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Found 36 with Last Name = 'takayama' and Initial = 's'
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072685((3,4,5-Trihydroxy-2-hydroxymethyl-6-methyl-piperid...)
Affinity DataKi:  1.5nMAssay Description:Compound was tested for inhibitory activity against alpha-1,2-Fucosidase obtained from Arthrobacter oxidans F1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072685((3,4,5-Trihydroxy-2-hydroxymethyl-6-methyl-piperid...)
Affinity DataKi:  8nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072685((3,4,5-Trihydroxy-2-hydroxymethyl-6-methyl-piperid...)
Affinity DataKi:  11nMAssay Description:Compound was tested for inhibitory activity against alpha-1,2-Fucosidase obtained from Arthrobacter oxidans F1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072687((S)-2-Amino-3-hydroxy-N-(3,4,5-trihydroxy-2-hydrox...)
Affinity DataKi:  19nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine epididymisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072687((S)-2-Amino-3-hydroxy-N-(3,4,5-trihydroxy-2-hydrox...)
Affinity DataKi:  30nMAssay Description:Compound was tested for inhibitory activity against alpha-1,2-Fucosidase obtained from Arthrobacter oxidans F1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072687((S)-2-Amino-3-hydroxy-N-(3,4,5-trihydroxy-2-hydrox...)
Affinity DataKi:  47nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1,4-galactosyltransferase 1(Bos taurus (Cattle))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072694(CHEMBL320104 | N-[4,5-Dihydroxy-6-hydroxymethyl-2-...)
Affinity DataKi:  3.50E+3nMAssay Description:Compound was tested for the inhibition recombinant bovine beta -1,4 -galactosyl transferase (beta-1,4-GalT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1,4-galactosyltransferase 1(Bos taurus (Cattle))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072688(CHEMBL111972 | N-[2-(6-Bromo-naphthalen-2-yloxy)-4...)
Affinity DataKi:  7.60E+3nMAssay Description:Compound was tested for the inhibition recombinant bovine beta -1,4 -galactosyl transferase (beta-1,4-GalT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-acetyllactosaminide alpha-1,3-galactosyltransferase(Sus scrofa)
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072692(CHEMBL2303732 | N-[2-(6-Bromo-naphthalen-2-yloxy)-...)
Affinity DataKi:  9.20E+3nMAssay Description:Compound was tested for the inhibition porcine alpha -1,3 -galactosyl transferase (alpha-1,3-GalT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1,4-galactosyltransferase 1(Bos taurus (Cattle))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072689(CHEMBL112241 | N-[4,5-Dihydroxy-6-hydroxymethyl-2-...)
Affinity DataKi:  9.50E+3nMAssay Description:Compound was tested for the inhibition recombinant bovine beta -1,4 -galactosyl transferase (beta-1,4-GalT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1,4-galactosyltransferase 1(Bos taurus (Cattle))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072693(CHEMBL114323 | N-[4,5-Dihydroxy-6-hydroxymethyl-2-...)
Affinity DataKi:  2.20E+4nMAssay Description:Compound was tested for the inhibition recombinant bovine beta -1,4 -galactosyl transferase (beta-1,4-GalT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-acetyllactosaminide alpha-1,3-galactosyltransferase(Sus scrofa)
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072690(CHEMBL326048 | N-[5-(4-Amino-3,5-dihydroxy-6-hydro...)
Affinity DataKi:  1.04E+5nMAssay Description:Compound was tested for the inhibition porcine alpha -1,3 -galactosyl transferase (alpha-1,3-GalT) at 0.2 mM concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1,4-galactosyltransferase 1(Bos taurus (Cattle))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072695(CHEMBL115776 | N-(5-Amino-2-benzyloxy-4-hydroxy-6-...)
Affinity DataKi:  8.50E+5nMAssay Description:Compound was tested for the inhibition recombinant bovine beta -1,4 -galactosyl transferase (beta-1,4-GalT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1,4-galactosyltransferase 1(Bos taurus (Cattle))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072691(CHEMBL2303731 | N-[2-(3,5-Dihydroxy-2-hydroxymethy...)
Affinity DataKi:  1.00E+6nMAssay Description:Compound was tested for the inhibition recombinant bovine beta -1,4 -galactosyl transferase (beta-1,4-GalT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072685((3,4,5-Trihydroxy-2-hydroxymethyl-6-methyl-piperid...)
Affinity DataIC50:  4nMAssay Description:Compound was tested for inhibitory activity against alpha-1,2-Fucosidase obtained from Arthrobacter oxidans F1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072685((3,4,5-Trihydroxy-2-hydroxymethyl-6-methyl-piperid...)
Affinity DataIC50:  11nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072685((3,4,5-Trihydroxy-2-hydroxymethyl-6-methyl-piperid...)
Affinity DataIC50:  11nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine epididymisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072687((S)-2-Amino-3-hydroxy-N-(3,4,5-trihydroxy-2-hydrox...)
Affinity DataIC50:  20nMAssay Description:Compound was tested for inhibitory activity against alpha-1,2-Fucosidase obtained from Arthrobacter oxidans F1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072682(CHEMBL115930 | {[(3,4,5-Trihydroxy-2-hydroxymethyl...)
Affinity DataIC50:  40nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072687((S)-2-Amino-3-hydroxy-N-(3,4,5-trihydroxy-2-hydrox...)
Affinity DataIC50:  40nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072684(2-Amino-N-(3,4,5-trihydroxy-2-hydroxymethyl-6-meth...)
Affinity DataIC50:  50nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072687((S)-2-Amino-3-hydroxy-N-(3,4,5-trihydroxy-2-hydrox...)
Affinity DataIC50:  56nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine epididymisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072683(3,4,5-Trihydroxy-2-hydroxymethyl-6-methyl-piperidi...)
Affinity DataIC50:  75nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine epididymisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072686(2-Aminomethyl-2-hydroxymethyl-6-methyl-piperidine-...)
Affinity DataIC50:  80nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine epididymisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072683(3,4,5-Trihydroxy-2-hydroxymethyl-6-methyl-piperidi...)
Affinity DataIC50:  110nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine epididymisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072684(2-Amino-N-(3,4,5-trihydroxy-2-hydroxymethyl-6-meth...)
Affinity DataIC50:  116nMAssay Description:Compound was tested for inhibitory activity against alpha-1,2-Fucosidase obtained from Arthrobacter oxidans F1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072683(3,4,5-Trihydroxy-2-hydroxymethyl-6-methyl-piperidi...)
Affinity DataIC50:  122nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine epididymisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072686(2-Aminomethyl-2-hydroxymethyl-6-methyl-piperidine-...)
Affinity DataIC50:  160nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine epididymisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072684(2-Amino-N-(3,4,5-trihydroxy-2-hydroxymethyl-6-meth...)
Affinity DataIC50:  170nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072682(CHEMBL115930 | {[(3,4,5-Trihydroxy-2-hydroxymethyl...)
Affinity DataIC50:  190nMAssay Description:Compound was tested for inhibitory activity against alpha-1,2-Fucosidase obtained from Arthrobacter oxidans F1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072682(CHEMBL115930 | {[(3,4,5-Trihydroxy-2-hydroxymethyl...)
Affinity DataIC50:  200nMAssay Description:Compound was tested for inhibitory activity against alpha-Fucosidase obtained from Bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50072686(2-Aminomethyl-2-hydroxymethyl-6-methyl-piperidine-...)
Affinity DataIC50:  206nMAssay Description:Compound was tested for inhibitory activity against alpha-1,2-Fucosidase obtained from Arthrobacter oxidansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50071379(CHEMBL3410227)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of human recombinant myostatin pre-incubated with compound for 1 hr before addition to human HepG2 cells assessed as reduction in myostati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50071379(CHEMBL3410227)
Affinity DataKd:  36nMAssay Description:Binding affinity to recombinant myostatin (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50071380(CHEMBL3410232)
Affinity DataKd:  30nMAssay Description:Binding affinity to recombinant myostatin (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50071381(CHEMBL3410234)
Affinity DataKd:  117nMAssay Description:Binding affinity to recombinant myostatin (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed