O
CC(C)(Cc1csc(n1)C1(C2CC2)C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2cnc(F)cc12)C(O)=O
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCC2)c2cc(Cl)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCC2)c2ncccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCC2)c2cc(F)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCC2)c2ncccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCO2)c2cc(F)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCO2)c2ccccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCO2)c2ncccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)C(=O)NO |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2nc(Cl)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2ncccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2c(F)ccc(F)c2F)c2cc(Cl)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2c(F)ccc(F)c2F)c2ccccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2c(F)cccc2F)c2cc(Cl)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccc(F)cc2)c2cc(Cl)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccc(F)cc2F)c2cc(Cl)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2cc(F)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2ccccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2ncccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2F)c2cc(Cl)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2F)c2cc(F)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1nn[nH]n1 |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(F)ccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ccccc12)c1nn[nH]n1 |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncc(F)cc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)C(O)=O |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1nn[nH]n1 |r|
CC(C)(Cc1csc(n1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ncccc2F)c2cc(Cl)ccc12)C(O)=O |r|
CC(C)(Cc1nc(co1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cc1nc(cs1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cn1cc(cn1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)C(O)=O
CC(C)(Cn1cc(cn1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cn1cc(cn1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(F)ccc12)C(O)=O
CC(C)(Cn1cc(cn1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)C(O)=O
CC(C)(Cn1cc(nn1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)C(O)=O
CC(C)(Cn1cc(nn1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)C(O)=O
CC(C)(F)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(NC(=O)CCc1ccc(cc1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)C(O)=O |r|
CC(C)(O)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(O)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(O)c1cnc(nc1O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)(Oc1ccccc1)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)C(C)(CC(O)=O)c1ccc(Cl)c(NC(=O)[C@@H]([C@@H](C)C(F)(F)F)c2ccc(Cl)cc2)c1 |r|
CC(C)C(CC(O)=O)c1ccc(Cl)c(NC(=O)C(C(C)C(F)(F)F)c2ccc(CC(F)(F)F)cc2)c1
CC(C)C(CC(O)=O)c1ccc(Cl)c(NC(=O)[C@@H]([C@@H](C)C(F)(F)F)c2ccc(Cl)cc2)c1 |r|
CC(C)C(CC(O)=O)c1ccc(Cl)c(NC(=O)[C@@H]([C@@H](C)C(F)(F)F)c2ccc(Cl)cc2)c1 |r|
CC(C)C(CC(O)=O)c1ccc(Cl)c(NC(=O)[C@@H]([C@@H](C)C(F)(F)F)c2ccc(cc2)C(C)(C)C)c1 |r|
CC(C)C(CC(O)=O)c1ccc(Cl)c(NC(=O)[C@@H]([C@@H](C)C(F)(F)F)c2ccc(cc2)C(C)C)c1 |r|
CC(C)C(CC(O)=O)c1ccc(Cl)c(NC(=O)[C@@H]([C@@H](C)C(F)(F)F)c2ccc(cc2)C2CC2(F)F)c1 |r|
CC(C)C(Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(=O)NC1CC1
CC(C)C1(CCN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O
CC(C)CCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1cc(O)c(Cl)c(F)c1
CC(C)CCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1cc(O)c(Cl)cn1
CC(C)CCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(Cl)c(O)c1
CC(C)CCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(F)c(O)c1
CC(C)CCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(O)c(F)c1
CC(C)CCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(O)cc1
CC(C)CCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(c(O)c1)C(F)(F)F
CC(C)CCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1cccc(O)c1
CC(C)CCc1nc(cn2ncnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1cc(O)ccn1
CC(C)COC(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)C[C@@H](N(C)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O |r|
CC(C)C[C@H](Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O |r|
CC(C)N(CC(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)N(C[C@H](O)CO)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
CC(C)NC(=O)NCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)S(=O)(=O)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(C)[C@@H](N(C)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O |r|
CC(C)[C@@H](Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(N)=O |r|
CC(C)[C@H](CN(C)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)NS(=O)(=O)C1CC1 |r|
CC(C)[C@H](N(C)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(=O)NS(=O)(=O)C1CC1 |r|
CC(C)[C@H](N(C)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O |r|
CC(C)[C@H](N(C)c1nc(ncc1F)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1)C(O)=O |r|
CC(C)[C@H](N(C)c1nc(ncc1F)-c1nc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O |r|
CC(C)[C@H](Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(=O)NS(=O)(=O)C1CC1 |r|
CC(C)[C@H](Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(N)=O |r|
CC(C)[C@H](Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O |r|
CC(CCO)(C(=O)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)S(C)(=O)=O
CC(Cc1ccc(cc1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)C(O)=O
CC(Cc1ccc(cc1)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2ncccc12)C(O)=O
CC(F)(F)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(NS(=O)(=O)c1ccc(C)cc1)C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC(O)(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
CC(O)(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(N)=O
CC(O)CN(CC(C)O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(C(=O)NC2CC2)C(=O)Nc2nc(nc(N)c12)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2c(N)cnc2c(Cc2cccc(F)c2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCC(F)(F)CC2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCC2)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1cc(Cl)c(O)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1cc(O)c(C#N)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1cc(O)c(C#N)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1cc(O)c(Cl)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1cc(O)c(c(F)c1)C(F)(F)F
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1cc(O)c(cn1)C(F)(F)F
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1ccc(Cl)c(O)c1Cl
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1ccc(Cl)c(O)n1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1ccc(O)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CC2CCCCC2)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(Cl)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(F)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(O)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC(F)(F)C(F)(F)F)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC2CCCCC2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC2CCCCC2)n1)c1ccc(F)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC2CCCCC2)n1)c1ccc(O)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC2CCCCC2)n1)c1ccc(O)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC2CCCCC2)n1)c1ccc(O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCC2CCCCC2)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(CCCC(F)(F)F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2c(F)cccc2F)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2c(F)cccc2F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2)n1)c1cc(O)c(C#N)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2)n1)c1cc(O)c(Cl)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2)n1)c1ccc(F)c(Cl)c1O
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2)n1)c1ccc(c(O)c1)C(F)(F)F
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2)n1)c1ncc(Cl)c(O)c1Cl
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2)n1)c1nccc(O)c1Cl
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2F)n1)c1cc(O)c(C#N)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2F)n1)c1cc(O)c(Cl)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2F)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)cc(F)c2F)n1)c1ccc(c(O)c1)C(F)(F)F
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)ccc2F)n1)c1cc(O)c(C#N)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)ccc2F)n1)c1cc(O)c(Cl)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)ccc2F)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)ccc2F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cc(F)ccc2F)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(Cl)cc2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(Cl)cc2)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)c(F)c2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1)c1ccc(F)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1)c1ccc(O)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1)c1ccc(O)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1)c1ccc(O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2F)n1)c1ccc(F)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2F)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(Cl)c2)n1)c1ccc(O)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(Cl)c2)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1)c1cc(O)c(C#N)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1)c1cc(O)c(Cl)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1)c1cc(O)c(cn1)C(F)(F)F
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1)c1ccc(O)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1)c1ccc(O)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1)c1ccc(c(O)c1)C(F)(F)F
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2)n1)c1ccc(O)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1cc(Cl)c(O)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1cc(O)c(C#N)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1cc(O)c(C#N)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1cc(O)c(Cl)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1cc(O)c(F)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1cc(O)c(cn1)C(F)(F)F
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1ccc(F)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1ccc(O)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1ccc(O)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2ccccc2F)n1)c1ccc(c(O)c1)C(F)(F)F
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CC2CCCCC2)n1)c1cc(Cl)c(O)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CC2CCCCC2)n1)c1cc(O)c(C#N)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CC2CCCCC2)n1)c1cc(O)c(C#N)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CC2CCCCC2)n1)c1cc(O)c(Cl)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CC2CCCCC2)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CC2CCCCC2)n1)c1cc(O)ccn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CC2CCCCC2)n1)c1ccc(Cl)c(O)c1Cl
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(F)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(O)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CCC(F)(F)C(F)(F)F)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CCCC(F)(F)F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(CCCCF)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(Cc2cc(F)cc(F)c2)n1)c1cc(O)c(C#N)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(Cc2ccc(F)cc2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(Cc2ccc(F)cc2)n1)c1ccc(O)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(Cc2ccc(F)cc2)n1)c1ccc(O)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(Cc2cccc(F)c2)n1)c1cc(O)ccn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(Cc2ccccc2F)n1)c1cc(O)c(C#N)c(Cl)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(Cc2ccccc2F)n1)c1cc(O)c(Cl)c(F)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1cn2ncnc2c(Cc2ccccc2F)n1)c1cc(O)c(Cl)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)c(Br)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)c(O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)c(c1)[N+]#[C-]
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1ccc(\C=C\C(O)=O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1ccc(cc1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1cccc(c1)-c1nn[nH]n1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1cccc(c1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1cn(CC(O)=O)nn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1cn(CC2(CC2)C(O)=O)nn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1cn(CCC(O)=O)nn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1nc(cs1)-c1ccc(cc1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1nc(cs1)-c1cccc(c1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1nn(CC(O)=O)c(=O)o1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)c1ccc(CC(O)=O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)c1ccc(CCCC(O)=O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)c1cccc(c1)-c1nn[nH]n1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)c1cn(CCC(O)=O)nn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)c1cnn(CCC(O)=O)n1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)c1nc(CC(O)=O)cs1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2cc(F)ccc12)c1nc(CCC(F)(F)C(O)=O)co1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1cc(ccn1)-c1nn[nH]n1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1cc(ccn1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(CCP(O)(O)=O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(CCS(O)(=O)=O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(CCc2nn[nH]n2)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(Cc2nn[nH]n2)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(OCC(O)=O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(\C=C\C(O)=O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(cc1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(cn1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1cccc(c1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1cccc(n1)-c1nn[nH]n1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1cccc(n1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccnc(c1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1nc(CCC(F)(F)C(O)=O)co1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1nc(CCC(O)=O)c[nH]1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1nc(C[C@@H](N)C(O)=O)co1 |r|
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1nc(co1)-c1ccc(cc1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1nc(cs1)-c1ccc(cc1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1nc2cc(ccc2o1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1nc2cc(ccc2s1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(F)ccc12)c1ccc(cc1)-c1nn[nH]n1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(F)ccc12)c1cccc(CCC(O)=O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(F)ccc12)c1cccc(c1)-c1nn[nH]n1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(F)ccc12)c1cccc(c1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ccccc12)c1ccc(CCc2nn[nH]n2)cn1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1ccc(CC(O)=O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1ccc(\C=C\C(O)=O)cc1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1cccc(CCC(O)=O)c1
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1nc(co1)-c1ccc(cc1)C(O)=O
CC1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1nc(cs1)-c1ccc(cc1)C(O)=O
CC1(C(=O)Nc2nc(nc(N3CC(O)(C3)C(F)(F)F)c12)-c1cn2ccnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(F)c(O)c1
CC1(C(=O)Nc2nc(nc(N3CC(O)(C3)C(F)(F)F)c12)-c1cn2ccnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(O)c(F)c1
CC1(C(=O)Nc2nc(nc(N3CCC(CC3)C(F)(F)F)c12)-c1cn2ncnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N3CCC(F)(F)CC3)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(N3CCC(F)(F)CC3)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1)c1cccc(O)c1
CC1(C(=O)Nc2nc(nc(NCC(O)C(F)(F)F)c12)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(NCC(O)C(F)(F)F)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(NCC(O)C(F)(F)F)c12)-c1cn2ncnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(NCCC(F)(F)F)c12)-c1cn2ncnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(Cl)c(O)c1
CC1(C(=O)Nc2nc(nc(NCCCC(F)(F)F)c12)-c1cn2ncnc2c(CCC(F)(F)C(F)(F)F)n1)c1ccc(Cl)c(O)c1
CC1(C(N)=O)C(=O)Nc2nc(nc(N)c12)-c1cc(-c2ccon2)n(CCC(F)(F)F)n1
CC1(C(N)=O)C(=O)Nc2nc(nc(N)c12)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(C)CCC(=O)N1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(C)CCC(N(C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O
CC1(C)CCN(C1=O)c1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(C2CCC(CCC(O)=O)CC2)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12 |(1.04,3.13,;1.44,1.64,;2.53,2.73,;4.02,2.33,;5.11,3.42,;4.71,4.91,;5.8,6,;7.28,5.6,;8.37,6.69,;9.86,6.29,;7.97,8.18,;3.22,5.31,;2.13,4.22,;2.35,.4,;3.89,.4,;1.44,-.85,;-.02,-.37,;-1.36,-1.14,;-2.69,-.37,;-2.69,1.17,;-1.36,1.94,;-1.36,3.48,;-.02,1.17,;-4.03,-1.14,;-4.27,-2.67,;-5.79,-2.91,;-6.34,-4.34,;-5.37,-5.54,;-5.92,-6.98,;-4.95,-8.18,;-3.43,-7.93,;-2.88,-6.5,;-3.85,-5.3,;-3.3,-3.86,;-6.49,-1.53,;-7.97,-1.14,;-8.37,.35,;-9.86,.75,;-7.28,1.44,;-5.8,1.04,;-5.4,-.45,)|
CC1(C2CCC(CCC(O)=O)CC2)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12 |(1.13,3.2,;1.53,1.71,;2.62,2.8,;4.11,2.4,;5.2,3.49,;4.8,4.98,;5.89,6.07,;7.37,5.67,;8.46,6.76,;9.95,6.36,;8.06,8.24,;3.31,5.38,;2.22,4.29,;2.44,.46,;3.98,.46,;1.53,-.78,;.07,-.31,;-1.27,-1.08,;-2.6,-.31,;-2.6,1.23,;-1.27,2,;-1.27,3.54,;.07,1.23,;-3.93,-1.08,;-3.93,-2.62,;-5.4,-3.09,;-5.8,-4.58,;-4.71,-5.67,;-5.11,-7.16,;-4.02,-8.24,;-2.53,-7.85,;-2.13,-6.36,;-3.22,-5.27,;-2.82,-3.78,;-6.3,-1.85,;-7.84,-1.68,;-8.46,-.28,;-9.95,.12,;-7.56,.97,;-6.03,.81,;-5.4,-.6,)|
CC1(CC1(Cl)Cl)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(CC1(F)F)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(CC1)C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(CC1)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(CC1)C(=O)Nc1cnc(nc1O)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
CC1(CCCCC1)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(CCCN(C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O
CC1(CCCO1)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(CCN(C1=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(=O)NC1CC1
CC1(CCN(C1=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(N)=O
CC1(CCN(C1=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O
CC1(CCN(C1=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)S(C)(=O)=O
CC1(Cc2ccccc2S1(=O)=O)C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1(N2CCC(CCC(O)=O)C2)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12
CC1(N2CCC(CCC(O)=O)CC2)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12
CC1CCC(Cc2nc(cn3ccnc23)-c2nc3NC(=O)C(C)(c3c(N)n2)c2ccc(Cl)c(O)c2)CC1 |(1.01,-6.29,;-.33,-5.52,;-1.66,-6.29,;-2.99,-5.52,;-2.99,-3.98,;-4.33,-3.21,;-4.33,-1.67,;-2.99,-.9,;-2.99,.64,;-4.33,1.41,;-5.66,.64,;-7.13,1.12,;-8.03,-.13,;-7.13,-1.37,;-5.66,-.9,;-1.66,1.41,;-.33,.64,;1.01,1.41,;2.47,.94,;3.38,2.18,;4.92,2.18,;2.47,3.43,;2.07,4.91,;1.01,2.95,;-.33,3.72,;-.33,5.26,;-1.66,2.95,;3.86,4.09,;3.98,5.63,;5.37,6.29,;6.64,5.42,;8.03,6.08,;6.52,3.88,;7.79,3.01,;5.13,3.22,;-1.66,-3.21,;-.33,-3.98,)|
CC1CCC(Cc2nc(cn3ccnc23)-c2nc3NC(=O)C(C)(c3c(N)n2)c2ccc(Cl)c(O)c2)CC1 |(1.21,-7.04,;-.12,-6.27,;-1.46,-7.04,;-2.79,-6.27,;-2.79,-4.73,;-4.12,-3.96,;-4.12,-2.42,;-2.79,-1.65,;-2.79,-.11,;-4.12,.66,;-5.46,-.11,;-6.92,.37,;-7.83,-.88,;-6.92,-2.12,;-5.46,-1.65,;-1.46,.66,;-.12,-.11,;1.21,.66,;2.67,.19,;3.58,1.43,;5.12,1.43,;2.67,2.68,;2.28,4.17,;1.21,2.2,;-.12,2.97,;-.12,4.51,;-1.46,2.2,;3.76,3.77,;3.37,5.26,;4.45,6.35,;5.94,5.95,;7.03,7.04,;6.34,4.46,;7.83,4.06,;5.25,3.37,;-1.46,-3.96,;-.12,-4.73,)|
CC1CCC(Cc2nc(cn3ccnc23)-c2nc3NC(=O)C(C)(c3c(N)n2)c2ccc(O)c(Cl)c2)CC1 |(1.21,-7.04,;-.12,-6.27,;-1.46,-7.04,;-2.79,-6.27,;-2.79,-4.73,;-4.12,-3.96,;-4.12,-2.42,;-2.79,-1.65,;-2.79,-.11,;-4.12,.66,;-5.46,-.11,;-6.92,.37,;-7.83,-.88,;-6.92,-2.12,;-5.46,-1.65,;-1.46,.66,;-.12,-.11,;1.21,.66,;2.67,.19,;3.58,1.43,;5.12,1.43,;2.67,2.68,;2.28,4.17,;1.21,2.2,;-.12,2.97,;-.12,4.51,;-1.46,2.2,;3.76,3.77,;3.37,5.26,;4.45,6.35,;5.94,5.95,;7.03,7.04,;6.34,4.46,;7.83,4.06,;5.25,3.37,;-1.46,-3.96,;-.12,-4.73,)|
CC1CCC(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3ccc(Cl)cc23)CC1 |(-1.39,-7.53,;-2.48,-6.44,;-3.97,-6.84,;-5.06,-5.75,;-4.66,-4.26,;-5.75,-3.17,;-5.35,-1.69,;-3.89,-1.21,;-3.89,.33,;-2.55,1.1,;-1.22,.33,;.11,1.1,;1.58,.62,;2.48,1.87,;4.02,1.87,;1.58,3.12,;.81,4.45,;2.91,3.89,;4.38,3.41,;5.28,4.66,;6.82,4.66,;7.59,5.99,;7.59,7.53,;6.26,6.76,;9.13,5.99,;9.9,7.32,;9.9,4.66,;4.38,5.9,;2.91,5.43,;.11,2.64,;-1.22,3.41,;-1.22,4.95,;-2.55,2.64,;-5.35,.81,;-5.98,2.21,;-7.51,2.37,;-8.41,1.13,;-9.9,1.53,;-7.79,-.28,;-6.26,-.44,;-3.17,-3.86,;-2.08,-4.95,)|
CC1CCC(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3ccc(F)cc23)CC1 |(-1.39,-7.53,;-2.48,-6.44,;-3.97,-6.84,;-5.06,-5.75,;-4.66,-4.26,;-5.75,-3.17,;-5.35,-1.69,;-3.89,-1.21,;-3.89,.33,;-2.55,1.1,;-1.22,.33,;.11,1.1,;1.58,.62,;2.48,1.87,;4.02,1.87,;1.58,3.12,;.81,4.45,;2.91,3.89,;4.38,3.41,;5.28,4.66,;6.82,4.66,;7.59,5.99,;7.59,7.53,;6.26,6.76,;9.13,5.99,;9.9,7.32,;9.9,4.66,;4.38,5.9,;2.91,5.43,;.11,2.64,;-1.22,3.41,;-1.22,4.95,;-2.55,2.64,;-5.35,.81,;-5.98,2.21,;-7.51,2.37,;-8.41,1.13,;-9.9,1.53,;-7.79,-.28,;-6.26,-.44,;-3.17,-3.86,;-2.08,-4.95,)|
CC1CCC(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3ccccc23)CC1 |(-2.06,-7.98,;-3.15,-6.89,;-4.64,-7.29,;-5.72,-6.2,;-5.33,-4.71,;-6.42,-3.62,;-6.02,-2.14,;-4.55,-1.66,;-4.55,-.12,;-3.22,.65,;-1.88,-.12,;-.55,.65,;.91,.17,;1.82,1.42,;3.36,1.42,;.91,2.67,;.52,4.15,;2.25,3.44,;3.71,2.96,;4.62,4.21,;6.1,4.61,;6.5,6.09,;5.02,6.49,;6.1,7.58,;7.99,6.49,;9.08,5.4,;8.39,7.98,;3.71,5.45,;2.25,4.98,;-.55,2.19,;-1.88,2.96,;-1.88,4.5,;-3.22,2.19,;-6.02,.36,;-6.64,1.76,;-8.17,1.92,;-9.08,.68,;-8.45,-.73,;-6.92,-.89,;-3.84,-4.31,;-2.75,-5.4,)|
CC1CCC(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3cccnc23)CC1 |(-2.14,-7.53,;-3.23,-6.44,;-4.71,-6.84,;-5.8,-5.75,;-5.4,-4.26,;-6.49,-3.17,;-6.1,-1.69,;-4.63,-1.21,;-4.63,.33,;-3.3,1.1,;-1.96,.33,;-.63,1.1,;.83,.62,;1.74,1.87,;3.28,1.87,;.83,3.12,;.06,4.45,;2.17,3.89,;3.63,3.41,;4.54,4.66,;6.08,4.66,;6.85,5.99,;6.85,7.53,;5.51,6.76,;8.39,5.99,;9.16,7.32,;9.16,4.66,;3.63,5.9,;2.17,5.43,;-.63,2.64,;-1.96,3.41,;-1.96,4.95,;-3.3,2.64,;-6.1,.81,;-6.72,2.21,;-8.25,2.37,;-9.16,1.13,;-8.53,-.28,;-7,-.44,;-3.92,-3.86,;-2.83,-4.95,)|
CC1CCC(Cn2nc(-c3nc4NC(=O)[C@@](C)(c5nc(CC(C)(C)C(O)=O)cs5)c4c(N)n3)c3ccc(F)cc23)CC1 |r,wU:15.15,(-1.39,-7.53,;-2.48,-6.44,;-3.97,-6.84,;-5.06,-5.75,;-4.66,-4.26,;-5.75,-3.17,;-5.35,-1.69,;-3.89,-1.21,;-3.89,.33,;-2.55,1.1,;-1.22,.33,;.11,1.1,;1.58,.62,;2.48,1.87,;4.02,1.87,;1.58,3.12,;.81,4.45,;2.91,3.89,;4.38,3.41,;5.28,4.66,;6.82,4.66,;7.59,5.99,;7.59,7.53,;6.26,6.76,;9.13,5.99,;9.9,7.32,;9.9,4.66,;4.38,5.9,;2.91,5.43,;.11,2.64,;-1.22,3.41,;-1.22,4.95,;-2.55,2.64,;-5.35,.81,;-5.98,2.21,;-7.51,2.37,;-8.41,1.13,;-9.9,1.53,;-7.79,-.28,;-6.26,-.44,;-3.17,-3.86,;-2.08,-4.95,)|
CC1CCC(Cn2nc(-c3nc4NC(=O)[C@@](C)(c5nc(CC(C)(C)C(O)=O)cs5)c4c(N)n3)c3cccnc23)CC1 |r,wU:15.15,(-2.14,-7.53,;-3.23,-6.44,;-4.71,-6.84,;-5.8,-5.75,;-5.4,-4.26,;-6.49,-3.17,;-6.1,-1.69,;-4.63,-1.21,;-4.63,.33,;-3.3,1.1,;-1.96,.33,;-.63,1.1,;.83,.62,;1.74,1.87,;3.28,1.87,;.83,3.12,;.06,4.45,;2.17,3.89,;3.63,3.41,;4.54,4.66,;6.08,4.66,;6.85,5.99,;6.85,7.53,;5.51,6.76,;8.39,5.99,;9.16,7.32,;9.16,4.66,;3.63,5.9,;2.17,5.43,;-.63,2.64,;-1.96,3.41,;-1.96,4.95,;-3.3,2.64,;-6.1,.81,;-6.72,2.21,;-8.25,2.37,;-9.16,1.13,;-8.53,-.28,;-7,-.44,;-3.92,-3.86,;-2.83,-4.95,)|
CC1CCC(Cn2nc(-c3nc4NC(=O)[C@](C)(c4c(N)n3)c3ccc(CCC(O)=O)cc3)c3ccc(Cl)cc23)CC1 |r,wU:15.15,(-1.44,-8.59,;-2.53,-7.5,;-4.02,-7.9,;-5.11,-6.81,;-4.71,-5.32,;-5.8,-4.23,;-5.4,-2.75,;-3.94,-2.27,;-3.94,-.73,;-2.6,.04,;-1.27,-.73,;.07,.04,;1.53,-.44,;2.44,.81,;3.98,.81,;1.53,2.06,;1.13,3.54,;.07,1.58,;-1.27,2.35,;-1.27,3.89,;-2.6,1.58,;2.62,3.14,;4.11,2.75,;5.2,3.84,;4.8,5.32,;5.89,6.41,;7.37,6.01,;8.46,7.1,;9.95,6.7,;8.06,8.59,;3.31,5.72,;2.22,4.63,;-5.4,-.25,;-6.03,1.15,;-7.56,1.31,;-8.46,.07,;-9.95,.47,;-7.84,-1.34,;-6.3,-1.5,;-3.22,-4.92,;-2.13,-6.01,)|
CC1CCCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CC1N(CCNC1=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCC(C)(C)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCCC(F)(F)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCCCCCn1nc(-c2nc3NC(=O)[C@](C)(c3c(N)n2)c2ccc(CCC(O)=O)cc2)c2ccc(Cl)cc12 |r|
CCCCCn1nc(-c2nc3NC(=O)[C@](C)(c3c(N)n2)c2ccc(CCC(O)=O)cc2)c2ccc(Cl)cc12 |r|
CCCCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1cc(O)c(Cl)c(F)c1
CCCCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1cc(O)c(Cl)cn1
CCCCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(Cl)c(O)c1
CCCCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(O)c(Cl)c1
CCCCc1nc(cn2ccnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(c(O)c1)C(F)(F)F
CCCCc1nc(cn2ncnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1cc(O)c(Cl)c(F)c1
CCCCc1nc(cn2ncnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1cc(O)ccn1
CCCCc1nc(cn2ncnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(Cl)c(O)c1
CCCCc1nc(cn2ncnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(F)c(O)c1
CCCCc1nc(cn2ncnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(O)c(Cl)c1
CCCCc1nc(cn2ncnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(O)c(F)c1
CCCCc1nc(cn2ncnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(O)cc1
CCCCc1nc(cn2ncnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(c(O)c1)C(F)(F)F
CCCCc1nc(cn2ncnc12)-c1nc2NC(=O)C(C)(c2c(N)n1)c1cccc(O)c1
CCCCn1nc(-c2nc3NC(=O)C(C)(c3c(N)n2)c2ccc(CC(C)(C)C(O)=O)cc2)c2ccc(Cl)cc12
CCCCn1nc(-c2nc3NC(=O)C(C)(c4cn(CC(O)=O)nn4)c3c(N)n2)c2ccc(Cl)cc12
CCCCn1nc(-c2nc3NC(=O)C(C)(c4cn(CCC(O)=O)nn4)c3c(N)n2)c2ccc(Cl)cc12
CCCCn1nc(-c2nc3NC(=O)C(C)(c4nc(CC(C)(C)C(O)=O)cs4)c3c(N)n2)c2cccnc12
CCCCn1nc(-c2nc3NC(=O)[C@](C)(c3c(N)n2)c2ccc(CCC(O)=O)cc2)c2ccc(C)nc12 |r|
CCCCn1nc(-c2nc3NC(=O)[C@](C)(c3c(N)n2)c2ccc(CCC(O)=O)cc2)c2ccc(Cl)cc12 |r|
CCCCn1nc(-c2nc3NC(=O)[C@](C)(c3c(N)n2)c2ccc(CCC(O)=O)cc2)c2ccc(Cl)nc12 |r|
CCCCn1nc(-c2nc3NC(=O)[C@](C)(c3c(N)n2)c2ccc(CCC(O)=O)cc2)c2cccnc12 |r|
CCCS(=O)(=O)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCN(CC)c1nc(ncc1F)-c1cc(-c2ccon2)n(CCC(F)(F)F)n1
CCN(CC1(CC1)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCOC(=O)C1(C)C(=O)Nc2cnc(nc12)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCOC(=O)C1(C)C(=O)Nc2nc(nc(N)c12)-c1cc(-c2ccon2)n(CCC(F)(F)F)n1
CCOC(=O)C1(C)C(=O)Nc2nc(nc(N)c12)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCOC(=O)C1(C)CCN(C1=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCOC(=O)C1=C(O)CN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |c:5|
CCOC(=O)CN1CCCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCOC(=O)c1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCOC(=O)c1cnc(nc1O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCOC(=O)c1csc(CN(C)c2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)n1
CCOCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CCOc1c(Nc2ccnc(n2)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)c(=O)c1=O
CC[C@H](NC(=O)CCc1ccc(cc1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)C(O)=O |r|
CC[C@H]1CCCN([C@H]1C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
CN(C(=O)C(C)(C)C)c1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(C(=O)OC(C)(C)C)c1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(C(=O)c1ccccc1)c1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(C)C(=O)Oc1cnc(nc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(C)S(=O)(=O)NCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(C)\C=N\c1cnc(nc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(C)c1ccccc1C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(CC(=O)NS(=O)(=O)c1ccccc1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(CC(C)(C)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(CC(C)(O)C(N)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(CC(O)(C(F)(F)F)C(F)(F)F)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(CC1(CC1)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(CCC(F)(F)F)n1
CN(CC1(CC1)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(CC1(CC1)C(O)=O)c1nc(ncc1F)-c1cc(-c2cscn2)n(Cc2ccccc2F)n1
CN(CC1(CC1)C(O)=O)c1nc(ncc1F)-c1cc(-c2nccs2)n(Cc2ccccc2F)n1
CN(CC1(CC1)C(O)=O)c1nc(ncc1F)-c1cc(C#N)n(Cc2ccccc2F)n1
CN(CC1(CC1)C(O)=O)c1nc(ncc1F)-c1cc(C(C)=O)n(Cc2ccccc2F)n1
CN(CC1(CC1)C(O)=O)c1nc(ncc1F)-c1cc(C(N)=O)n(Cc2ccccc2F)n1
CN(CC1(CC1)C(O)=O)c1nc(ncc1F)-c1cc(C)n(Cc2ccccc2F)n1
CN(CC1(CCC1)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(CCS(N)(=O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(CCS(O)(=O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(C[C@@H](O)CO)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
CN(C[C@H](O)CO)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
CN(Cc1nc(cn1C)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(Cc1nc(co1)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(Cc1nc(cs1)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN(Cc1nn[nH]n1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CN([C@@H](C1CC1)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
CN([C@@H](Cc1ccccn1)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
CN([C@@H]1CC[C@@H](C1)C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
CN(c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C12CC(C1)(C2)C(O)=O
CN(c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)S(C)(=O)=O
CN1CCN(CC1)c1nc(nc2NC(=O)C(C)(c12)c1ccc(Cl)c(O)c1)-c1cn2ccnc2c(Cc2ccc(F)cc2)n1
CNC(=O)C(C)(O)CN(C)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CNS(=O)(=O)CCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CNc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)CS(=O)(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)N(C)c1c(N)nc(nc1N)-c1cc(-c2ccccc2)n(Cc2ccccc2F)n1
COC(=O)N(C)c1c(N)nc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)N(C)c1c(N)nc(nc1N)-c1cc(-c2ccsc2)n(Cc2ccccc2F)n1
COC(=O)N(C)c1c(N)nc(nc1N)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
COC(=O)N(C)c1cnc(nc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)N(C)c1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)N1CCN(C(C1)OC=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)NCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)NCC(Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
COC(=O)Nc1c(N)nc(nc1N)-c1cc(-c2ccccc2)n(Cc2ccccc2F)n1
COC(=O)Nc1c(N)nc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)Nc1c(N)nc(nc1N)-c1cc(-c2ccsc2)n(Cc2ccccc2F)n1
COC(=O)Nc1c(N)nc(nc1N)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
COC(=O)Nc1c(N)nc(nc1N)-c1cc(-c2nccs2)n(Cc2ccccc2F)n1
COC(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)Nc1nc(ncc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)Nc1nc(ncc1[N+]([O-])=O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COC(=O)[C@@H]1CCC(=O)N1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
COC(C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)(c1ccccc1)C(F)(F)F
COC(C)(C)C(CC(O)=O)c1ccc(Cl)c(NC(=O)[C@@H]([C@@H](C)C(F)(F)F)c2ccc(Cl)cc2)c1 |r|
COC1CCCN(C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COCC(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COCCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COCCS(=O)(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COCCS(=O)(=O)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COCCn1nc(-c2nc3NC(=O)C(C)(c3c(N)n2)c2cccc(CC(C)(C)C(O)=O)c2)c2ccc(Cl)cc12
COCCn1nc(-c2nc3NC(=O)[C@](C)(c3c(N)n2)c2ccc(CCC(O)=O)cc2)c2ccc(Cl)cc12 |r|
CO[C@@](C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)(c1ccccc1)C(F)(F)F |r|
CO[C@H](C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)c1ccccc1 |r|
COc1cc(on1)C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COc1ccc(cc1)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COc1ccc(cc1)C1=Nc2nc(ncc2C(C)(C)O1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |t:9|
COc1ccc(cc1OC)S(=O)(=O)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COc1ccc2C(OC=O)N(CCc2c1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COc1cccc(c1)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COc1cccc(n1)-c1cc(nn1Cc1ccccc1F)-c1ncccn1
COc1ccccc1C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
COc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CS(=O)(=O)C1(CNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)CC1
CS(=O)(=O)C1CCN(C1)c1nc(ncc1F)C1=NC(Cc2ccccc2F)C(=C1)c1ccon1 |c:30,t:18|
CS(=O)(=O)CC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CS(=O)(=O)CC(=O)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CS(=O)(=O)CCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CS(=O)(=O)CCC(Nc1nc(ncc1F)-c1cc(-c2ccon2)n(CCC(F)(F)F)n1)C(F)(F)F
CS(=O)(=O)CCC(Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
CS(=O)(=O)CCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CS(=O)(=O)CS(=O)(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CS(=O)(=O)NC(=O)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CS(=O)(=O)NCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CS(=O)(=O)NCC(O)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
CS(=O)(=O)NCCC(Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
CS(=O)(=O)c1cnc(nc1O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
C[C@@H](Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)c1nnc(o1)C(F)(F)F |r|
C[C@@H]1CCCN([C@@H]1C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
C[C@@H]1CN(C[C@@H]1C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
C[C@@H]1[C@@H](CCCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O |r|
C[C@H](NC(=O)CCc1ccc(cc1)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)C(O)=O |r|
C[C@H](O)C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
C[C@H]([C@H](C(=O)Nc1cc(ccc1Cl)C(C)(CC(O)=O)C1CCC1)c1ccc(Cl)cc1)C(F)(F)F |r|
C[C@H]([C@H](C(=O)Nc1cc(ccc1Cl)C(CC(O)=O)C1(F)CC1)c1ccc(Cl)cc1)C(F)(F)F |r|
C[C@H]([C@H](C(=O)Nc1cc(ccc1Cl)C(CC(O)=O)C1CC1)c1ccc(Cl)cc1)C(F)(F)F |r|
C[C@H]([C@H](C(=O)Nc1cc(ccc1Cl)C(CC(O)=O)C1CCC1)c1ccc(Cl)cc1)C(F)(F)F |r|
C[C@H]([C@H](C(=O)Nc1cc(ccc1Cl)C(CC1CC1)CC(O)=O)c1ccc(Cl)cc1)C(F)(F)F |r|
C[C@H]1CCCN([C@@H]1C(=O)NS(=O)(=O)C1CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
C[C@H]1CCCN([C@@H]1C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
C[C@H]1CCCN([C@H]1C(=O)NS(=O)(=O)C1CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
C[C@H]1CCCN([C@H]1C(O)=O)c1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
C[C@H]1CCCN([C@H]1C(O)=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
C[C@H]1CCCN([C@H]1C(O)=O)c1nc(ncc1F)-c1cc(C#N)n(Cc2ccccc2F)n1 |r|
C[C@H]1CCCN([C@H]1C(O)=O)c1nc(ncc1F)-c1cc(C)n(Cc2ccccc2F)n1 |r|
C[C@H]1CCCN([C@H]1OC=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2cccc(F)c2F)n1 |r|
C[C@H]1CCCN([C@H]1OC=O)c1nc(ncc1F)-c1cc(C(C)=O)n(Cc2ccccc2F)n1 |r|
C[C@H]1CCCN([C@H]1c1nn[nH]n1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
C[C@H]1[C@H](CCCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(O)=O |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CC(F)(F)C2)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCC(F)(F)CC2)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCC2)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCC2)c2ccccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CC2CCCCC2)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12)c1ccc(CCc2nn[nH]n2)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(F)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12)c1nc(CCC(O)=O)cs1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2nc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2ncc(F)cc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2ncccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(CCCC(F)(F)F)c2ncccc12)c1nc(CCC(O)=O)cs1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2c(F)cccc2F)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccc(F)cc2)c2ccccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)c(O)cc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1cc(C[C@@H](N)C(O)=O)cs1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(CCC(=O)NS(C)(=O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(CCc2nn[nH]n2)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12)c1ccc(CCc2noc(=O)[nH]2)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(F)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ccccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ccccc12)c1ccc(CCc2nn[nH]n2)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncc(F)cc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1ccc(CCC(=O)NCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1ccc(CCC(=O)NCc2nn[nH]n2)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1ccc(CCC(=O)N[C@H](CO)C(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2ncccc12)c1ccc(CCc2nn[nH]n2)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ncccc2F)c2cc(Cl)ccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ncccc2F)c2ccccc12)c1ccc(CCC(O)=O)cc1 |r|
C[C@]1(C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ncccc2F)c2ccccc12)c1ccc(CCc2nn[nH]n2)cc1 |r|
C\C=C(/C)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Cc1cc(Cl)nc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Cc1cc(N)nc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Cc1cc(ccc1CCC(O)=O)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12
Cc1cc(ccc1O)C1(C)C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1
Cc1cc(nn1Cc1ccccc1F)-c1ccccn1
Cc1cc(nn1Cc1ccccc1F)-c1ncc(F)c(=O)[nH]1
Cc1cc(nn1Cc1ccccc1F)-c1ncc(F)c(NC(CO)CO)n1
Cc1cc(nn1Cc1ccccc1F)-c1ncc(F)c(NCC(O)(C(F)(F)F)C(F)(F)F)n1
Cc1ccc(Cn2nc(-c3nc4NC(=O)[C@](C)(c4c(N)n3)c3ccc(CCC(O)=O)cc3)c3ccc(Cl)cc23)cc1 |r|
Cc1ccc(F)c(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3ccc(Cl)cc23)c1
Cc1ccc(F)c(Cn2nc(-c3nc4NC(=O)[C@@](C)(c5nc(CC(C)(C)C(O)=O)cs5)c4c(N)n3)c3ccc(Cl)cc23)c1 |r|
Cc1ccc(cc1)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Cc1ccc(cc1O)C1(C)C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1
Cc1ccc2c(nn(CCCC(F)(F)F)c2n1)-c1nc2NC(=O)[C@](C)(c2c(N)n1)c1ccc(CCC(O)=O)cc1 |r|
Cc1ccc2c(nn(Cc3ccc(C)c(F)c3F)c2n1)-c1nc2NC(=O)[C@](C)(c2c(N)n1)c1ccc(CCC(O)=O)cc1 |r|
Cc1ccc2c(nn(Cc3ccccc3F)c2c1)-c1nc2NC(=O)[C@](C)(c2c(N)n1)c1ccc(CCC(O)=O)cc1 |r|
Cc1cccc(C)c1C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Cc1cccc(Cc2nc(cn3ccnc23)-c2nc3NC(=O)C(C)(c3c(N)n2)c2ccc(O)c(F)c2)c1
Cc1cccc(Cc2nc(cn3ccnc23)-c2nc3NC(=O)C(C)(c3c(N)n2)c2cccc(O)c2)c1
Cc1cccc(Cn2nc(-c3nc4NC(=O)C(C)(c5cnn(CC(C)(C)C(O)=O)c5)c4c(N)n3)c3ccc(F)cc23)c1F
Cc1cccc(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3ccc(Cl)cc23)c1
Cc1cccc(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3ccc(Cl)cc23)c1F
Cc1cccc(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3ccc(F)cc23)c1F
Cc1cccc(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3ccccc23)c1
Cc1cccc(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3ccccc23)c1F
Cc1cccc(Cn2nc(-c3nc4NC(=O)[C@@](C)(c5nc(CC(C)(C)C(O)=O)cs5)c4c(N)n3)c3ccc(Cl)cc23)c1F |r|
Cc1cccc(Cn2nc(-c3nc4NC(=O)[C@](C)(c4c(N)n3)c3ccc(CCC(O)=O)cc3)c3ccc(Cl)cc23)c1 |r|
Cc1cccc(Cn2nc(-c3nc4NC(=O)[C@](C)(c4c(N)n3)c3ccc(CCC(O)=O)cc3)c3ccccc23)c1 |r|
Cc1cccc(c1)C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Cc1ccccc1C(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Cc1ccccc1Cn1nc(-c2nc3NC(=O)[C@](C)(c3c(N)n2)c2ccc(CCC(O)=O)cc2)c2ccc(Cl)cc12 |r|
Cc1ccnc(Cn2nc(-c3nc4NC(=O)C(C)(c5nc(CC(C)(C)C(O)=O)co5)c4c(N)n3)c3ccc(Cl)cc23)c1F
Cc1ccnc(Cn2nc(-c3nc4NC(=O)[C@@](C)(c5nc(CC(C)(C)C(O)=O)cs5)c4c(N)n3)c3ccc(Cl)cc23)c1F |r|
Cc1cn(CC(=O)Nc2ccnc(n2)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)c(=O)[nH]c1=O
Cc1cn2cc(nc(Cc3cccc(F)c3)c2n1)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(Cl)c(O)c1
Cc1cn2cc(nc(Cc3ccccc3F)c2n1)-c1nc2NC(=O)C(C)(c2c(N)n1)c1ccc(Cl)c(O)c1
Cc1cnc(cc1O)C1(C)C(=O)Nc2nc(nc(N)c12)-c1cn2ccnc2c(Cc2cccc(F)c2)n1
Cc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Cc1csc(n1)-c1cc(nn1Cc1ccccc1F)-c1ncccn1
Cc1nc(nc(O)c1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Cc1nc(sc1CC(O)=O)[C@]1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(CCC(F)(F)C(F)(F)F)c2ncccc12 |r|
Cc1nnc(CNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)o1
Cc1oc(nc1CC(C)(C)C(O)=O)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2cc(Cl)ccc12
Cc1oc(nc1CC(C)(C)C(O)=O)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2cccc(F)c2)c2cc(F)ccc12
Cc1oc(nc1CC(C)(C)C(O)=O)C1(C)C(=O)Nc2nc(nc(N)c12)-c1nn(Cc2ccccc2F)c2cc(Cl)ccc12
Clc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncccn1
Cn1c2c(N)nc(nc2[nH]c1=O)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
Cn1c2c(N)nc(nc2[nH]c1=O)-c1cc(-c2nccs2)n(Cc2ccccc2F)n1
Fc1ccc(CS(=O)(=O)Nc2ccnc(n2)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)cc1
Fc1ccc(CS(=O)(=O)Nc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)cc1
Fc1ccc(cc1)S(=O)(=O)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Fc1cccc(Cn2nc(cc2-c2ccon2)-c2ncccn2)c1
Fc1cccc(Cn2nc(cc2-c2ccon2)-c2ncccn2)c1F
Fc1cccc(F)c1Cn1nc(cc1-c1ccon1)-c1ncccn1
Fc1ccccc1Cn1nc(cc1-c1ccccn1)-c1ccccn1
Fc1ccccc1Cn1nc(cc1-c1ccccn1)-c1ncccn1
Fc1ccccc1Cn1nc(cc1-c1ccco1)-c1ccccn1
Fc1ccccc1Cn1nc(cc1-c1ccco1)-c1ncccn1
Fc1ccccc1Cn1nc(cc1-c1cccs1)-c1ncccn1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nc(Cl)cc(n1)-c1cccnc1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NC(=O)C(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NC(=O)C2(CC2)C#N)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NC(=O)C2(CC2)C(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NC(=O)N2CCOCC2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NC(C(=O)NC2CC2)C(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NC2CCCNC2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NC2CCOC2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NC2CN(C2)S(=O)(=O)C(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NC2CNC(=O)C2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NCC(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NCC2(CC2)NS(=O)(=O)C(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NCC2(CC2)c2ncc[nH]2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NCCNS(=O)(=O)C(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NCCS(=O)(=O)C(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NCCS(=O)(=O)NCC(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NCCSC(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NCc2n[nH]c(=O)[nH]2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NCc2nnc(o2)C(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NS(=O)(=O)C2CC2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NS(=O)(=O)CC(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NS(=O)(=O)CCC(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NS(=O)(=O)c2ccccc2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(NS(=O)(=O)c2cccnc2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(N[C@H]2CCNC2=O)n1 |r|
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(S)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)-n1[nH]cnc1=O
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1C(=O)CCC1=O
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1C(=O)CCS1(=O)=O
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1C(CCC1=O)C(F)(F)F
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CC(C1)NC(=O)C(F)(F)F
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CC(C1)NS(=O)(=O)C(F)(F)F
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCC(C1)S(=O)(=O)NC(=O)C1CC1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCC(CC1)S(=O)(=O)N1CCOCC1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCC(CC1)S(=O)(=O)NC(=O)C1CC1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCCC2CC12
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCCCC1=O
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCCS1(=O)=O
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCC[C@@H](C1)c1ccccc1 |r|
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCNC(=O)C1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCNCC1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCNCC1OC=O
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCOCC1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCc2[nH]nc(c2C1)C(F)(F)F
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCc2ccccc2C1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCc2nc[nH]c2C1OC=O
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(F)c(n1)N1CCn2c(C1)nnc2C(F)(F)F
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc(NS(=O)(=O)CCC(F)(F)F)cn1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc2OC(C(=O)Nc2n1)(C(F)(F)F)C(F)(F)F
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncc2[nH]c(=O)[nH]c2n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)C(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)C2(CC2)C#N)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)C2(CC2)C(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)C2(CC2)OCc2ccccc2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)C2(CCOCC2)OCc2ccccc2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)C2CC2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)C2CCC(=O)N2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)C2CCCO2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)C2CCOCC2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)C2CNC(=O)C2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)CC#N)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)CC(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)CN2C(=O)c3ccccc3C2=O)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)CN2CCOC2=O)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)CN2Cc3ccccc3C2=O)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)CNC(=O)CN2C(=O)c3ccccc3C2=O)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)CNC(=O)Cc2ccccc2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)CNC(=O)OCc2ccccc2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)CS(=O)(=O)c2ccc(Cl)cc2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)CS(=O)(=O)c2ccccc2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)Cc2nccs2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)Cn2cnc3ccccc3c2=O)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)Nc2ccccc2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2cc(n[nH]2)C2CC2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2cc[nH]n2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2ccc[nH]2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2cccc(=O)[nH]2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2ccco2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2cccs2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2ccncn2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2cnco2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2cncs2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2cocn2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NC(=O)c2cscn2)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(NS(=O)(=O)CC(F)(F)F)n1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(n1)N1C(COC1=O)C(F)(F)F
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(n1)N1CC(OC1=O)C(F)(F)F
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1nccc(n1)N1CCOCC1
Fc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncccn1
Fc1ccccc1Cn1nc(cc1-c1ccsc1)-c1ccccn1
Fc1ccccc1Cn1nc(cc1-c1ccsc1)-c1ncccn1
Fc1ccccc1Cn1nc(cc1-c1cscn1)-c1ncccn1
Fc1ccccc1Cn1nc(cc1-c1ncco1)-c1ncccn1
Fc1ccccc1Cn1nc(cc1-c1nccs1)-c1ccccn1
Fc1ccccc1Cn1nc(cc1-c1nccs1)-c1ncccn1
Fc1ccccc1Cn1nc(cc1-c1ncon1)-c1ccccn1
Fc1ccccc1Cn1nc(cc1-c1nnco1)-c1ccccn1
Fc1ccccc1Cn1nc(cc1C#N)-c1ncccn1
Fc1ccccc1Cn1nc(cc1C1CCC1)-c1ccccn1
Fc1ccccc1Cn1nc(cc1[N+]#[C-])-c1ccccn1
NC(=O)C(Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
NC(=O)C(O)(CNc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
NC(=O)C(O)(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2cccc(F)c2F)n1)C(F)(F)F
NC(=O)C(O)(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
NC(=O)C(O)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NC(=O)C1(CC1)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NC(=O)C1(CNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)CC1
NC(=O)C1(O)CCN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NC(=O)C1CCC(=O)N1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NC(=O)C1CN(C(=O)C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NC(=O)CC(Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
NC(=O)CCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NC(=O)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(CCC(F)(F)F)n1
NC(=O)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NC(=O)NCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NC(=O)[C@@](O)(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F |r|
NC(=O)[C@H](CO)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
NC(=O)[C@](O)(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F |r|
NC(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
NCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NCC(=O)Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NCC(O)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NCCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NS(=O)(=O)C1CCN(C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NS(=O)(=O)C1CCN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NS(=O)(=O)CCCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
NS(=O)(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1cc(N)nc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1cc(nc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)-c1cccnc1
Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1ccnc(n1)-c1cc(-c2ccsc2)n(Cc2ccccc2F)n1
Nc1ccnc(n1)-c1cc(-c2cnco2)n(Cc2ccccc2F)n1
Nc1ccnc(n1)-c1cc(-c2cocn2)n(Cc2ccccc2F)n1
Nc1ccnc(n1)-c1cc(-c2cscn2)n(Cc2ccccc2F)n1
Nc1ccnc(n1)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
Nc1ccnc(n1)-c1cc(-c2nccs2)n(Cc2ccccc2F)n1
Nc1cnc(nc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1cnc(nc1N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1cnc(nc1N)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
Nc1cnc(nc1NCC(O)(C(F)(F)F)C(F)(F)F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(nc2CS(=O)(=O)Cc12)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(nc2NC(=O)C(C3CC3)(c12)c1ccc(CCC(O)=O)cc1)-c1nn(CCC(F)(F)C(F)(F)F)c2cc(Cl)ccc12
Nc1nc(nc2NC(=O)C(C3CC3)(c12)c1ccc(CCC(O)=O)cc1)-c1nn(Cc2ccccc2F)c2ncccc12
Nc1nc(ncc1-c1ccccc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1-c1ccccn1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1-c1cccnc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1-c1ccncc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1-c1ccsc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1-c1nccs1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1C#N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1C(F)(F)F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1C(O)=O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1C1(CC1)OCC=C)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1C1(O)CC1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1C1CC1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1F)-c1cc(-c2ccon2)n(CCC(F)(F)F)n1
Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1F)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
Nc1nc(ncc1N1CCCC1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1N1CCCC1=O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1N1CCOC1=O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1N1CCOCC1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1N1Cc2ccccc2C1=O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)C(F)(F)c1ccccc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)C1(CC1)C(F)(F)F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)C1(CC1)C(F)(F)F)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)C1(CC1)[N+]#[C-])-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)C1(CCC1)C(F)(F)F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)C1(CCC1)c1ccccc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)C12CC3CC(CC(C3)C1)C2)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |TLB:17:16:19:13.12.11,17:12:19:18.15.16,THB:18:10:13:17.15.16,18:16:13:19.10.11|
Nc1nc(ncc1NC(=O)C1CC1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)C1CC2CC1C=C2)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |c:17|
Nc1nc(ncc1NC(=O)CCCCl)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)CN1C(=O)c2ccccc2C1=O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)OCCCl)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)OCc1ccccc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)[C@@H]1CCCN1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
Nc1nc(ncc1NC(=O)[C@@H]1CCCN1C(=O)C(F)(F)F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
Nc1nc(ncc1NC(=O)\C=C\c1ccccc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1ccc(Cl)cc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1ccc(F)cc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1cccc(Cl)c1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1cccc(F)c1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1cccc(O)n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1cccc(OC(F)(F)F)c1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1cccc(c1)C(F)(F)F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1ccccc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1ccccc1)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1ccccc1Cl)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1ccccc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1ccccc1OC(F)(F)F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1ccccn1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1cccnc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1ccncc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1ccon1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1cnco1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1cocn1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1cscn1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NC(=O)c1nccs1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1NCc1ccccc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Nc1nc(ncc1Nc1nccs1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C(CC(F)F)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C(F)(F)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C(Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
OC(=O)C(O)(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2cccc(F)c2F)n1)C(F)(F)F
OC(=O)C(O)(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
OC(=O)C1(CC1)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C1(CC1)c1ccc(Nc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)cc1
OC(=O)C1(CCCC1)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C1(CCN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)c1ccccc1
OC(=O)C1(CNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)CC1
OC(=O)C1(CNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)CCCC1
OC(=O)C1(F)CCN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C1(O)CCN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C12CC(C1)(C2)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C12CC1CN(C2)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C1CCCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C1CCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C1CCc2ccccc2N1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C1CN(C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)C1N(Cc2ccccc12)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)CC(Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
OC(=O)CC1(CCOCC1)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)CC1CCN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)CCCCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)CCCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(=O)[C@@H](Cc1cc2ccccc2[nH]1)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@@H]1CCCC[C@H]1Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@@H]1CCc2ccccc2[C@@H]1Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@@H]1CN(C[C@H]1C(F)(F)F)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@@H]1COCCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@@H]1Cc2ccccc2N1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@@H]1Cc2ccccc2[C@@H]1Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@@H]1[C@H]2CC[C@H](C2)N1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@@H]1[C@H]2CC[C@H](O2)[C@@H]1Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@H](Cc1cc2ccccc2[nH]1)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@H]1CCC[C@H](C1)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@H]1COCCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@H]1C[C@@H](CCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F |r|
OC(=O)[C@H]1C[C@H](CCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F |r|
OC(=O)[C@H]1[C@H](CCCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F |r|
OC(=O)[C@H]1[C@H]2CC[C@H](C2)[C@H]1Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)[C@]1(CC2CC[C@H]1C2)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC(=O)c1cc(nn1Cc1ccccc1F)-c1ncc(F)c(NCC(O)(C(F)(F)F)C(F)(F)F)n1
OC(=O)c1ccc(CNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)s1
OC(=O)c1cccc(CCNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)c1
OC(=O)c1cccn1-c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC(C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)(C(F)(F)F)C(F)(F)F
OC(C(=O)Nc1nc(ncc1N1CCOCC1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)(C(F)(F)F)C(F)(F)F
OC(C1CN(C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)(C(F)(F)F)C(F)(F)F
OC(CC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)(C(F)(F)F)C(F)(F)F
OC(CNc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)(C(F)(F)F)C(F)(F)F
OC(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(CCC(F)(F)F)n1)(C(F)(F)F)C(F)(F)F
OC(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2cccc(F)c2F)n1)(C(F)(F)F)C(F)(F)F
OC(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)(C(F)(F)F)C(F)(F)F
OC(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
OC(CNc1nc(ncc1F)-c1cc(C#N)n(Cc2ccccc2F)n1)(C(F)(F)F)C(F)(F)F
OC(CNc1nc(ncc1[N+]([O-])=O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)(C(F)(F)F)C(F)(F)F
OC1(CC1)C(=O)N1CC(C1)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC1(CC1)C(=O)NC1CN(C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC1(CC1)C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC1(CN(C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
OC1(CNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)CCOCC1
OC1(CNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)CNC1
OC1=CC(=O)CC(C1)C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |t:1|
OC1=CC(=O)CN(C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |t:1|
OC1CCN(C1=O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC(=O)N(CC(F)(F)F)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC(CC(F)F)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC(CO)(CO)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC(CO)NC(=O)[C@@H](CO)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OCC(CO)Nc1cnnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC(CO)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC(F)(F)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC(Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
OCC(O)(CCl)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC(O)(CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F
OCC1(CC1)Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC1(O)CCN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCC1Cn2c(CN1c1nc(ncc1F)-c1cc(-c3ccon3)n(Cc3ccccc3F)n1)nnc2C(F)(F)F
OCCCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCCN(CCO)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCCNS(=O)(=O)CCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCCS(=O)(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OCCc1cnc(nc1O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OC[C@@H](O)CN(CC1CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC[C@@H](O)CNS(=O)(=O)CCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC[C@@H](O)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC[C@@H]1C[C@@H](O)CN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC[C@@H]1[C@H](O)CCN1c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC[C@H](O)CNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC[C@H]1CCN([C@@H](CO)C1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
OC[C@H]1CN(C(=O)O1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
ONS(=O)(=O)CCNc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
OS(=O)(=O)C1CCN(CC1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
O[C@@H](C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1)C(F)(F)F |r|
O[C@@H]1Cc2ccccc2[C@@H]1Nc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
O[C@H]1CCN(C[C@H]1O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
O[C@H]1CN(C[C@@H](O)[C@H]1O)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1 |r|
Oc1c(F)cc(CNc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)cc1F
Oc1c(Nc2ccnc(n2)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)c(=O)c1=O
Oc1cc(=O)c2c(O)nc(nc2o1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1cc(O)nc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1ccc(C[C@H](Nc2nc(ncc2F)-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)OC=O)cc1 |r|
Oc1ccc2C(OC=O)N(CCc2c1)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1ccccc1C(=O)Nc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1ccccc1Cn1nc(cc1-c1ccon1)-c1ncccn1
Oc1ccnc(n1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1coc(n1)-c1cc(nn1Cc1ccccc1F)-c1ncccn1
Oc1n[nH]c2CCN(Cc12)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1n[nH]c2CN(CCc12)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(nc(O)c1[N+]([O-])=O)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(nc2CS(=O)(=O)Cc12)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1Br)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1C#N)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1C#N)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
Oc1nc(ncc1C(F)(F)F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1Cl)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1F)-c1cc(-c2ccon2)n(CCC(F)(F)F)n1
Oc1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1F)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
Oc1nc(ncc1NC(=O)c1ccccc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1S(=O)(=O)N1CCOCC1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1S(=O)(=O)c1cc(Cl)ccc1Cl)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1S(=O)(=O)c1ccc(F)cc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1S(=O)(=O)c1ccccc1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
Oc1nc(ncc1S(=O)(=O)c1ccccc1)-c1cc(-c2ncco2)n(Cc2ccccc2F)n1
Oc1noc2CN(CCc12)c1nc(ncc1F)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1
[#6]\[#6](-[#6])=[#6]\[#6](=O)-[#7]-c1cnc(nc1-[#7])-c1cc(-c2ccon2)n(-[#6]-c2ccccc2F)n1
[#7]-c1nc(ncc1\[#7]=[#6](/c1ccccc1)-c1ccccc1)-c1cc(-c2ncco2)n(-[#6]-c2ccccc2F)n1
[O-][N+](=O)c1cnc(nc1N1CCOCC1)-c1cc(-c2ccon2)n(Cc2ccccc2F)n1