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Found 193 with Last Name = 'zeng' and Initial = 'w'
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM50109647(2-{1-[2-(2,3-Dihydro-benzofuran-5-yl)-ethyl]-pyrro...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM50109647(2-{1-[2-(2,3-Dihydro-benzofuran-5-yl)-ethyl]-pyrro...)
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266051((4-(furan-2-yl)-2-(2-(thiophen-2-yl)ethylamino)thi...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
South China University of Technology

Curated by ChEMBL
LigandPNGBDBM50233190(CHEMBL4104953)
Affinity DataKi:  16nMAssay Description:Inhibition of human liver carboxylesterase 1 using o-nitrophenyl acetate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266020((4-(furan-2-yl)-2-(furan-2-ylmethylamino)thiazol-5...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266021((4-(furan-2-yl)-2-(thiophen-2-ylmethylamino)thiazo...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266022((2-(2-(benzo[d][1,3]dioxol-5-yl)ethylamino)-4-(fur...)
Affinity DataKi:  61nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266019((2-(3,4-difluorobenzylamino)-4-(furan-2-yl)thiazol...)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265981((4-(furan-2-yl)-2-(methylamino)thiazol-5-yl)(pheny...)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
South China University of Technology

Curated by ChEMBL
LigandPNGBDBM50233193(CHEMBL4062476)
Affinity DataKi:  88nMAssay Description:Inhibition of human liver carboxylesterase 1 using o-nitrophenyl acetate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266084((2-(benzyl(furan-2-ylmethyl)amino)-4-(furan-2-yl)t...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265982((4-(furan-2-yl)-2-(isobutylamino)thiazol-5-yl)(phe...)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
South China University of Technology

Curated by ChEMBL
LigandPNGBDBM50463531(CHEMBL4242425)
Affinity DataKi:  92nMAssay Description:Inhibition of human liver carboxylesterase 1 using o-nitrophenyl acetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266052((4-(furan-2-yl)-2-(3-phenylpropylamino)thiazol-5-y...)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266018((2-(1-(2-fluorobenzyl)piperidin-4-ylamino)-4-(fura...)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265984((4-(furan-2-yl)-2-(2-methoxypropylamino)thiazol-5-...)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266055((4-(furan-2-yl)-2-((furan-2-ylmethyl)(methyl)amino...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM82423(CAS_132947 | NSC_132947 | TRIPITRAMINE)
Affinity DataKi:  180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265983((4-(furan-2-yl)-2-(2-methoxyethylamino)thiazol-5-y...)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM82423(CAS_132947 | NSC_132947 | TRIPITRAMINE)
Affinity DataKi:  220nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265985(CHEMBL460172 | N-(2-(5-benzoyl-4-(furan-2-yl)thiaz...)
Affinity DataKi:  281nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  320nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265986(1-(4-(5-benzoyl-4-(furan-2-yl)thiazol-2-ylamino)pi...)
Affinity DataKi:  455nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  720nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265986(1-(4-(5-benzoyl-4-(furan-2-yl)thiazol-2-ylamino)pi...)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265982((4-(furan-2-yl)-2-(isobutylamino)thiazol-5-yl)(phe...)
Affinity DataKi:  1.28E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  1.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266020((4-(furan-2-yl)-2-(furan-2-ylmethylamino)thiazol-5...)
Affinity DataKi:  1.46E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Creighton University

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  1.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265985(CHEMBL460172 | N-(2-(5-benzoyl-4-(furan-2-yl)thiaz...)
Affinity DataKi:  2.42E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266054((2-(benzyl(methyl)amino)-4-(furan-2-yl)thiazol-5-y...)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266021((4-(furan-2-yl)-2-(thiophen-2-ylmethylamino)thiazo...)
Affinity DataKi:  2.99E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266055((4-(furan-2-yl)-2-((furan-2-ylmethyl)(methyl)amino...)
Affinity DataKi:  3.42E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266022((2-(2-(benzo[d][1,3]dioxol-5-yl)ethylamino)-4-(fur...)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265981((4-(furan-2-yl)-2-(methylamino)thiazol-5-yl)(pheny...)
Affinity DataKi:  3.58E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266018((2-(1-(2-fluorobenzyl)piperidin-4-ylamino)-4-(fura...)
Affinity DataKi:  3.71E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265984((4-(furan-2-yl)-2-(2-methoxypropylamino)thiazol-5-...)
Affinity DataKi:  3.97E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266052((4-(furan-2-yl)-2-(3-phenylpropylamino)thiazol-5-y...)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266051((4-(furan-2-yl)-2-(2-(thiophen-2-yl)ethylamino)thi...)
Affinity DataKi: >6.70E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50265983((4-(furan-2-yl)-2-(2-methoxyethylamino)thiazol-5-y...)
Affinity DataKi:  6.78E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266053((2-(dimethylamino)-4-(furan-2-yl)thiazol-5-yl)(phe...)
Affinity DataKi:  6.82E+3nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266086((2-(benzyl(2-(thiophen-2-yl)ethyl)amino)-4-(furan-...)
Affinity DataKi:  7.14E+3nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266019((2-(3,4-difluorobenzylamino)-4-(furan-2-yl)thiazol...)
Affinity DataKi: >7.50E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266085((4-(furan-2-yl)-2-(methyl(2-(thiophen-2-yl)ethyl)a...)
Affinity DataKi:  8.17E+3nMAssay Description:Displacement of [3H]SCH-58261 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266054((2-(benzyl(methyl)amino)-4-(furan-2-yl)thiazol-5-y...)
Affinity DataKi:  9.46E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266086((2-(benzyl(2-(thiophen-2-yl)ethyl)amino)-4-(furan-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50266085((4-(furan-2-yl)-2-(methyl(2-(thiophen-2-yl)ethyl)a...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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