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Found 270 with Last Name = 'palomo' and Initial = 'v'
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602886(CHEMBL5182036)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602886(CHEMBL5182036)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of TTBK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM7262(14-nitro-8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12,...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant GSK3betaMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347535(CHEMBL1801637)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347531(CHEMBL1801633)
Affinity DataIC50:  47nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50229962(1-(4-methoxybenzyl)-3-(5-nitrothiazol-2-yl)urea | ...)
Affinity DataIC50:  104nMAssay Description:Inhibition of human recombinant GSK3betaMore data for this Ligand-Target Pair
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602885(CHEMBL5193906)
Affinity DataIC50:  120nMAssay Description:Inhibition of TTBK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTau-tubulin kinase 2(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602885(CHEMBL5193906)
Affinity DataIC50:  170nMAssay Description:Inhibition of TTBK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602904(CHEMBL5204869)
Affinity DataIC50:  240nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382610(CHEMBL2022413)
Affinity DataIC50:  300nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382604(CHEMBL2022420 | CHEMBL2024373)
Affinity DataIC50:  300nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382608(CHEMBL2022415)
Affinity DataIC50:  300nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602917(CHEMBL5200069)
Affinity DataIC50:  330nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602907(CHEMBL5193488)
Affinity DataIC50:  340nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602930(CHEMBL5181249)
Affinity DataIC50:  360nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602922(CHEMBL5184336)
Affinity DataIC50:  370nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602921(CHEMBL5180098)
Affinity DataIC50:  380nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602903(CHEMBL5198544)
Affinity DataIC50:  390nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602932(CHEMBL5178965)
Affinity DataIC50:  390nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602910(CHEMBL5209196)
Affinity DataIC50:  420nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602906(CHEMBL5187459)
Affinity DataIC50:  440nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602920(CHEMBL5187125)
Affinity DataIC50:  450nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602931(CHEMBL5197012)
Affinity DataIC50:  480nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602917(CHEMBL5200069)
Affinity DataIC50:  490nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM7876(2-bromo-1-(4-bromophenyl)ethan-1-one | Halomethyl ...)
Affinity DataIC50:  500nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347526(CHEMBL1801628)
Affinity DataIC50:  500nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382615(CHEMBL2024372)
Affinity DataIC50:  500nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602911(CHEMBL5171328)
Affinity DataIC50:  520nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602900(CHEMBL5185704 | US11814388, Compound 3)
Affinity DataIC50:  520nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347533(CHEMBL1801635)
Affinity DataIC50:  580nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382627(CHEMBL2024362)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382606(CHEMBL2022418 | CHEMBL2024361)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382619(CHEMBL2022416)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602929(CHEMBL5193034)
Affinity DataIC50:  610nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602925(CHEMBL5188513)
Affinity DataIC50:  650nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602926(CHEMBL5200160 | US11814388, Compound 9)
Affinity DataIC50:  750nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602934(CHEMBL5206548)
Affinity DataIC50:  750nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602909(CHEMBL5197789)
Affinity DataIC50:  750nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602905(CHEMBL5208565)
Affinity DataIC50:  770nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602899(CHEMBL5207783)
Affinity DataIC50:  790nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382607(CHEMBL2022417)
Affinity DataIC50:  800nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602916(CHEMBL5196033)
Affinity DataIC50:  840nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602903(CHEMBL5198544)
Affinity DataIC50:  850nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347534(CHEMBL1801636)
Affinity DataIC50:  890nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382625(CHEMBL558982)
Affinity DataIC50:  900nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382603(CHEMBL2022421)
Affinity DataIC50:  900nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Quimica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50382605(CHEMBL2022414 | CHEMBL2022419)
Affinity DataIC50:  900nMAssay Description:Inhibition of human recombinant GSK3beta after 30 mins by luminescence assay in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602907(CHEMBL5193488)
Affinity DataIC50:  970nMAssay Description:Inhibition of recombinant human TTBK2 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50602933(CHEMBL5178462)
Affinity DataIC50:  990nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTau-tubulin kinase 1(Homo sapiens (Human))
Csic

Curated by ChEMBL
LigandPNGBDBM50328192(CHEMBL1257781 | N-(4-(Trifluoromethoxy)phenyl)-7H-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails PubMed
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