Compile Data Set for Download or QSAR
maximum 50k data
Found 128 with Last Name = 'cha' and Initial = 'xy'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407214(CHEMBL2008608)
Affinity DataKi:  4.5nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029788(8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-...)
Affinity DataKi:  6.10nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataKi:  8.70nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataKi:  8.70nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407211(CHEMBL2111684)
Affinity DataKi:  9.40nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407211(CHEMBL2111684)
Affinity DataKi:  9.40nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  23.3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407213(CHEMBL2111685)
Affinity DataKi:  32nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  33.9nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407212(CHEMBL2111686)
Affinity DataKi:  36nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407213(CHEMBL2111685)
Affinity DataKi:  45nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029788(8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-...)
Affinity DataKi:  65.3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataKi:  121nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataKi:  122nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029790(5-(3-Methoxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  138nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029788(8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-...)
Affinity DataKi:  240nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407214(CHEMBL2008608)
Affinity DataKi:  271nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407211(CHEMBL2111684)
Affinity DataKi:  392nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataKi:  491nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407213(CHEMBL2111685)
Affinity DataKi: >500nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi: >500nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029788(8-[1-(3,4-Dichloro-phenyl)-meth-(E)-ylidene]-5-(3-...)
Affinity DataKi: >500nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407213(CHEMBL2111685)
Affinity DataKi: >500nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407214(CHEMBL2008608)
Affinity DataKi: >500nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407212(CHEMBL2111686)
Affinity DataKi:  505nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029782(5-(3-Hydroxy-phenyl)-2-methyl-8-[1-phenyl-meth-(E)...)
Affinity DataKi:  576nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50037188(5-(3-Hydroxy-phenyl)-2,2-dimethyl-7-oxo-8-[1-pheny...)
Affinity DataKi: >700nMAssay Description:Inhibition of radioligand [3H]-DAMGO binding to rat brain mu receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407212(CHEMBL2111686)
Affinity DataKi:  762nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407211(CHEMBL2111684)
Affinity DataKi:  889nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50037188(5-(3-Hydroxy-phenyl)-2,2-dimethyl-7-oxo-8-[1-pheny...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407211(CHEMBL2111684)
Affinity DataKi:  1.98E+3nMAssay Description:Inhibition of radioligand [3H]-DADLE binding to rat brain delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407212(CHEMBL2111686)
Affinity DataKi:  2.54E+3nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50407214(CHEMBL2008608)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50037188(5-(3-Hydroxy-phenyl)-2,2-dimethyl-7-oxo-8-[1-pheny...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50037189(5-(3-Methoxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50037188(5-(3-Hydroxy-phenyl)-2,2-dimethyl-7-oxo-8-[1-pheny...)
Affinity DataKi:  5.40E+3nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataKi:  3.18E+4nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataKi:  3.18E+4nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of [3H]DAMGO radioligand binding to rat brain opioid receptor mu 1.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of [3H]DAMGO radioligand binding to rat brain opioid receptor mu 1.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50034605(3-[16-methyl-10,16-diazatetracyclo[11.3.1.02,11.04...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of [3H]DAMGO radioligand binding to rat brain opioid receptor mu 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of [3H]-U-69,593 radioligand binding to Guinea pig Opioid receptor kappa 1; not determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of [3H]DADLE radioligand binding to rat brain opioid receptor delta 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of [3H]U-69593 radioligand binding to Guinea pig opioid receptor kappa 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  4.10nMAssay Description:Opioid activity against delta-receptor of isolated mouse vas deferens(MVD) at 30 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50034598((+) 3-[13-phenethyl-9,13-diazatetracyclo[10.3.1.02...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of [3H]DADLE radioligand binding to rat brain opioid receptor delta 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50034595(3-[13-pentyl-9,13-diazatetracyclo[10.3.1.02,10.03,...)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of [3H]DADLE radioligand binding to rat brain opioid receptor delta 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50034600((+) 3-[13-methyl-9,13-diazatetracyclo[10.3.1.02,10...)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of [3H]DADLE radioligand binding to rat brain opioid receptor delta 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  7.37nMAssay Description:Inhibition of [3H]DADLE radioligand binding to rat brain opioid receptor delta 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of [3H]DADLE radioligand binding to rat brain opioid receptor delta 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 128 total ) | Next | Last >>
Jump to: