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Found 21 with Last Name = 'lazarus' and Initial = 'ra'
TargetPhenylalanine-4-hydroxylase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028430(2-Amino-6-phenyl-7,8-dihydro-3H,6H-pyrimido[5,4-b]...)
Affinity DataKi:  200nMAssay Description:Tested for competitive binding inhibition against phenylalanine hydroxylase in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylalanine-4-hydroxylase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028428(2,6-Diamino-5-phenylsulfanyl-3H-pyrimidin-4-one | ...)
Affinity DataKi:  4.70E+3nMAssay Description:Tested for competitive binding inhibition against phenylalanine hydroxylase in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylalanine-4-hydroxylase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028426(2-Amino-5-oxo-6-phenyl-5,6,7,8-tetrahydro-3H-5lamb...)
Affinity DataKi:  7.00E+3nMAssay Description:Tested for competitive binding inhibition against phenylalanine hydroxylase in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylalanine-4-hydroxylase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028425(2-Amino-6-methyl-7,8-dihydro-3H,6H-pyrimido[5,4-b]...)
Affinity DataKi:  3.60E+4nMAssay Description:Tested for competitive binding inhibition against phenylalanine hydroxylase in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylalanine-4-hydroxylase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028424(2-Amino-7,8-dihydro-3H,6H-pyrimido[5,4-b][1,4]thia...)
Affinity DataKi:  8.50E+4nMAssay Description:Tested for competitive binding inhibition against phenylalanine hydroxylase in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylalanine-4-hydroxylase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028427(2-Amino-6-methyl-5-oxo-5,6,7,8-tetrahydro-3H-5lamb...)
Affinity DataKi:  1.25E+5nMAssay Description:Tested for competitive binding inhibition against phenylalanine hydroxylase in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylalanine-4-hydroxylase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028431(2-Amino-5-oxo-5,6,7,8-tetrahydro-3H-5lambda*4*-pyr...)
Affinity DataKi:  4.00E+5nMAssay Description:Tested for competitive binding inhibition against phenylalanine hydroxylase in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylalanine-4-hydroxylase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028429(2-Amino-3,5,6,7-tetrahydro-pyrimido[4,5-b][1,4]thi...)
Affinity DataKi:  5.00E+5nMAssay Description:Tested for competitive binding inhibition against phenylalanine hydroxylase in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119052(Biotinylated E-76 peptide analogue | CHEMBL269354)
Affinity DataIC50:  1nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119057(ALCDNPRIDRWYCQFVEG peptide analogue | Biotinylated...)
Affinity DataIC50:  1nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119050(ALCDNPRIDRWYCQFVEG peptide analogue | Biotinylated...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119049(Biotinylated E-76 peptide analogue | CHEMBL439285)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119048(Biotinylated E-76 peptide analogue | CHEMBL437872)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119055(Biotinylated E-76 peptide analogue | CHEMBL414777)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119056(Biotinylated E-76 peptide analogue | CHEMBL439444)
Affinity DataIC50:  4nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119047(Biotinylated E-76 peptide analogue | CHEMBL441926)
Affinity DataIC50:  10nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119053(Biotinylated E-76 peptide analogue | CHEMBL415402)
Affinity DataIC50:  12nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119054(Biotinylated E-76 peptide analogue | CHEMBL429011)
Affinity DataIC50:  13nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119059(Biotinylated E-76 peptide analogue | CHEMBL410836)
Affinity DataIC50:  13nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119051(Biotinylated E-76 peptide analogue | CHEMBL415837)
Affinity DataIC50:  15nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119058(Biotinylated E-76 peptide analogue | CHEMBL410279)
Affinity DataIC50:  20nMAssay Description:Inhibition of amino terminally biotinylated E-76 peptide binding to immobilized fVIIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed