Compile Data Set for Download or QSAR
maximum 50k data
Found 69 with Last Name = 'carrero-lérida' and Initial = 'j'
TargetPurine nucleoside phosphorylase(Plasmodium falciparum)
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50195587(1,4-DIDEOXY-4-AZA-1-(S)-(9-DEAZAHYPOXANTHIN-9-YL)-...)
Affinity DataKi:  0.860nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Plasmodium falciparum)
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330391(5-(3-(benzyloxy)benzyl)-1-((2-hydroxyethoxy)methyl...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine phosphorylase 1(Homo sapiens (Human))
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330391(5-(3-(benzyloxy)benzyl)-1-((2-hydroxyethoxy)methyl...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of human uridine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Plasmodium falciparum)
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330390(5'-methylthio-immucillin-H | CHEMBL1275659)
Affinity DataKi:  2.70nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330390(5'-methylthio-immucillin-H | CHEMBL1275659)
Affinity DataKi:  303nMAssay Description:Inhibition of human PNPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine phosphorylase 1(Homo sapiens (Human))
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50078082(5-(3-Benzyloxy-benzyl)-pyrimidine-2,4,6-trione | C...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of human uridine phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Plasmodium falciparum)
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330388(3-((2-Pyrrolidine-1-yl)-ethyl)uracil | CHEMBL12757...)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400466(CHEMBL2178479)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400445(CHEMBL2179048)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400454(CHEMBL2179039)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400452(CHEMBL2179041)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50359622(CHEMBL1928432)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Plasmodium falciparum)
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330394(1-((2-Pyrrolidine-1-yl)-ethyl)uracil | CHEMBL12756...)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400446(CHEMBL2179047)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400455(CHEMBL2179038)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50223806(CHEMBL392137 | N-(5'-deoxy-alpha-D-thymidin-5'-yl)...)
Affinity DataKi:  3.10E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400451(CHEMBL2179042)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400453(CHEMBL2179040)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400447(CHEMBL2179046)
Affinity DataKi:  4.70E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400448(CHEMBL2179045)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400456(CHEMBL2179037)
Affinity DataKi:  5.20E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Plasmodium falciparum)
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330395(1-((3-Pyrrolidine-1-yl)-propyl)uracil | CHEMBL1275...)
Affinity DataKi:  5.90E+4nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400457(CHEMBL2179036)
Affinity DataKi:  6.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400459(CHEMBL2179034)
Affinity DataKi:  6.40E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400471(CHEMBL2178506)
Affinity DataKi:  6.50E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400449(CHEMBL2179044)
Affinity DataKi:  6.90E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Plasmodium falciparum)
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330389(3-((2-(l-Prolinol)-1-yl)-ethyl)uracil | CHEMBL1275...)
Affinity DataKi:  7.50E+4nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50223798(CHEMBL391451 | N-(5'-deoxy-alpha-D-thymidin-5'-yl)...)
Affinity DataKi:  8.80E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50223805(CHEMBL442081 | N'-(4-chlorophenyl)-N-(5'-deoxy-alp...)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Plasmodium falciparum)
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330397(1-((4-Pyrrolidine-1-yl)-butyl)uracil | CHEMBL12757...)
Affinity DataKi:  1.05E+5nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400474(CHEMBL2178504)
Affinity DataKi:  1.06E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400450(CHEMBL2179043)
Affinity DataKi:  1.07E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Plasmodium falciparum)
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330398(1-((4-(l-Prolinol)-1-yl)-butyl)uracil | CHEMBL1275...)
Affinity DataKi:  1.13E+5nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400473(CHEMBL2177119)
Affinity DataKi:  1.14E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400468(CHEMBL2178477)
Affinity DataKi:  1.32E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Plasmodium falciparum)
Instituto De ParasitologíA Y Biomedicina LóPez-Neyra

Curated by ChEMBL
LigandPNGBDBM50330396(1-((3-(l-Prolinol)-1-yl)-propyl)uracil | CHEMBL127...)
Affinity DataKi:  1.36E+5nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400470(CHEMBL2178507)
Affinity DataKi:  1.38E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400469(CHEMBL2178508)
Affinity DataKi:  1.59E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400476(CHEMBL2178502)
Affinity DataKi:  1.66E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400467(CHEMBL2178478)
Affinity DataKi:  1.67E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400478(CHEMBL2178500)
Affinity DataKi:  1.98E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400460(CHEMBL2179033)
Affinity DataKi:  2.01E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400475(CHEMBL2178503)
Affinity DataKi:  2.05E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400458(CHEMBL2179035)
Affinity DataKi:  2.22E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400462(CHEMBL2179031)
Affinity DataKi:  3.02E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400482(CHEMBL2178496)
Affinity DataKi:  5.41E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400481(CHEMBL2178497)
Affinity DataKi:  5.41E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400461(CHEMBL2179032)
Affinity DataKi:  7.42E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400465(CHEMBL2178509)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetdTMP kinase(Plasmodium falciparum (isolate 3D7))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50400464(CHEMBL2178510)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of recombinant Plasmodium falciparum TMPK using TMP as substrate by pyruvate kinase and lactate dehydrogenase enzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 69 total ) | Next | Last >>
Jump to: