Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 58 with Last Name = 'kugimiya' and Initial = 'a'
TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111610(US8623903, I-23)
Affinity DataKi:  1.40nM IC50:  1.60nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111612(US8623903, I-31)
Affinity DataKi:  4.30nM IC50:  2.90nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111611(US8623903, I-30)
Affinity DataKi:  5.40nM IC50:  1.20nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111606(US8623903, I-14)
Affinity DataKi:  5.60nM IC50:  2.20nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111597(US8623903, I-1)
Affinity DataKi:  7.70nM IC50:  4.70nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111598(US8623903, I-5)
Affinity DataKi:  22nM IC50:  4.10nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111607(US8623903, I-16)
Affinity DataIC50:  1.30nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111600(US8623903, I-7)
Affinity DataIC50:  1.80nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111602(US8623903, I-9)
Affinity DataIC50:  2nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111609(US8623903, I-21)
Affinity DataIC50:  3nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111608(US8623903, I-20)
Affinity DataIC50:  3.80nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111599(US8623903, I-6)
Affinity DataIC50:  4.80nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111601(US8623903, I-8)
Affinity DataIC50:  4.90nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111604(US8623903, I-11)
Affinity DataIC50:  4.90nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111603(US8623903, I-10)
Affinity DataIC50:  6.90nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111605(US8623903, I-12)
Affinity DataIC50:  6.90nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetProstaglandin D2 receptor 2(Human)
Shionogi

US Patent
LigandPNGBDBM111613(US8623903, I-32)
Affinity DataIC50:  7nMAssay Description:A prepared WP was homogenated and a membrane fraction was collected with high-speed centrifugation. A compound of the present invention was added to ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147469(US8957219, II-2-67)
Affinity DataIC50:  29nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147471(US8957219, II-2-144)
Affinity DataIC50:  29nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147472(US8957219, II-2-211)
Affinity DataIC50:  32nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147473(US8957219, II-2-291)
Affinity DataIC50:  56nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147470(US8957219, II-2-131)
Affinity DataIC50:  92nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM47169(US8957219, II-2-1)
Affinity DataIC50:  110nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM47168(US8957219, II-1-1)
Affinity DataIC50:  230nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147468(US8957219, II-1-246)
Affinity DataIC50:  280nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147467(US8957219, II-1-202)
Affinity DataIC50:  290nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM20182((1S,2R,5S,10S,11S,14R,15R)-14-[(2R)-6-hydroxy-6-me...)
Affinity DataIC50:  300nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147464(US8957219, II-1-11)
Affinity DataIC50:  560nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351538(CHEMBL1824673)
Affinity DataIC50:  700nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351539(CHEMBL1824674)
Affinity DataIC50:  900nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351538(CHEMBL1824673)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells by densitometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147465(US8957219, II-1-17)
Affinity DataIC50:  1.30E+3nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351541(CHEMBL1824676)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Human)
Shionogi

US Patent
LigandPNGBDBM147466(US8957219, II-1-190)
Affinity DataIC50:  2.10E+3nMT: 37°CAssay Description:After the present compound dissolved in DMSO was added to become 0.5% DMSO to the reaction buffer consisting of 20 mM tris hydrochloric acid (pH7.4),...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351540(CHEMBL1824675)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351534(CHEMBL1824669)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351535(CHEMBL1824670)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351529(CHEMBL1824664)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351536(CHEMBL1824671)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM78179(2-(2-propyl-4-pyridyl)-4-(p-tolyl)thiazole;hydrobr...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351521(CHEMBL1824658)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351537(CHEMBL1824672)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351542(CHEMBL1824661)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351533(CHEMBL1824668)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351531(CHEMBL1824666)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351530(CHEMBL1824665)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351526(CHEMBL1616869)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM78179(2-(2-propyl-4-pyridyl)-4-(p-tolyl)thiazole;hydrobr...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells by densitometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351528(CHEMBL1824663)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM93773(4-(4-chlorophenyl)-2-(2-propyl-4-pyridinyl)thiazol...)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 58 total ) | Next | Last >>
Jump to: