955 SMILES Strings for Serine/threonine-protein kinase Sgk1

Compound Name
SMILES String
O=Nc1c([nH]c2ccccc12)C1C(=O)Nc2ccccc12
COc1ccc(cc1OC)-c1cc2c(nc[nH]c2=O)s1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cnc2cn[nH]c2n1
Fc1cc(ccc1NS(=O)(=O)c1cc(Cl)ccc1Cl)-c1cnc2cn[nH]c2n1
Fc1cc(ccc1NS(=O)(=O)c1cccc(Cl)c1Cl)-c1cnc2cn[nH]c2n1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)c(F)c1
NNc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1cnc2c(N)n[nH]c2n1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)c(F)c1
Cc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
Cc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cnc2c(C)n[nH]c2n1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Fc1cc(F)c(cc1Cl)S(=O)(=O)Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Cc1nn(C)c(Cl)c1S(=O)(=O)Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2c(C)nn(C)c2Cl)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(ccc2F)C#N)cc1
COc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cnc2c(N)n[nH]c2n1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2Cl)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2ccc(F)cc2Cl)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cccc(F)c2Cl)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2ccccc2Cl)cc1
Cc1nn(C)cc1S(=O)(=O)Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2c(C)nn(C)c2Cl)cc1
CC(C)c1[nH]nc(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(\C=C\CCN2CCCC3(CCNCC3)C2)cc1C |r|
Nc1ccc(cn1)-c1ccc2ncc3c(n(-c4cccc(c4)C(F)(F)F)c(=O)[nH]c3=O)c2n1
Cc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(N2CCOCC2)c2cn[nH]c2n1
OC1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |(44.14,-2.28,;42.6,-2.28,;41.82,-3.61,;40.29,-3.61,;39.52,-2.26,;40.28,-.93,;41.83,-.94,;37.97,-2.27,;37.2,-3.6,;35.66,-3.61,;34.89,-4.94,;35.66,-6.28,;37.2,-6.27,;38.22,-7.42,;39.63,-6.81,;39.48,-5.28,;37.98,-4.95,;33.36,-4.93,;32.58,-6.27,;31.04,-6.26,;30.28,-4.92,;28.73,-4.91,;27.96,-6.24,;29.29,-7.02,;27.96,-7.78,;26.42,-6.25,;25.65,-4.92,;24.1,-4.92,;23.33,-3.59,;23.34,-6.25,;24.11,-7.58,;25.65,-7.58,;26.42,-8.92,;31.04,-3.59,;32.58,-3.59,)|
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCC(O)CC2)c2cn[nH]c2n1 |(-8.75,3.52,;-8.75,1.98,;-10.09,1.21,;-10.09,-.33,;-8.75,-1.16,;-8.75,-2.7,;-8.75,-4.24,;-7.42,-.33,;-7.42,1.21,;-6.08,-1.1,;-4.75,-1.87,;-6.85,-2.44,;-5.31,.23,;-3.77,.23,;-3,-1.1,;-1.46,-1.1,;-.69,.23,;-1.46,1.56,;-3,1.56,;.85,.23,;1.62,1.56,;3.16,1.56,;3.93,2.9,;5.47,2.9,;6.24,1.56,;7.78,1.56,;8.55,2.9,;10.09,2.9,;7.78,4.23,;6.24,4.23,;3.93,.23,;5.43,-.09,;5.59,-1.62,;4.19,-2.25,;3.16,-1.1,;1.62,-1.1,)|
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(-c2cccnc2)c2cn[nH]c2n1
Cc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(N2CCOCC2)c2cn[nH]c2n1
Cc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
CN1CCN(CC1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
CN1CCN(CC1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1nc(N2CCNCC2)c2cn[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(N2CCNCC2)c2cn[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(N2CCNCC2)c2cn[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(NCc2ccccn2)c2cn[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(NCc2cccnc2)c2cn[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(NCc2ccncc2)c2cn[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(Oc2ccncc2)c2cn[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(Oc2ccncc2)c2cn[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(-c2ccncc2)c2cn[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(Oc2cccnc2)c2cn[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(Oc2cccnc2)c2cn[nH]c2n1
OCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
OCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OCCCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
OCCCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OCCCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Oc1ccc(Oc2nc(nc3[nH]ncc23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3F)cc2)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(-n2ccnc2)c2cn[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(-n2cncn2)c2cn[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(-n2cncn2)c2cn[nH]c2n1
OCCCNc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OCCCNc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
NCCCNc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
NCCCNc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OCCNc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OCCNc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
OCCNc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
NCCNc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
NCCNc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
NCCCNc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
NCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
NCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
NCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
CC(C)(CO)COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CC(C)(CO)COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
CC(C)(CO)COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
OC1CCC(C1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
OC1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1 |(2.51,7.8,;3.28,6.46,;4.82,6.46,;5.59,5.13,;4.82,3.79,;3.28,3.79,;2.51,5.13,;5.59,2.46,;4.82,1.13,;3.28,1.13,;2.51,-.21,;3.28,-1.54,;4.82,-1.54,;5.85,-2.68,;7.25,-2.06,;7.09,-.53,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;.2,1.13,)|
NCCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
NCCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
NCCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OC1CCN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OC1CCN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
OC1CN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OC1CN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
CC1(C)C(O)C(C)(C)N1c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OC1CCN(CC1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OC1CCN(CC1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
OC1CCCN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
OC1CCC(C1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
O[C@H]1CC[C@H](CC1)Nc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r,wU:4.7,1.0,(2.51,7.8,;3.28,6.46,;4.82,6.46,;5.59,5.13,;4.82,3.79,;3.28,3.79,;2.51,5.13,;5.59,2.46,;4.82,1.13,;3.28,1.13,;2.51,-.21,;3.28,-1.54,;4.82,-1.54,;5.85,-2.68,;7.25,-2.06,;7.09,-.53,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;.2,1.13,)|
O[C@H]1CC[C@H](CC1)Nc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1 |r,wU:4.7,1.0,(2.51,7.8,;3.28,6.46,;4.82,6.46,;5.59,5.13,;4.82,3.79,;3.28,3.79,;2.51,5.13,;5.59,2.46,;4.82,1.13,;3.28,1.13,;2.51,-.21,;3.28,-1.54,;4.82,-1.54,;5.85,-2.68,;7.25,-2.06,;7.09,-.53,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;.2,1.13,)|
O[C@H]1CC[C@H](CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r,wU:1.0,4.7,(2.51,7.8,;3.28,6.46,;4.82,6.46,;5.59,5.13,;4.82,3.79,;3.28,3.79,;2.51,5.13,;5.59,2.46,;4.82,1.13,;3.28,1.13,;2.51,-.21,;3.28,-1.54,;4.82,-1.54,;5.85,-2.68,;7.25,-2.06,;7.09,-.53,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;.2,1.13,)|
O[C@H]1CC[C@H](CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1 |r,wU:1.0,4.7,(2.51,7.8,;3.28,6.46,;4.82,6.46,;5.59,5.13,;4.82,3.79,;3.28,3.79,;2.51,5.13,;5.59,2.46,;4.82,1.13,;3.28,1.13,;2.51,-.21,;3.28,-1.54,;4.82,-1.54,;5.85,-2.68,;7.25,-2.06,;7.09,-.53,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;.2,1.13,)|
O[C@H]1CCCC[C@H]1Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
O[C@@H]1CCCC[C@@H]1Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1 |r|
OC1CC[C@@H](CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1 |r,wU:4.7,(2.51,7.8,;3.28,6.46,;2.51,5.13,;3.28,3.79,;4.82,3.79,;5.59,5.13,;4.82,6.46,;5.59,2.46,;4.82,1.13,;3.28,1.13,;2.51,-.21,;3.28,-1.54,;4.82,-1.54,;5.85,-2.68,;7.25,-2.06,;7.09,-.53,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-7.09,-4.62,;-1.34,1.13,;.2,1.13,)|
OC1CCC[C@@H](C1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
OC1CCC[C@@H](C1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1 |r|
CC(C)(O)CCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
O[C@@H]1CCC[C@H]1Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
O[C@@H]1CCC[C@H]1Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1 |r|
OCCCSc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(O[C@H]2CCC(O)CC2)c2cn[nH]c2n1 |r,wU:23.24,(-8.43,3.85,;-7.09,3.08,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-5.76,-.77,;-5.76,.77,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-3.65,-.21,;-2.11,-.21,;-1.34,-1.54,;.2,-1.54,;.97,-.21,;.2,1.13,;-1.34,1.13,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;3.28,3.79,;2.51,5.13,;3.28,6.46,;2.51,7.8,;4.82,6.46,;5.59,5.13,;5.59,-.21,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,)|
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(O[C@@H]2CCC(O)C2)c2cn[nH]c2n1 |r|
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(O[C@H]2CCC(O)CC2)c2cn[nH]c2n1 |r,wU:22.23,(-7.09,3.08,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-5.76,-.77,;-5.76,.77,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-3.65,-.21,;-2.11,-.21,;-1.34,-1.54,;.2,-1.54,;.97,-.21,;.2,1.13,;-1.34,1.13,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;3.28,3.79,;2.51,5.13,;3.28,6.46,;2.51,7.8,;4.82,6.46,;5.59,5.13,;5.59,-.21,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,)|
Cc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
CN1N=C(C)C(C1Cl)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(C)n[nH]c2n1 |t:2|
Cc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCC(O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1 |(8.24,.5,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;5.59,5.13,;4.82,6.46,;3.28,6.46,;2.51,7.8,;2.51,5.13,;3.28,3.79,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-7.09,-4.62,;-1.34,1.13,;.2,1.13,)|
Cc1n[nH]c2nc(nc(C3CCC(O)C3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(NC3CC[C@H](O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1 |r,wD:13.13,(8.24,.5,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;3.28,3.79,;2.51,5.13,;3.28,6.46,;2.51,7.8,;4.82,6.46,;5.59,5.13,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-7.09,-4.62,;-1.34,1.13,;.2,1.13,)|
Cc1n[nH]c2nc(nc(NC3CCCC(O)C3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(NC3CCCC(O)C3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(OC3CC[C@H](O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1 |r,wD:13.13,(8.24,.5,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;3.28,3.79,;2.51,5.13,;3.28,6.46,;2.51,7.8,;4.82,6.46,;5.59,5.13,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;.2,1.13,)|
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CC[C@H](O)CC2)c2c(C)n[nH]c2n1 |r,wD:26.28,(-8.43,3.85,;-7.09,3.08,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-5.76,-.77,;-5.76,.77,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-3.65,-.21,;-2.11,-.21,;-1.34,-1.54,;.2,-1.54,;.97,-.21,;.2,1.13,;-1.34,1.13,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;3.28,3.79,;2.51,5.13,;3.28,6.46,;2.51,7.8,;4.82,6.46,;5.59,5.13,;5.59,-.21,;7.09,-.53,;8.24,.5,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,)|
Cc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc3OCCOc3cc2Cl)cc1
COc1cc(F)c(cc1OC)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(C)n[nH]c2n1
COc1cc(Br)c(cc1OC)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(C)n[nH]c2n1
COc1cc(C)c(cc1OC)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(C)n[nH]c2n1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNC(=O)C2)c2cn[nH]c2n1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(O)c2cn[nH]c2n1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(N2CC(CO)C2)c2cn[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(N2CC(CO)C2)c2cn[nH]c2n1
OCC1CN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCCC(N)=O)c2cn[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCCC(N)=O)c2cn[nH]c2n1
NC(=O)CCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
NC(=O)CCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCC(N)=O)c2cn[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCC(N)=O)c2cn[nH]c2n1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCC(N)=O)c2cn[nH]c2n1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2C[C@@H](O)C[C@@H](O)C2)c2cn[nH]c2n1 |r|
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2C[C@@H](O)C[C@@H](O)C2)c2cn[nH]c2n1 |r|
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCc2cn[nH]c2)c2cn[nH]c2n1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2O[C@H](O)[C@H](O)[C@@H](O)[C@@H]2O)c2cn[nH]c2n1 |r|
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2O[C@H](O)[C@H](O)[C@@H](O)[C@@H]2O)c2cn[nH]c2n1 |r|
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNC(=O)C2)c2cn[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(O)c2cn[nH]c2n1
Clc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNC(=O)C2)c2cn[nH]c2n1
Cc1n[nH]c2nc(nc(OC3CCC(O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(ccc2F)C#N)cc1 |(8.24,.5,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;7.13,2.46,;7.9,1.13,;9.44,1.13,;10.21,2.46,;11.75,2.46,;9.44,3.79,;7.9,3.79,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-7.09,3.08,;-7.09,4.62,;-1.34,1.13,;.2,1.13,)|
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCC(O)CC2)c2c(C)n[nH]c2n1 |(-8.43,3.85,;-7.09,3.08,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-5.76,-.77,;-5.76,.77,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-3.65,-.21,;-2.11,-.21,;-1.34,-1.54,;.2,-1.54,;.97,-.21,;.2,1.13,;-1.34,1.13,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;7.13,2.46,;7.9,1.13,;9.44,1.13,;10.21,2.46,;11.75,2.46,;9.44,3.79,;7.9,3.79,;5.59,-.21,;7.09,-.53,;8.24,.5,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,)|
COc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCC(O)CC2)c2c(C)n[nH]c2n1 |(-8.43,3.85,;-7.09,3.08,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-7.09,-4.62,;-5.76,-.77,;-5.76,.77,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-3.65,-.21,;-2.11,-.21,;-1.34,-1.54,;.2,-1.54,;.97,-.21,;.2,1.13,;-1.34,1.13,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;7.13,2.46,;7.9,1.13,;9.44,1.13,;10.21,2.46,;11.75,2.46,;9.44,3.79,;7.9,3.79,;5.59,-.21,;7.09,-.53,;8.24,.5,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,)|
Cc1n[nH]c2nc(nc(OC3CCC(O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2C#N)cc1 |(8.24,.5,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;7.13,2.46,;7.9,1.13,;9.44,1.13,;10.21,2.46,;11.75,2.46,;9.44,3.79,;7.9,3.79,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-7.09,-4.62,;-1.34,1.13,;.2,1.13,)|
OC1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(ccc2F)C#N)cc1 |(11.75,2.46,;10.21,2.46,;9.44,1.13,;7.9,1.13,;7.13,2.46,;7.9,3.79,;9.44,3.79,;5.59,2.46,;4.82,1.13,;3.28,1.13,;2.51,-.21,;3.28,-1.54,;4.82,-1.54,;5.85,-2.68,;7.25,-2.06,;7.09,-.53,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-7.09,3.08,;-7.09,4.62,;-1.34,1.13,;.2,1.13,)|
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCC(O)CC2)c2cn[nH]c2n1 |(-8.43,3.85,;-7.09,3.08,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-5.76,-.77,;-5.76,.77,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-3.65,-.21,;-2.11,-.21,;-1.34,-1.54,;.2,-1.54,;.97,-.21,;.2,1.13,;-1.34,1.13,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;7.13,2.46,;7.9,1.13,;9.44,1.13,;10.21,2.46,;11.75,2.46,;9.44,3.79,;7.9,3.79,;5.59,-.21,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,)|
COc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCC(O)CC2)c2cn[nH]c2n1 |(-8.43,3.85,;-7.09,3.08,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-7.09,-4.62,;-5.76,-.77,;-5.76,.77,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-3.65,-.21,;-2.11,-.21,;-1.34,-1.54,;.2,-1.54,;.97,-.21,;.2,1.13,;-1.34,1.13,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;7.13,2.46,;7.9,1.13,;9.44,1.13,;10.21,2.46,;11.75,2.46,;9.44,3.79,;7.9,3.79,;5.59,-.21,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,)|
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(C2CC2)c2cn[nH]c2n1
Cc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C2CC2)c2cn[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC)c2cn[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC)c2cn[nH]c2n1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C2CC2)c2cn[nH]c2n1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(CCCCl)c2cn[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C2CC2)c2cn[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(CCCCl)c2cn[nH]c2n1
COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC)c2c(N)n[nH]c2n1
COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC)c2c(N)n[nH]c2n1
COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Fc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNC2)c2cn[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNC2)c2cn[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNC2)c2cn[nH]c2n1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNC2)c2cn[nH]c2n1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(F)(F)F)c2cn[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(F)(F)F)c2cn[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(F)(F)F)c2cn[nH]c2n1
FC(F)(F)COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
FC(F)(F)COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2ccc(F)cc2Cl)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)c(F)c2)cc1
CCS(=O)(=O)c1ccc(Cl)cc1Cn4c(=O)[nH]c3c(Cl)c(CN2CC[C@@H](NC(=O)CN)C2)c(C(F)(F)F)cc3c4=O
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)C2SC=C(Cl)C=C2)cc1 |c:26,t:23|
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)C2SC=C(Cl)C(Cl)=C2)cc1 |c:27,t:23|
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2Cl)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2F)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)C2=CC(Br)=CCS2)cc1 |c:24,t:21|
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)C2=CSCC=C2Br)cc1 |c:25,t:21|
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)C2=CSCC=C2Cl)cc1 |c:25,t:21|
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)C2=C(Cl)SCC(Cl)=C2)cc1 |c:21,27|
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2C#N)cc1
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)cc(F)c2F)cc1
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2F)cc1
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2F)cc1
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2Cl)cc1
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)C2=CC(Cl)=C(Cl)CS2)cc1 |t:21,24|
COc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)C2=C(Cl)SCC(Cl)=C2)cc1 |c:21,27|
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCN2CCCC2=O)c2cn[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCN2CCCC2=O)c2cn[nH]c2n1
Clc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCN2CCCC2=O)c2cn[nH]c2n1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CNC2)c2cn[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CNC2)c2cn[nH]c2n1
Clc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CNC2)c2cn[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CNC2)c2cn[nH]c2n1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(F)(F)F)c2c(N)n[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(F)(F)F)c2c(N)n[nH]c2n1
Nc1n[nH]c2nc(nc(OCC(F)(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Nc1n[nH]c2nc(nc(OCC(F)(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(F)(F)F)c2c(N)n[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNC2)c2cn[nH]c2n1
NCCCOc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCCN)c2cn[nH]c2n1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCCN)c2cn[nH]c2n1
Fc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C2CC2)c2cn[nH]c2n1
Fc1ccccc1S(=O)(=O)Nc1ccc(cc1)-c1nc(C2CC2)c2cn[nH]c2n1
Cc1n[nH]c2nc(nc(OCCCN)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCCCN)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCCCN)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCCCN)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1n[nH]c2nc(nc(OCCCN)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCCN)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OCCCN)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(OC3CCC(O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1 |(8.24,.5,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;5.59,5.13,;4.82,6.46,;3.28,6.46,;2.51,7.8,;2.51,5.13,;3.28,3.79,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;.2,1.13,)|
Cc1n[nH]c2nc(nc(OC3CCC(O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |(8.24,.5,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;5.59,5.13,;4.82,6.46,;3.28,6.46,;2.51,7.8,;2.51,5.13,;3.28,3.79,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;.2,1.13,)|
Cc1n[nH]c2nc(nc(OC3CCC(O)CC3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1 |(8.24,.5,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;5.59,5.13,;4.82,6.46,;3.28,6.46,;2.51,7.8,;2.51,5.13,;3.28,3.79,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;.2,1.13,)|
Cc1n[nH]c2nc(nc(OC3CCC(O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1 |(8.24,.5,;7.09,-.53,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;5.59,5.13,;4.82,6.46,;3.28,6.46,;2.51,7.8,;2.51,5.13,;3.28,3.79,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;.2,1.13,)|
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCC(O)CC2)c2c(C)n[nH]c2n1 |(-8.43,3.85,;-7.09,3.08,;-7.09,1.54,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-5.76,-.77,;-5.76,.77,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-3.65,-.21,;-2.11,-.21,;-1.34,-1.54,;.2,-1.54,;.97,-.21,;.2,1.13,;-1.34,1.13,;2.51,-.21,;3.28,1.13,;4.82,1.13,;5.59,2.46,;4.82,3.79,;5.59,5.13,;4.82,6.46,;3.28,6.46,;2.51,7.8,;2.51,5.13,;3.28,3.79,;5.59,-.21,;7.09,-.53,;8.24,.5,;7.25,-2.06,;5.85,-2.68,;4.82,-1.54,;3.28,-1.54,)|
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCCN)c2cn[nH]c2n1
Cc1n[nH]c2nc(nc(OCCCN)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2)c2cn[nH]c2n1
Fc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2)c2cn[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2)c2cn[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2)c2cn[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2)c2cn[nH]c2n1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2)c2cn[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2)c2cn[nH]c2n1
Fc1ccccc1S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2)c2cn[nH]c2n1
NCC1(COc2nc(nc3[nH]ncc23)-c2ccc(NS(=O)(=O)c3cc(F)ccc3F)cc2)COC1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2(CN)COC2)c2cn[nH]c2n1
NCC1(COc2nc(nc3[nH]ncc23)-c2ccc(NS(=O)(=O)c3ccccc3F)cc2)COC1
NCC1(COc2nc(nc3[nH]ncc23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3F)cc2)COC1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2(CN)COC2)c2cn[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2(CN)COC2)c2cn[nH]c2n1
NCC1(COc2nc(nc3[nH]ncc23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3C#N)cc2)COC1
NCC1(COc2nc(nc3[nH]ncc23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3Cl)cc2)COC1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2(CN)COC2)c2cn[nH]c2n1
CN1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
CN1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Fc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2(F)F)c2cn[nH]c2n1
Fc1ccccc1S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2(F)F)c2cn[nH]c2n1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2(F)F)c2cn[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2(F)F)c2cn[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2(F)F)c2cn[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2(F)F)c2cn[nH]c2n1
FC1(F)CNCCC1Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
FC1(F)CNCCC1Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2(F)F)c2cn[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCN(C)CC2)c2cn[nH]c2n1
CN1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCCNC2)c2cn[nH]c2n1
Cc1n[nH]c2nc(nc(OC3CCNCC3(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCNCC3(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCNCC3(F)F)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCNCC3(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2(F)F)c2c(C)n[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2(F)F)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OC3CCNCC3(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(OC3CCNCC3(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(OC3CCNCC3(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Fc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCCNC2)c2cn[nH]c2n1
Fc1ccccc1S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCCNC2)c2cn[nH]c2n1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCCNC2)c2cn[nH]c2n1
CN1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCCNC2)c2cn[nH]c2n1
CN1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2Cl)cc1
Cc1n[nH]c2nc(nc(OCC3CNCCO3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCC3CNCCO3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNCCO2)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OCC3CNCCO3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCC3CNCCO3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCC3CNCCO3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCCNC2)c2c(C)n[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNCCO2)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OC3CCNCC3F)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCNCC3F)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCNCC3F)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCNCC3F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(OC3CCNCC3F)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2F)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OC3CCNCC3F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCNCC2F)c2c(C)n[nH]c2n1
Fc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNCCO2)c2cn[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNCCO2)c2cn[nH]c2n1
Fc1ccccc1S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNCCO2)c2cn[nH]c2n1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNCCO2)c2cn[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNCCO2)c2cn[nH]c2n1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Fc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNCCO2)c2cn[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNCCO2)c2cn[nH]c2n1
Cc1n[nH]c2nc(nc(OCC3CNCCO3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
CN1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC2CNCCO2)c2cn[nH]c2n1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2ccccc2Cl)cc1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2ccc(F)cc2Cl)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCCNC2)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OC3CCCNC3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(OC3CCCNC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCCNC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1n[nH]c2nc(nc(OC3CCCNC3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cccc(F)c2Cl)cc1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2Cl)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(C)C)c2c(N)n[nH]c2n1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2F)cc1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2F)cc1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)sc2Cl)cc1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(C)C)c2c(N)n[nH]c2n1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CC(C)Oc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(C)C)c2c(N)n[nH]c2n1
CC(C)COc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2Cl)cc1
Cc1n[nH]c2nc(nc(OC3CCCNC3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCCNC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCN(CCF)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCN(CCF)CC2)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OC3CCN(CCF)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1n[nH]c2nc(nc(OC3CCN(CCF)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCN(CC2)C(C)C)c2c(C)n[nH]c2n1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCN(CCF)CC2)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OC3CCN(CCF)CC3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
CC(C)COc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Nc1n[nH]c2nc(nc(OCC3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCN(CC2)C(C)C)c2c(C)n[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(CO)CO)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OCC(CO)CO)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCC(CO)CO)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Cc1n[nH]c2nc(nc(OCC(CO)CO)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(F)(F)CN)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OCC(F)(F)CN)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Cc1n[nH]c2nc(nc(OCC(F)(F)CN)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(F)(F)CN)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OCC(F)(F)CN)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCC(F)(F)CN)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCC(CO)CO)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCC(CO)CO)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OCC(CO)CO)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCC(CO)CO)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(NCC(F)(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1n[nH]c2nc(nc(NCC(F)(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(NCC(F)(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2nc(nc(NCC(F)(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(OCCCO)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCCCO)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OCCCO)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OCCCO)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(OC3CCN(CC(F)(F)F)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCN(CC(F)(F)F)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCN(CC(F)(F)F)CC2)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OC3CCN(CC(F)(F)F)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2Cl)cc1
Cc1n[nH]c2nc(nc(OC3CCN(CC(F)(F)F)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCN(CC(F)(F)F)CC2)c2c(C)n[nH]c2n1
Cc1n[nH]c2nc(nc(OC3CCN(CC(F)(F)F)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2nc(nc(OCCCO)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Cc1n[nH]c2nc(nc(OCCCO)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COCCCOc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2Cl)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCN(CC2)C2CCC2)c2cn[nH]c2n1
COCCCN1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Fc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCN(CC2)C2CC2)c2cn[nH]c2n1
COCCCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCN(CC3)C3CCC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2Cl)cc1
CCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
CCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
CCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2F)cc1
CCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COCCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COCCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
COCCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
CCN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
CCN1CCCC(C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CCN1CCCC(C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2Cl)cc1
CCN1CCCC(C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
CCN1CCCC(C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
CCN1CCCC(C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
CCN1CCCC(C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CCN1CCCC(C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2F)cc1
CCCOc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
CCOc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)c(F)c1
OC1CCN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1
OC1CN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1
OC1CN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)c(F)c1
OC1CCN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)c(F)c1
OC1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)c(F)c1 |(2.51,7.8,;3.28,6.46,;4.82,6.46,;5.59,5.13,;4.82,3.79,;3.28,3.79,;2.51,5.13,;5.59,2.46,;4.82,1.13,;3.28,1.13,;2.51,-.21,;3.28,-1.54,;4.82,-1.54,;5.85,-2.68,;7.25,-2.06,;7.09,-.53,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;-2.11,2.46,;.2,1.13,)|
OC1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1 |(2.51,7.8,;3.28,6.46,;4.82,6.46,;5.59,5.13,;4.82,3.79,;3.28,3.79,;2.51,5.13,;5.59,2.46,;4.82,1.13,;3.28,1.13,;2.51,-.21,;3.28,-1.54,;4.82,-1.54,;5.85,-2.68,;7.25,-2.06,;7.09,-.53,;5.59,-.21,;.97,-.21,;.2,-1.54,;-1.34,-1.54,;-2.11,-.21,;-3.65,-.21,;-4.42,-1.54,;-5.19,-2.87,;-3.09,-2.31,;-5.76,-.77,;-5.76,.77,;-7.09,1.54,;-7.09,3.08,;-8.43,.77,;-8.43,-.77,;-7.09,-1.54,;-7.09,-3.08,;-1.34,1.13,;-2.11,2.46,;.2,1.13,)|
OCC1CN(C1)c1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1
Fc1cc(ccc1NS(=O)(=O)c1cc(Cl)ccc1F)-c1nc(OC2CNC2)c2cn[nH]c2n1
Fc1cc(ccc1NS(=O)(=O)c1cc(Cl)ccc1F)-c1nc(C2CC2)c2cn[nH]c2n1
CC(C)Oc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Cc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Cc1n[nH]c2nc(nc(N3CCC4(COC4)C3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
CCOc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(N)n[nH]c2n1
Cc1cc(cc(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(N)n[nH]c2n1)C#N
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(N)n[nH]c2n1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2C#N)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cccc(c2)C#N)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2ccc3OCCCOc3c2)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc3OCCCOc3cc2Br)cc1
Cc1nn(C)c(Cl)c1S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(N)n[nH]c2n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(N)n[nH]c2n1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2Cl)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)sc2Cl)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C)c2c(N)n[nH]c2n1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C)c2c(N)n[nH]c2n1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2ccc(F)c(c2)C#N)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2C#N)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cccc(c2)C#N)cc1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C)c2c(N)n[nH]c2n1
Cc1ccc(cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(C)c2c(N)n[nH]c2n1)C#N
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cccc(F)c2C#N)cc1
Cc1nn(C)c(Cl)c1S(=O)(=O)Nc1ccc(cc1)-c1nc(C)c2c(N)n[nH]c2n1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc3OCCCOc3cc2Cl)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc3OCCCOc3cc2Br)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2c(Cl)ccc3OCCCOc23)cc1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2Cl)cc1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2Cl)cc1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2Cl)cc1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2F)cc1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2ccc(F)cc2Cl)cc1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2F)cc1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C2CC2)c2c(N)n[nH]c2n1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2ccccc2C#N)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C)c2cn[nH]c2n1
Cc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2ccc(F)c(c2)C#N)cc1
Cc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(c2)C#N)cc1
Cc1ccc(cc1S(=O)(=O)Nc1ccc(cc1)-c1nc(C)c2cn[nH]c2n1)C#N
Cc1nc(nc2[nH]nc(N3CCC4(COC4)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1nc(nc2[nH]nc(N3CC4(COC4)C3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1nc(nc2[nH]nc(N3CCCC4(COC4)C3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Nc1n[nH]c2nc(nc(C3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)sc2Cl)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2Cl)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2F)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2ccc(F)cc2Cl)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)sc2Cl)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2Cl)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2F)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2Cl)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2F)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2F)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
COCCc1n[nH]c2nc(nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2F)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
COc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C2CC2)c2c(N)n[nH]c2n1
COCCc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2C#N)cc1
COc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(N)n[nH]c2n1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cccc(F)c2F)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2ccccc2Cl)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2ccc(F)cc2Cl)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(N)n[nH]c2n1
Cc1nc(nc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2c(F)ccc(Cl)c2F)cc1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2c(F)ccc(Cl)c2F)cc1
Cc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2ccccc2C(N)=O)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1F)-c1ncc2c(C)n[nH]c2n1
COc1cc(ccc1NS(=O)(=O)c1cc(Cl)ccc1Cl)-c1ncc2c(C)n[nH]c2n1
Cc1nc(nc2[nH]nc(NC(=O)C3CC(O)C3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1 |(3.11,2.06,;2.34,.73,;.8,.73,;.03,-.61,;.8,-1.94,;2.34,-1.94,;3.37,-3.09,;4.77,-2.46,;4.61,-.93,;5.7,.16,;7.19,-.24,;7.59,-1.72,;8.28,.85,;9.82,.85,;9.82,2.39,;10.91,3.48,;8.28,2.39,;3.11,-.61,;-1.51,-.61,;-2.28,-1.94,;-3.82,-1.94,;-4.59,-.61,;-6.13,-.61,;-6.9,-1.94,;-5.57,-2.71,;-7.67,-3.27,;-8.24,-1.17,;-8.24,.37,;-9.57,1.14,;-9.57,2.68,;-10.91,.37,;-10.91,-1.17,;-9.57,-1.94,;-9.57,-3.48,;-3.82,.73,;-2.28,.73,)|
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(NC(=O)C3CC3)n[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(NC(=O)C3CCCC3)n[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(NC(=O)C3CCCCC3)n[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(NC(=O)c3cccc(Cl)c3Cl)n[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(NC(=O)C3CCOCC3)n[nH]c2n1
Clc1ccc(cc1)C(=O)Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(NC(=O)Cc3ccccc3)n[nH]c2n1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(NC(=O)c3ccsc3)n[nH]c2n1
Cc1nc(nc2[nH]nc(NC(=O)C3CCOCC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(NC(=O)C3CCNCC3)n[nH]c2n1
Cc1nc(nc2[nH]nc(NCC3CCOCC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(NCc3ccccc3)n[nH]c2n1
Nc1n[nH]c2cc(nc(O)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Nc1n[nH]c2cc(nc(O)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Oc1nc(cc2[nH]nc(NS(=O)(=O)c3cc(Cl)ccc3Cl)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Nc1n[nH]c2cc(nc(O)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(N)c2cn1
Nc1n[nH]c2cc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Nc1n[nH]c2cc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Nc1n[nH]c2cc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Nc1n[nH]c2cc(ncc12)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2Cl)cc1
Nc1n[nH]c2cc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)sc2Cl)cc1
Nc1n[nH]c2cc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1n[nH]c2cc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1n[nH]c2cc(ncc12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2cc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]ncc2cn1
Cc1ccc(cc1S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]ncc2cn1)C#N
Clc1ccc(CNC(=O)Nc2n[nH]c3nc(ncc23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3Cl)cc2)cc1
Clc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncc2c(NC(=O)NCC3CCOCC3)n[nH]c2n1
Nc1n[nH]c2nc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(N)c2c(n1)C(F)(F)F
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
COc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(N)c2c(n1)C(F)(F)F
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2cc(Cl)sc2Cl)cc1
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2F)cc1
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2Cl)cc1
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2ccc(F)cc2Cl)cc1
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2F)cc1
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(N)c2c(n1)C(F)(F)F
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(N)c2c(n1)C(F)(F)F
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2ccccc2Cl)cc1
Nc1n[nH]c2cc(nc(c12)C(F)(F)F)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2F)cc1
Cc1n[nH]c2cc(nc(OC3CCN(CC3)C3CC3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Cc1n[nH]c2cc(nc(OC3CCN(CC3)C3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
CC(C)N1CC(COc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3F)cc2)C1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OCC2CN(C2)C(C)C)n1
CC(C)N1CC(COc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(C)ccc3F)cc2)C1
CC(C)N1CC(COc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3Cl)cc2)C1
CC(C)N1CC(COc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3ccccc3F)cc2)C1
CC(C)N1CC(COc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(F)ccc3F)cc2)C1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OCC2CN(C2)C(C)C)n1
CCCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
CCCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
CCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2cc(nc(Oc3ccc(O)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2cc(nc(Oc3ccc(O)nc3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(Oc2ccc(O)nc2)n1
Cc1n[nH]c2cc(nc(Oc3ccc(O)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2cc(nc(Oc3ccc(O)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1n[nH]c2cc(nc(Oc3ccc(O)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2cc(nc(Oc3ccc(O)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CCCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2Cl)cc1
CCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
CCCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
CCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2F)cc1
CCCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2F)cc1
CCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2Cl)cc1
CCCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2Cl)cc1
CCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2F)cc1
CCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2Cl)cc1
Cc1n[nH]c2cc(nc(OC3CCOCC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2cc(nc(OC3CCOCC3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Cc1n[nH]c2cc(nc(OC3CCOCC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
CN1C(C)(C)CC(CC1(C)C)Oc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN1C(C)(C)CC(CC1(C)C)Oc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
CN1C(C)(C)CC(CC1(C)C)Oc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
CN1C(C)(C)CC(CC1(C)C)Oc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
COc1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(F)ccc3F)cc2)cn1
COc1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3Cl)cc2)cn1
COc1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3ccccc3F)cc2)cn1
Cc1n[nH]c2cc(nc(OC3CCOCC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2cc(nc(OC3CC(C)(C)NC(C)(C)C3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2cc(nc(OC3CC(C)(C)NC(C)(C)C3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OC2CC(C)(C)NC(C)(C)C2)n1
Cc1n[nH]c2cc(nc(OC3CC(C)(C)NC(C)(C)C3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OC2CC(C)(C)NC(C)(C)C2)n1
CN1C(C)(C)CC(CC1(C)C)Oc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OC2CC(C)(C)N(C)C(C)(C)C2)n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OC2CC(C)(C)N(C)C(C)(C)C2)n1
COc1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3F)cc2)cn1
Cc1n[nH]c2cc(nc(OC3CCN(CC3)C3CCC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1n[nH]c2cc(nc(OC3CCN(CC3)C3CCC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Cc1n[nH]c2cc(nc(OC3CCN(CC3)C3CCC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2cc(nc(OC3CCN(CC3)C3CCC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2Cl)cc1
Cc1n[nH]c2cc(nc(OC3CCN(CC3)C3CCC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2F)cc1
Cc1n[nH]c2cc(nc(OC3CCN(CC3)C3CCC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)c(F)cc2Cl)cc1
COc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OC2CCN(CC2)C2CCC2)n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OC2CCN(CC2)C2CCC2)n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OC2CCN(CC2)C2CCC2)n1
Cc1n[nH]c2cc(nc(OC3CC(C)(C)NC(C)(C)C3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CN1C(C)(C)CC(CC1(C)C)Oc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
CC(=O)N1CCC(CC1)Oc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2cc(nc(OC3CC(C)(C)NC(C)(C)C3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
Cc1n[nH]c2cc(nc(OC3CC(C)(C)NC(C)(C)C3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2Cl)cc1
Cc1n[nH]c2cc(nc(OC3CCC(=O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2cc(nc(OC3CCC(=O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(Oc2ccc(OC)nc2)n1
COc1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(C)ccc3C#N)cc2)cn1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(Oc2ccc(OC)nc2)n1
COc1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(C)ccc3F)cc2)cn1
Cc1n[nH]c2cc(nc(Oc3ccnc(O)c3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Cc1n[nH]c2cc(nc(Oc3ccnc(O)c3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2cc(nc(Oc3ccnc(O)c3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OC2CCN(CC2)C(C)=O)n1
CC(=O)N1CCC(CC1)Oc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OC2CCN(CC2)C(C)=O)n1
CC(=O)N1CCC(CC1)Oc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2F)cc1
CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
CCCOc1nc(cc2[nH]nc(N)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(Oc2ccnc(OC)c2)n1
COc1cc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3F)cc2)ccn1
COc1cc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(C)ccc3C#N)cc2)ccn1
COc1cc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(F)ccc3F)cc2)ccn1
COc1cc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3Cl)cc2)ccn1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(Oc2ccnc(OC)c2)n1
COc1cc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3ccccc3F)cc2)ccn1
COc1cc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(C)ccc3F)cc2)ccn1
CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(OC)ccc2Cl)cc1
CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(Oc2ccc(N)nc2)n1
Cc1n[nH]c2cc(nc(Oc3ccc(N)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2cc(nc(Oc3ccc(N)nc3)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(Oc2ccc(N)nc2)n1
Cc1n[nH]c2cc(nc(Oc3ccc(N)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2cc(nc(Oc3ccc(N)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
Cc1n[nH]c2cc(nc(Oc3ccc(N)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Cc1n[nH]c2cc(nc(Oc3ccc(N)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2C#N)cc1
CN(C)C(=O)CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(C)ccc2F)cc1
CN(C)C(=O)CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN(C)C(=O)CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OCCC(=O)N(C)C)n1
CN(C)C(=O)CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
CN(C)C(=O)CCOc1nc(cc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(OCCC(=O)N(C)C)n1
CN(C)c1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(C)ccc3F)cc2)cn1
CN(C)c1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3F)cc2)cn1
CN(C)c1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3ccccc3F)cc2)cn1
CN(C)c1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3Cl)cc2)cn1
CN(C)c1ccc(Oc2nc(cc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(F)ccc3F)cc2)cn1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(Oc2ccc(nc2)N(C)C)n1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cc2[nH]nc(C)c2c(Oc2ccc(nc2)N(C)C)n1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)C=C)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)N2CCCC2)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccc(cc2)C#N)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccc(CN)cc2)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)C(C)C)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)N2CCCCC2)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cccnc2)cc1
CN(C)CCOc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN(C)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN(C)CCCOc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN(C)CCCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1cnc(NS(=O)(=O)c2cc(Cl)ccc2F)nc1
Cc1n[nH]c2nc(nc(NCc3ccncc3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(CNS(=O)(=O)c2cc(Cl)ccc2F)o1
CN(C)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccncc2F)cc1
CN(C)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccc(N)nc2)cc1
CC(C)N1CC(C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN(CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1)C=O
COc1ccncc1S(=O)(=O)Nc1ccc(cc1)-c1nc(NCCN(C)C)c2c(C)n[nH]c2n1
CN(CCO)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccccn2)cc1
CN(CCO)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cccnc2)cc1
CN(CCO)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN(C)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cccnc2)cc1
CN(C)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2ccccn2)cc1
CC(C)N1CC(C1)Nc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(NCCN3CCOCC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COc1ccnc(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(NCCN(C)C)c2c(C)n[nH]c2n1
CC(C)N1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1
Cc1n[nH]c2nc(nc(O[C@@H]3CCNC[C@@H]3F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
CN(C)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(ccn2)C(F)(F)F)cc1
CCN(CC)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(NCCN3CCCC3)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CN1CC(C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
CN(C)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1
Cc1n[nH]c2nc(nc(O[C@@H]3CNC[C@@H]3F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
CN(C)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Cc1n[nH]c2nc(nc(O[C@H]3CCNC[C@H]3F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
Cc1n[nH]c2nc(nc(O[C@H]3CCNC[C@@H]3F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
Cc1n[nH]c2nc(nc(O[C@H]3CCNC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
Cc1n[nH]c2nc(nc(O[C@@H]3CNCC3(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
Cc1n[nH]c2nc(nc(O[C@@H]3CCN(CCO)C[C@@H]3F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
Cc1n[nH]c2nc(nc(O[C@@H]3CCNC[C@H]3F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
CCN1C[C@H](F)[C@@H](C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
CN1C[C@H](F)[C@@H](C1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |
CN1CC[C@@H](Oc2nc(nc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(ccn3)C(F)(F)F)cc2)[C@@H](F)C1 |r|
CN1CC[C@@H](Oc2nc(nc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3ccccn3)cc2)[C@@H](F)C1 |r|
CN1CC[C@@H](Oc2nc(nc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3F)cc2C)[C@@H](F)C1 |r|
CN1CC[C@@H](Oc2nc(nc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3F)c(F)c2)[C@@H](F)C1 |r|
Cc1n[nH]c2nc(nc(O[C@@H]3CCN(CCO)CC3(F)F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r|
CN(CCO)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(ccn2)C(F)(F)F)cc1
CC(C)Oc1ccnc(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(NCCN(C)C)c2c(C)n[nH]c2n1
CN(C)CC(F)(F)CNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN(C)CC(F)(F)CNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(ccn2)C(F)(F)F)cc1
CN(CCO)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1
CN1CCC(CC1)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)c(F)c1
COc1ccnc(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(OC2CCN(CC2)C(C)C)c2c(C)n[nH]c2n1
CN(C)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)c(F)c1
CN(C)CCNc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)c(Cl)c1
CN(CCO)CCOc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
COc1cc(ccc1NS(=O)(=O)c1cc(F)ccc1F)-c1nc(NCCN(C)C)c2c(C)n[nH]c2n1
CN(C)CCN(C)c1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CCN(CC)CC=Cc1[nH]c(=O)c2c3n(C)c(Nc4c(Cl)cccc4Cl)nc3ccc2c1C |w:6.5|
CC(C)(N)c1ccc(cc1)-c1nc2ccccc2nc1-c1ccccc1
OC1CCC(CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1 |(68.02,-2.5,;66.48,-2.49,;65.7,-3.83,;64.16,-3.83,;63.39,-2.48,;64.16,-1.15,;65.7,-1.16,;61.85,-2.48,;61.08,-3.82,;59.54,-3.83,;58.77,-5.16,;59.54,-6.5,;61.08,-6.49,;62.1,-7.64,;63.51,-7.03,;63.36,-5.5,;61.86,-5.17,;57.23,-5.15,;56.46,-6.49,;54.91,-6.48,;54.15,-5.14,;52.61,-5.13,;51.84,-6.46,;53.17,-7.23,;51.83,-8,;50.29,-6.47,;49.52,-5.14,;47.98,-5.14,;47.2,-3.81,;47.22,-6.47,;47.99,-7.8,;49.53,-7.8,;50.3,-9.14,;51.07,-10.47,;54.92,-3.81,;56.46,-3.81,)|
O[C@H]1CC[C@@H](CC1)Oc1nc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1 |r,wU:4.7,wD:1.0,(43,-11.27,;41.45,-11.27,;40.68,-9.93,;39.13,-9.93,;38.37,-11.26,;39.14,-12.6,;40.68,-12.61,;36.83,-11.26,;36.06,-12.6,;34.52,-12.6,;33.75,-13.93,;34.52,-15.27,;36.05,-15.27,;37.07,-16.42,;38.48,-15.8,;38.34,-14.27,;36.83,-13.94,;32.21,-13.93,;31.43,-15.26,;29.89,-15.26,;29.13,-13.92,;27.59,-13.91,;26.81,-15.24,;28.15,-16.01,;26.81,-16.78,;25.27,-15.25,;24.5,-13.91,;22.96,-13.92,;22.18,-12.58,;22.2,-15.25,;22.96,-16.57,;24.5,-16.58,;25.27,-17.91,;29.9,-12.59,;31.44,-12.59,)|
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(O[C@H]2CC[C@H](O)CC2)c2c(C)n[nH]c2n1 |r,wU:23.24,wD:26.28,(46.54,-10.36,;45.77,-11.7,;46.55,-13.04,;45.79,-14.37,;46.56,-15.69,;48.1,-15.7,;48.87,-17.03,;48.87,-14.36,;48.1,-13.03,;50.41,-14.36,;51.74,-15.13,;50.41,-15.9,;51.18,-13.03,;52.72,-13.03,;53.49,-14.38,;55.03,-14.38,;55.81,-13.05,;55.03,-11.7,;53.49,-11.71,;57.34,-13.05,;58.11,-11.72,;59.65,-11.72,;60.42,-10.38,;61.96,-10.38,;62.73,-9.05,;64.28,-9.05,;65.05,-10.39,;66.59,-10.39,;64.27,-11.72,;62.73,-11.72,;60.43,-13.06,;61.93,-13.39,;63.08,-12.37,;62.08,-14.92,;60.67,-15.54,;59.65,-14.39,;58.11,-14.39,)|
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1nc(C2CC2)c2cn[nH]c2n1
Nc1n[nH]c2nc(ncc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)c(F)cc2F)cc1
Cc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cnc2c(N)n[nH]c2n1
COc1ccc(F)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cnc2c(N)n[nH]c2n1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Cc1ccc(C#N)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cnc2c(N)n[nH]c2n1
Cc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
COc1cc(O)ccc1\C=N\NC(=O)Cc1cccc(O)c1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1ccc2c(N)n[nH]c2c1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cc(Br)ccc2Cl)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cc(Br)ccc2F)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2F)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cccc3ccccc23)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2cc(Cl)sc2Cl)cc1
COc1ccc(Cl)c(c1)S(=O)(=O)Nc1ccc(cc1)-c1cnc2c(N)n[nH]c2n1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2ccc(cc2Cl)C(F)(F)F)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)Cc2cc(F)ccc2F)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2ccc(Br)s2)cc1
Cn1cc(c(n1)C(F)(F)F)S(=O)(=O)Nc1ccc(cc1)-c1ccc2c(N)n[nH]c2c1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2ccco2)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cc(Cl)sc2Cl)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2ccccc2)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2ccccc2Cl)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2Cl)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2C#N)cc1
Cc1ccc(cc1S(=O)(=O)Nc1ccc(cc1)-c1ccc2c(N)n[nH]c2c1)C#N
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2C#N)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cc(ccc2F)C(F)(F)F)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2ccccc2F)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cccc(F)c2F)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1
Nc1n[nH]c2nc(cnc12)-c1ccc(NS(=O)(=O)c2ccc(Cl)cc2Cl)cc1
CCCCCS(=O)(=O)Nc1ccc(cc1)-c1ccc2c(N)n[nH]c2c1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)C2CCCCC2)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)C2CC2)cc1
Nc1n[nH]c2cc(ccc12)-c1ccc(NS(=O)(=O)Cc2ccccc2)cc1
Cc1n[nH]c(C)c1S(=O)(=O)Nc1ccc(cc1)-c1ccc2c(N)n[nH]c2c1
CN(C)c1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CCCC1
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CCOCC1C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CCC1C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)[C@H](C)C(=O)N(C)C
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CCC[C@@H]1C(=O)N(C)C
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CC[C@@H](C1)C(N)=O
CNC(=O)[C@@H](C)N(C)Cc1cc2c(Nc3cccc(Cl)c3F)ncnc2cc1OC
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)C1(CCN(CC1)C(C)C)C(N)=O
COCCN1CC(C1)(N(C)Cc1cc2c(Nc3cccc(Cl)c3F)ncnc2cc1OC)C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)[C@@H](CO)C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CCC[C@H]1CC(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CCC[C@@H]1C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)[C@@H](C)C(N)=O
COCCN(Cc1cc2c(Nc3cccc(Cl)c3F)ncnc2cc1OC)[C@@H](C)C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CCCC[C@@H]1C(N)=O
CNC(=O)[C@H]1CCCN1Cc1cc2c(Nc3cccc(Cl)c3F)ncnc2cc1OC
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(CCN(C)C)[C@@H](C)C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN[C@H](C)C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)C1(CCN(C)CC1)C(N)=O
COCC[C@H](N(C)Cc1cc2c(Nc3cccc(Cl)c3F)ncnc2cc1OC)C(N)=O
COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1CN1CCC[C@H]1C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C(C)C)[C@@H](C)C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)[C@H](C)C(N)=O
COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1CN1CCC[C@@H]1C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CC(C1)C(N)=O
CO[C@@H]1C[C@@H](N(Cc2cc3c(Nc4cccc(Cl)c4F)ncnc3cc2OC)C1)C(N)=O
COC[C@H](N(C)Cc1cc2c(Nc3cccc(Cl)c3F)ncnc2cc1OC)C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)CC(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)C1(CN(C)C1)C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)C1(CN(C1)C(C)C)C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CCN(C)CC1C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)C1CCNC1=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN1CCC[C@H]1C(N)=O
COc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1CN(C)[C@@H](CN(C)C)C(N)=O
Oc1ccc(cc1)-c1ccc(cc1)-c1n[nH]c-2c1Cc1cc(ccc-21)C(=O)NCc1ccncc1
O[C@H]1CC[C@@H](CC1)NC(=O)c1ccc-2c(Cc3c(n[nH]c-23)-c2ccc(cc2)-c2ccc(O)cc2)c1 |wU:4.7,wD:1.0,(19.77,-1.9,;21.02,-1.01,;22.42,-1.66,;23.69,-.77,;23.53,.76,;22.14,1.41,;20.89,.52,;24.79,1.65,;26.19,1.01,;26.33,-.53,;27.44,1.9,;27.3,3.44,;28.55,4.33,;29.95,3.7,;30.1,2.15,;31.61,1.81,;32.4,3.14,;33.83,3.77,;33.68,5.31,;32.16,5.65,;31.37,4.31,;35.16,2.99,;35.15,1.44,;36.46,.66,;37.81,1.42,;37.82,2.96,;36.49,3.74,;39.13,.64,;39.12,-.9,;40.44,-1.67,;41.78,-.91,;43.11,-1.69,;41.78,.63,;40.46,1.4,;28.85,1.26,)|
COc1cc(ccc1N)-c1ccc2c(Nc3ccc(cc3NC2=O)C(C)(C)C(=O)Nc2ccc(cc2)N2CCOCC2)c1
COc1cc(ccc1N)-c1ccc2c(Nc3ccc(CC(=O)Nc4ccc(cc4)N4CCOCC4)cc3NC2=O)c1
Nc1nnc2c3cc(-c4ccccc4)c(nc3ccn12)-c1ccc(CN2CCC(CC2)c2nnc([nH]2)-c2ccccn2)cc1
OCCNCc1nnc2c3cc(-c4ccccc4)c(nc3ccn12)-c1ccc(CN2CCC(CC2)c2nnc([nH]2)-c2ccccn2)cc1
CN1CCN(Cc2nnc3c4cc(-c5ccccc5)c(nc4ccn23)-c2ccc(CN3CCC(CC3)c3nnc([nH]3)-c3ccccn3)cc2)CC1
ClCc1nnc2c3cc(-c4ccccc4)c(nc3ccn12)-c1ccc(CN2CCC(CC2)c2nnc([nH]2)-c2ccccn2)cc1
Cc1nnc2c3cc(-c4ccccc4)c(nc3ccn12)-c1ccc(CN2CCC(CC2)c2nnc([nH]2)-c2ccccn2)cc1
C(N1CCC(CC1)c1nnc([nH]1)-c1ccccn1)c1ccc(cc1)-c1nc2ccn3cnnc3c2cc1-c1ccccc1
NC(=O)Nc1nnc2c3cc(-c4ccccc4)c(nc3ccn12)-c1ccc(CN2CCC(CC2)c2nnc([nH]2)-c2ccccn2)cc1
S=c1[nH]nc2c3cc(-c4ccccc4)c(nc3ccn12)-c1ccc(CN2CCC(CC2)c2nnc([nH]2)-c2ccccn2)cc1
O=c1[nH]nc2c3cc(-c4ccccc4)c(nc3ccn12)-c1ccc(CN2CCC(CC2)c2nnc([nH]2)-c2ccccn2)cc1
Cn1c2nc(Nc3ccc4[nH]ccc4c3)ncc2cc(c1=O)S(=O)(=O)c1ccc(F)cc1F
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)NC)OC
c1ccc(cc1)c2cc3c(c[nH]c3nc2)c4ccc(cc4)C(=O)O
c1ccc2cc(ccc2c1)c3cc4c(c[nH]c4nc3)c5ccc(cc5)CC(=O)O
COC(=O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1ccccc1
CC(=O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1ccccc1
NCc1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1ccccc1
c1[nH]c2ncc(cc2c1-c1ccc(cc1)-c1nnn[nH]1)-c1ccccc1
CCc1cc(ccc1C(O)=O)-c1c[nH]c2ncc(cc12)-c1ccccc1
CC(C)Cc1cc(ccc1C(=O)O)c2c[nH]c3c2cc(cn3)c4ccccc4
OC(=O)c1ccc(cc1C1CCCC1)-c1c[nH]c2ncc(cc12)-c1ccccc1
CC(C(O)=O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1ccc2ccccc2c1
CC(C)(C(O)=O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1ccc2ccccc2c1
CC(C)(C(O)=O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1ccccc1
CC(C)(C(O)=O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1cccc(c1)C#N
O=C1OC(\C=C\c2ccccc2)=N/C/1=C\c1cccnc1 |c:12|
NCCn1cc(-c2cc(-c3cc4ccccc4s3)c3[nH]ncc3c2)c2nc(N)ncc12
CC1(C)C(=O)N([C@H]2CCc3c2cccc3O)c2nc(Nc3ccccc3)ncc12 |r|
N[C@H](CNc1nnc(s1)-c1ccc2cnccc2c1)Cc1ccc(cc1)C(F)(F)F |r|
O=C(Cc1ccccc1)Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(Nc2cccc(c2)N2CCOCC2)n1
Nc1ncnc2n[nH]c(Nc3ccc(F)cc3)c12
Nc1n[nH]c2cc(ccc12)-c1ccnc(N)n1
CNc1cncc(n1)-c1c[nH]c(=O)c(NC(=O)c2ccc(cc2)N2CCC[C@H]2CN2CCCC2)c1 |r|
CC(C)(C)c1cc(c(s1)NC(=O)Nc2cccc(c2Cl)Cl)C(=O)N3CCC(=O)N(CC3)CCN(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(OCCN2CCOCC2)c2ccccc12)C(C)(C)C
C[C@@H]1CCC(CN1)N1CC[C@@]2(C1)CN(C(=O)c1cc3ccc(F)cc3[nH]1)c1ccccc21 |r|
COc1ccc(cc1)N1Cc2cnc(Nc3ccccc3)nc2N([C@@H]2CC[C@@H](O)C2)C1=O |r|
CCCNC(=O)c1ccc(Nc2nc(NCC(F)(F)F)c3cc[nH]c3n2)cc1
CC1(C)OCC(=O)Nc2cc(Nc3nc(NCC(F)(F)F)c4occc4n3)ccc12
c1ccc2c(c1)nc(s2)C(C#N)c3ccnc(n3)NCCc4cccnc4
COc1ccc(cc1)N1Cc2cnc(Nc3ccc(F)cc3)nc2N(C2CC[C@@H](O)C2)C1=O
C[C@@H]1C[C@H]2CN1CCn1[nH]c3c(cccc3c1=O)-c1nc3c(O2)cccc3[nH]c1=O
CC(C)NCc1ccc(Nc2cc(n[nH]2)-c2ccc(cc2)-c2ccc(O)cc2O)cc1
Clc1cc2NC(=O)Nc3cnc(C#N)c(OCCCCOc2cc1NCc1cncs1)n3
OC(=O)c1ccc2nc(-c3ccccc3)c(nc2c1)-c1ccc(CN2CCC(CC2)n2c3ccccc3[nH]c2=O)cc1
OC(=O)c1ccc2nc(-c3ccc(CN4CCC(CC4)n4c5ccccc5[nH]c4=O)cc3)c(nc2c1)-c1ccccc1
O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(cc2)-c2nc3ccc(cc3nc2-c2ccccc2)-c2nnn[nH]2)CC1
CCN(CC)CCNC(=O)c1ccc2nc(-c3ccc(CN4CCC(CC4)n4c5ccccc5[nH]c4=O)cc3)c(nc2c1)-c1ccccc1
CCN(CC)CCNC(=O)c1ccc2nc(-c3ccccc3)c(nc2c1)-c1ccc(CN2CCC(CC2)n2c3ccccc3[nH]c2=O)cc1
O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(cc2)-c2nc3cc(ccc3nc2-c2ccccc2)-c2nnn[nH]2)CC1
Cc1ccc(cc1-c1ccc2c(noc2c1)C1CCNCC1)C(=O)Nc1cccc(c1)N1CCOCC1
Cc1nnc(o1)-c1ccc(c(C)c1)-c1cc(ccc1C)C(=O)Nc1cccc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)N2CCCC2)cc1-c1ccc2c(noc2c1)C1CCNCC1
Cc1nnc(o1)-c1ccc(c(C)c1)-c1cc(NC(=O)c2ccnc(c2)N2CCCC2)ccc1C
Cc1ccc(cc1-c1ccc2c(noc2c1)C1CCNCC1)C(=O)NC1CC1
Cc1nnc(o1)-c1ccc(c(C)c1)-c1cc(ccc1C)C(=O)NC1CC1
Cc1ccc(cc1-c1ccc2c(c1)nnn(CC1CC1)c2=O)C(=O)NC1CC1
Cc1ccc(cc1-c1ccc2ccncc2c1)C(=O)NC1CC1
Cc1ccc(cc1-c1ccc(cc1)C(=O)NCC1CC1)C(=O)NC1CC1
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(c2)-c2ccc(cc2C)-c2nnc(C)o2)CC1
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(c2)-c2ccc3ccncc3c2)CC1
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(c2)-c2ccc3c(N)noc3c2)CC1
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(c2)-c2ccc(cc2)-c2csc(N)n2)CC1
C[C@@H]1CCN(C[C@@H]1N(C)c1ncnc2[nH]ccc12)C(=O)CC#N |r|
[#6]C1([#6])[#6]-2=[#6]-3-[#6]=[#6]-4-[#6](-[#6]-[#6]-[#7+]-5=[#6]-4C([#6])([#6])c4cc(-[#6]-[#6](=O)-[#7]-[#6]-[#6]-[#6]-[#6]-[#6@@H](-[#7]-[#6](=O)-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6]-[#6]-[#6]-[#6]-[#6]-[#7]-[#6](=O)-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#7]-[#6]-[#6]-[#7]S(=O)(=O)c6cccc7cnccc67)-[#6](-[#7])=O)ccc-54)-[#8]-[#6]-3-[#6]-[#6]-[#7]-2-c2ccc(cc12)S([#6])(=O)=O |r,c:3,5,10|
COc1ccc(NC(=O)Cc2nc(cs2)-c2ccc(cc2)[N+]([O-])=O)cc1
CC(C)(C)Nc1c(Nc2ccnc(Nc3ccc(cc3)-c3ccncc3)n2)c(=O)c1=O
COc1cc2CCN=C(c3ccc(Cl)c(Cl)c3)c2cc1Cl |t:7|
COc1cc2CCN=C(c3cccc(Cl)c3)c2cc1Cl |t:7|
c1cc(c(cc1Cl)CNc2ncc(c(n2)NC3CCCC3)C(=O)NCCCN4CCOC4=O)Cl
Clc1ccc(Cl)c(CNc2ncc(C(=O)NCCCN3CCCC3=O)c(NC3CCCC3)n2)c1
COc1ccccc1CNc2ncc(c(n2)NC3CCCC3)C(=O)NCCCN4CCCC4=O
COc1ccc(CCNc2ncc(C(=O)NCCCN3CCCC3=O)c(NC3CCCC3)n2)cc1OC
Cc1c(F)c(ccc1C(=O)N1CCOc2ccc(cc2C1)-c1ccc(N)nc1)S(C)(=O)=O
CN1CCN(Cc2ccc(cc2)-c2cnc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)CC1
O=C(Cc1cccc(OCCCN2CCNCC2)c1)Nc1nc(cs1)-c1ccncc1
O=C(Cc1cccc(OCCCC2CCNCC2)c1)Nc1nc(cs1)-c1ccncc1
CS(=O)(=O)Nc1cccc(CC(=O)Nc2nc(cs2)-c2c[nH]c3ncccc23)c1
O=C(Cc1cccc(OCCCC2CCNCC2)c1)Nc1nc(cs1)-c1c[nH]c2ncccc12
CN1CCN(CCCOc2cccc(CC(=O)Nc3nc(cs3)-c3c[nH]c4ncccc34)c2)CC1
Oc1cccc(CNC(=O)Nc2nc(cs2)-c2ccncc2)c1
OC(=O)C1CN(Cc2ccc(OCc3ccc(Cl)c(Cl)c3)cc2)C1
[H][C@]12C[C@H]([C@@H](OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)CCOCCOCCOCCNC(=O)CCC1=[N+]2C(C=C1)=Cc1c(C)cc(C)n1[B-]2(F)F |r,c:63,65,t:60|
[H][C@]12C[C@@H](NCCOCCOCCOCCNC(=O)CCC3=[N+]4C(C=C3)=Cc3c(C)cc(C)n3[B-]4(F)F)[C@@H](OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r,c:24,26,t:21|
CN(C)c1ccc(cc1)C(=O)Nc1cccc(NC(=O)COc2ccc3c(c2)occc3=O)c1
Cn1ncc(Cl)c1-c1cc(oc1Cl)C(=O)N[C@@H]1CN[C@H](CCO)C[C@H]1c1ccc(F)c(F)c1 |r,wU:16.17,19.21,wD:24.27,(5.73,-5.85,;5.41,-7.35,;4,-7.98,;4.16,-9.51,;5.66,-9.83,;6.29,-11.24,;6.44,-8.5,;7.97,-8.34,;9,-9.49,;10.41,-8.86,;10.25,-7.33,;8.75,-7.01,;8.12,-5.6,;11.75,-9.64,;11.74,-11.18,;13.08,-8.87,;14.41,-9.65,;14.41,-11.18,;15.74,-11.96,;17.08,-11.19,;18.41,-11.96,;19.74,-11.2,;21.07,-11.97,;17.08,-9.64,;15.75,-8.88,;15.75,-7.35,;14.42,-6.58,;14.42,-5.03,;15.75,-4.26,;15.74,-2.72,;17.08,-5.03,;18.41,-4.25,;17.09,-6.58,)|
Cn1ncc(Cl)c1-c1cc(oc1Cl)C(=O)N[C@@H]1CNCC[C@H]1c1ccc(F)c(F)c1
Cn1ncc(Cl)c1-c1cc(oc1Cl)C(=O)N[C@H](CN)Cc1ccc(F)c(F)c1 |r,wD:16.18,(2.37,-.54,;3.52,.49,;3.36,2.02,;4.77,2.65,;5.8,1.51,;7.33,1.67,;5.03,.17,;5.65,-1.23,;7.16,-1.55,;7.32,-3.09,;5.91,-3.71,;4.88,-2.57,;3.35,-2.73,;8.65,-3.86,;9.99,-3.09,;8.65,-5.4,;9.99,-6.17,;11.32,-5.4,;12.65,-6.17,;9.99,-7.71,;11.32,-8.48,;12.65,-7.71,;13.99,-8.48,;13.99,-10.02,;15.32,-10.79,;12.65,-10.79,;12.65,-12.33,;11.32,-10.02,)|
CNC(=O)C[C@@H]1C[C@H]([C@@H](CN1)NC(=O)c1cc(c(Cl)o1)-c1c(Cl)cnn1C)c1ccc(F)c(F)c1 |r,wU:8.11,5.4,wD:7.29,(76.34,-11.8,;75,-12.56,;73.67,-11.79,;73.68,-10.25,;72.34,-12.55,;71.01,-11.78,;71.01,-10.23,;69.68,-9.47,;68.34,-10.24,;68.34,-11.77,;69.67,-12.55,;67.01,-9.46,;65.68,-10.23,;65.67,-11.77,;64.34,-9.46,;62.93,-10.08,;61.9,-8.93,;62.68,-7.6,;62.05,-6.19,;64.18,-7.92,;60.37,-9.09,;59.59,-10.42,;60.22,-11.83,;58.09,-10.1,;57.93,-8.57,;59.34,-7.94,;59.66,-6.44,;69.68,-7.94,;68.35,-7.17,;68.35,-5.62,;69.68,-4.85,;69.67,-3.31,;71.01,-5.62,;72.34,-4.84,;71.02,-7.17,)|
COc1cc(ccc1OCc2ccc(cc2)C3CC3)C4CN(C4)C(=O)c5cc(ccn5)COC[C@H](CO)O
Cc1sc(cc1-c1cnn2cc(Cl)cnc12)C(=O)N[C@@H]1[C@H](N)CCCC1(F)F |r|
Cn1cc(cn1)-c1cnc2c(cnn2c1)-c1csc(c1)C(=O)N[C@@H]1CCCC[C@@H]1N |r|
FC(F)(F)CNC(=O)c1cc(cs1)-c1cnn2cc(cnc12)-c1ccc(OCCN2CCCCC2)cc1
Cn1cc(cn1)-c1cnc2c(cnn2c1)-c1csc(c1)C(=O)NCC(F)(F)F
C[C@@H]1C[C@H]1C(=O)N1CCN(C[C@H]1C)c1cnc(C#N)c(n1)-c1cnn(C)c1 |r|
OCCNc1nc(NCCc2ccccc2)c2cnn(\C=C\c3ccccc3)c2n1
Cn1nccc1-c1ccc(C(=O)N[C@@H]2CNCC[C@H]2c2ccc(F)c(F)c2)c(F)c1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)N[C@@H]2CCNC2)c2cn[nH]c2n1 |r|
CN1CCC(C1)NC(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
CC(C)N1CC[C@@H](C1)NC(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1 |r|
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)NC2CCN(C2)C2CC2)c2cn[nH]c2n1
OCCN1CCC(C1)NC(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)NC2CCN(CC3CC3)C2)c2cn[nH]c2n1
NC(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
CNC(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
CCNC(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
CC(C)NC(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
CN(CCO)C(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
NCCNC(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)N2CCNCC2)c2cn[nH]c2n1
CN1CC(C1)NC(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
CN1CCC(CNC(=O)c2cc(nc3[nH]ncc23)-c2ccc(NS(=O)(=O)c3cccc(Cl)c3Cl)cc2)C1
CCN1CCC(CNC(=O)c2cc(nc3[nH]ncc23)-c2ccc(NS(=O)(=O)c3cccc(Cl)c3Cl)cc2)C1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)NCc2ncc[nH]2)c2cn[nH]c2n1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)NCc2nn[nH]n2)c2cn[nH]c2n1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)NCc2nncs2)c2cn[nH]c2n1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)NCc2cocn2)c2cn[nH]c2n1
Nc1nc(CNC(=O)c2cc(nc3[nH]ncc23)-c2ccc(NS(=O)(=O)c3cccc(Cl)c3Cl)cc2)cs1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)NCc2ncn[nH]2)c2cn[nH]c2n1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)NCCc2cc[nH]n2)c2cn[nH]c2n1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)NCCn2cnnc2)c2cn[nH]c2n1
CCOc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN(C)C(=O)CCOc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OCC3(CN)COC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCOCC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCC(=O)CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(Oc3ccc(O)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(Oc3ccc(N)nc3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CC(C)N1CC(COc2nc(nc3[nH]nc(C)c23)-c2ccc(NS(=O)(=O)c3cc(Cl)ccc3F)cc2)C1
Cc1n[nH]c2nc(nc(OC3CCNCC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CC(C)(C)NC(C)(C)C3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN1C(C)(C)CC(CC1(C)C)Oc1nc(nc2[nH]nc(C)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCNCC3F)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
Cc1n[nH]c2nc(nc(OC3CCN(CC3)C3CC3)c12)-c1ccc(NS(=O)(=O)c2cc(Cl)ccc2F)cc1
CN(C)CCCNC(=O)c1cc(nc2[nH]ncc12)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1
Clc1cccc(c1Cl)S(=O)(=O)Nc1ccc(cc1)-c1cc(C(=O)NCc2cc[nH]n2)c2cn[nH]c2n1
CN1Cc2nn(C)c(C#N)c2-c2cnc3[nH]cc(-c4cn(CCCC1=O)nc4C(F)(F)F)c3c2
CN1Cc2nn(C)c(C#N)c2-c2cnc3[nH]c(F)c(-c4cn(CCCC1=O)nc4C(F)(F)F)c3c2
c1ccc2c(c1)/C(=C/3\C(=N\O)\c4ccccc4N3)/C(=O)N2
C[C@@H](C(F)(F)F)N(Cc1ccc(cc1)F)C(=O)CN2C(=O)[C@]3(CCc4c3ccc(c4)NC(=O)NC)OC2=O
Cc1cc2c(c[nH]c2nc1)Cc3ccc(nc3F)NCc4cc(cnc4OC)F
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)NC)OC
CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O |r|
COc1cc2c(cc1NC(=O)/C=C/CN3CCCCC3)c(ncn2)Nc4ccc(c(c4)Cl)F
CCOc1cc(ccc1Nc2ncc3c(n2)N(c4ccccc4C(=O)N3C)C)N5CCC(CC5)O
Cc1cn(CCN2CCN(CC2)c2ccccc2-c2cc(cc(c2)C(=O)NCCCN2CCCC2)C#N)c2ccccc12
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(nn3-c3ccc4ncccc4c3)C(C)(C)C)c(F)c2)ccn1
c1cc(c(cc1I)F)Nc2c(ccc(c2F)F)C(=O)N3CC(C3)([C@@H]4CCCCN4)O
O=C(NCC#N)c1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1
CC[C@@H]1CN(C[C@@H]1c1cnc2cnc3[nH]ccc3n12)C(=O)NCC(F)(F)F |r|