Affinity DataKi: 12nMAssay Description:Antagonist potency against adenosine A2B receptor of guinea pig thoracic aortic smooth muscleMore data for this Ligand-Target Pair
Affinity DataKi: 4.52E+3nMAssay Description:Antagonist potency at cloned recombinant human adenosine A2B receptor transfected in CHO cells by cAMP assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of PRKKA1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of MER (unknown origin)More data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ROCK1 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of ITK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of ROCK1 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of ITK (unknown origin)More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of ERBB4 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of ERBB4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of EPHA3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of EPHA3 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of p38 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of p38 (unknown origin)More data for this Ligand-Target Pair
Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of PRKKA1 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of MER (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of HER4 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataIC50: <2.00E+4nMAssay Description:Inhibition of HER4 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataKd: <1nMAssay Description:Binding affinity to ASK1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Inhibition of ASK1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Takeda Research In California
Curated by ChEMBL
Takeda Research In California
Curated by ChEMBL
Affinity DataEC50: 24nMAssay Description:Inhibition of ASK1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
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