Affinity DataKi: 0.0120nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Inhibitory activity of the compound against Coagulation factor Xa (serine protease) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.0440nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:In vitro inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.105nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.117nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibitory activity of the compound against factor Xa,activity expressed as Ki nMMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Binding affinity of the compound towards factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:In vitro inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:In vitro inhibitory activity of the compound against Coagulation factor X was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:In vitro binding affinity towards factor XaMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Inhibition Protein kinase C (PKC)More data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:In vitro inhibitory activity against coagulation factor XMore data for this Ligand-Target Pair