Compile Data Set for Download or QSAR
maximum 50k data
Found 30 with Last Name = 'michiels' and Initial = 'j'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368791(CHEMBL4171931)
Affinity DataKi:  0.617nMAssay Description:Displacement of [3H]ZM241385 human A2AR (1 to 316 residues) expressed in Pichia pastoris SMD1168 cell membranes incubated for 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368789(CHEMBL4164058)
Affinity DataKi:  0.891nMAssay Description:Displacement of [3H]ZM241385 human A2AR (1 to 316 residues) expressed in Pichia pastoris SMD1168 cell membranes incubated for 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368790(CHEMBL4159904)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]ZM241385 human A2AR (1 to 316 residues) expressed in Pichia pastoris SMD1168 cell membranes incubated for 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368792(CHEMBL4167502)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]ZM241385 human A2AR (1 to 316 residues) expressed in Pichia pastoris SMD1168 cell membranes incubated for 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368791(CHEMBL4171931)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]ZM241385 human A2AR (1 to 316 residues) expressed in Pichia pastoris SMD1168 cell membranes incubated for 0.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368792(CHEMBL4167502)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]ZM241385 human A2AR (1 to 316 residues) expressed in Pichia pastoris SMD1168 cell membranes incubated for 0.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368790(CHEMBL4159904)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]ZM241385 human A2AR (1 to 316 residues) expressed in Pichia pastoris SMD1168 cell membranes incubated for 0.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368789(CHEMBL4164058)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]ZM241385 human A2AR (1 to 316 residues) expressed in Pichia pastoris SMD1168 cell membranes incubated for 0.5 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436321(CHEMBL3037796)
Affinity DataIC50:  0.260nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436320(CHEMBL3037792)
Affinity DataIC50:  0.280nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436319(CHEMBL3037791)
Affinity DataIC50:  0.300nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436318(CHEMBL3037787)
Affinity DataIC50:  0.320nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436317(CHEMBL3037785)
Affinity DataIC50:  0.350nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436316(CHEMBL3037786)
Affinity DataIC50:  0.5nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436315(CHEMBL2398774)
Affinity DataIC50:  0.520nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436314(CHEMBL3037790)
Affinity DataIC50:  0.860nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436313(CHEMBL3037788)
Affinity DataIC50:  1.10nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436312(CHEMBL3037797)
Affinity DataIC50:  1.40nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436326(CHEMBL3037789)
Affinity DataIC50:  5.20nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436325(CHEMBL3037793)
Affinity DataIC50:  5.30nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436324(CHEMBL3037798)
Affinity DataIC50:  8.10nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436323(CHEMBL3037794)
Affinity DataIC50:  284nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea

Curated by ChEMBL
LigandPNGBDBM50436322(CHEMBL3037795)
Affinity DataIC50:  2.03E+3nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50467334(AIDS-105293 | Dapivirine | R-147681 | TMC-120)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50484289(CHEMBL1829450)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50484288(CHEMBL1829447)
Affinity DataIC50:  5.47E+5nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50484290(CHEMBL1830529)
Affinity DataIC50:  7.60E+5nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50484291(CHEMBL1829465)
Affinity DataIC50:  9.28E+5nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50368792(CHEMBL4167502)
Affinity DataEC50:  794nMAssay Description:Photoaffinity labelling of purified human A2AR (1 to 316 residues) by SDS-PAGE analaysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed