TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University of Li£Ge
Curated by ChEMBL
University of Li£Ge
Curated by ChEMBL
Affinity DataKi: 0.00400nMAssay Description:Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5-HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5-HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding affinity against rat 5-hydroxytryptamine 2 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Binding affinity to 5HT1A receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.870nMAssay Description:Binding affinity against dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:In vitro binding affinity against Dopamine D2 receptor in rat striatal tissue.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-8-OH-OPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.21nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5-HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.61nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5-HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.69nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.77nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:In vitro binding affinity against rat 5-hydroxytryptamine 2 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.85nMAssay Description:Binding affinity to 5HT1A receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.89nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5-HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding affinity against Dopamine D2 receptor in rat striatal tissue.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity to 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:In vitro binding affinity at human cloned Dopamine receptor D4 expressed in Sf9 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.32nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.42nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.48nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5-HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]-8-OH-OPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.75nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.87nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity to 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:In vitro binding affinity against rat 5-hydroxytryptamine 2 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]-8-OH-OPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]-8-OH-OPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:In vitro binding affinity against rat 5-hydroxytryptamine 2 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:In vitro binding affinity against rat 5-hydroxytryptamine 2 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:In vitro binding affinity against rat 5-hydroxytryptamine 2 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:In vitro binding affinity against Dopamine D2 receptor in rat striatal tissue.More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity against dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.59nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.64nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.84nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.19nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:In vitro binding affinity against Muscarinic acetylcholine receptors in rat brain.More data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Displacement of [3H]-8-OH-OPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.15nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:In vitro binding affinity against rat 5-hydroxytryptamine 2 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:In vitro binding affinity at serotonin 5-hydroxytryptamine 2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]-8-OH-OPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Displacement of [3H]-8-OH-OPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]-8-OH-OPAT from human recombinant 5HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.27nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5-HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.36nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5-HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:In vitro binding affinity at human cloned Dopamine receptor D2L expressed in Sf9 cell membranesMore data for this Ligand-Target Pair