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Found 511 with Last Name = 'buckner' and Initial = 'fs'
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13321(1-Methyl-1H-imidazole-4-sulfonic Acid (2-Bromoally...)
Affinity DataIC50:  0.400nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13307(1-Methyl-1H-imidazole-4-sulfonic Acid Benzyl-{2-[(...)
Affinity DataIC50:  0.5nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50067584((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bip...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of mammalian protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13320(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  0.600nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13311(1-Methyl-1H-imidazole-4-sulfonic Acid {2-[(4-Cyano...)
Affinity DataIC50:  0.600nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13323(1-Methyl-1H-imidazole-4-sulfonic Acid Benzyl-[6-cy...)
Affinity DataIC50:  0.600nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13320(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  0.700nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13328(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  0.800nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13321(1-Methyl-1H-imidazole-4-sulfonic Acid (2-Bromoally...)
Affinity DataIC50:  0.800nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM16182((2S)-2-[(4-{[(1H-imidazol-4-ylmethyl)amino]methyl}...)
Affinity DataIC50:  0.860nMAssay Description:Inhibition of mammalian protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13319(BMS-386914 | CHEMBL183536 | [[6-Cyano-1-(3-methyl-...)
Affinity DataIC50:  0.900nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13325(4-{[[6-Cyano-1-(3-methyl-3H-imidazol-4-ylmethyl)-1...)
Affinity DataIC50:  1.10nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13323(1-Methyl-1H-imidazole-4-sulfonic Acid Benzyl-[6-cy...)
Affinity DataIC50:  1.20nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13319(BMS-386914 | CHEMBL183536 | [[6-Cyano-1-(3-methyl-...)
Affinity DataIC50:  1.20nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13322(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  1.20nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13331(N-tert-butyl-2-({6-isocyano-1-[(1-methyl-1H-imidaz...)
Affinity DataIC50:  1.40nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13322(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  1.5nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13324(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  1.5nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50067584((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bip...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of Trypanosoma brucei protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50476682(CHEMBL428712 | PB-43)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM16182((2S)-2-[(4-{[(1H-imidazol-4-ylmethyl)amino]methyl}...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of Trypanosoma brucei protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13331(N-tert-butyl-2-({6-isocyano-1-[(1-methyl-1H-imidaz...)
Affinity DataIC50:  1.80nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13309(N-(2-{(4-bromophenyl)[(1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50:  1.90nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13308(N-benzyl-N-(2-{(4-bromophenyl)[(1-methyl-1H-imidaz...)
Affinity DataIC50:  2nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13310(N-(2-{(4-cyanophenyl)[(1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50:  2.10nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50476678(CHEMBL395222)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13327(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  2.80nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50234534(CHEMBL4088945)
Affinity DataIC50:  3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM13328(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  3nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13328(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  3nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13325(4-{[[6-Cyano-1-(3-methyl-3H-imidazol-4-ylmethyl)-1...)
Affinity DataIC50:  3.20nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50476685(CHEMBL232104)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM13324(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13324(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  3.40nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM13327(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13327(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50:  3.80nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50133285((E)-3-Carboxy-acrylateallyl-{6-[4-(4-chloro-benzoy...)
Affinity DataIC50:  4.30nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in T. bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM13315(1-Methyl-1H-imidazole-4-sulfonic Acid {2-[(4-Cyano...)
Affinity DataIC50:  4.5nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50133285((E)-3-Carboxy-acrylateallyl-{6-[4-(4-chloro-benzoy...)
Affinity DataIC50:  4.60nMAssay Description:Tested for Oxidosqualene-lanosterol cyclase inhibition in P. cariniiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50476680(CHEMBL234757)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent RNA helicase RhlE(Plasmodium falciparum (malaria parasite P. falcipa...)
University of Washington At Seattle

LigandPNGBDBM16180((2S)-2-{[4-({[(2S)-1-cyclohexyl-3-(ethylsulfanyl)p...)
Affinity DataIC50:  5nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM13335(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13335(N-tert-Butyl-2-[[6-cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  5nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50476679(CHEMBL232523)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50138762((S)-2-[(5-{[Bis-(1H-imidazol-4-ylmethyl)-amino]-me...)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of Trypanosoma brucei protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13332(N-tert-Butyl-2-[[6-isocyano-1-(3-methyl-3H-imidazo...)
Affinity DataIC50:  6nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50476681(CHEMBL234151 | PB-91)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50138763((S)-2-({2'-Methyl-5-[2-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of Trypanosoma brucei protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University of Washington

Curated by ChEMBL
LigandPNGBDBM50476676(CHEMBL231662)
Affinity DataIC50:  7nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington At Seattle

LigandPNGBDBM13315(1-Methyl-1H-imidazole-4-sulfonic Acid {2-[(4-Cyano...)
Affinity DataIC50:  7.5nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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