Affinity DataKi: 27nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 196nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 636nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 813nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 926nMAssay Description:Compound was evaluated for its binding affinity towards Muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 2.25E+3nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 2.46E+3nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 2.69E+3nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 3.03E+3nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 3.07E+3nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 3.66E+3nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 5.38E+3nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 5.46E+3nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 5.64E+3nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 5.86E+3nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 7.06E+3nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+4nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+4nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+4nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 1.59E+4nMAssay Description:Compound was evaluated for its binding affinity towards Muscarinic acetylcholine receptor M1 in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 2.76E+4nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 3.81E+4nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
Affinity DataKi: 4.05E+4nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 6.55E+4nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor in rat cortexMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Southern California
Curated by ChEMBL
University Of Southern California
Curated by ChEMBL
Affinity DataIC50: <0.100nMAssay Description:Inhibition of MAO-A (unknown origin) expressed in mouse GL26 cells using 14C 5-hydroxytryptamine as substrate pre-incubated for 20 mins followed by s...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Southern California
Curated by ChEMBL
University Of Southern California
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of MAO-A (unknown origin) expressed in mouse GL26 cells using 14C 5-hydroxytryptamine as substrate pre-incubated for 20 mins followed by s...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of EGF-R or PDGFR-beta kinase autophosphorylation activity. The assay was performed in 96-well...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of EGF-R or PDGFR-beta kinase autophosphorylation activity. The assay was performed in 96-well...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Southern California
Curated by ChEMBL
University Of Southern California
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of MAO-A (unknown origin) expressed in mouse GL26 cells using 14C 5-hydroxytryptamine as substrate pre-incubated for 20 mins followed by s...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of EGF-R or PDGFR-beta kinase autophosphorylation activity. The assay was performed in 96-well...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of EGF-R or PDGFR-beta kinase autophosphorylation activity. The assay was performed in 96-well...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of EGF-R or PDGFR-beta kinase autophosphorylation activity. The assay was performed in 96-well...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of EGF-R or PDGFR-beta kinase autophosphorylation activity. The assay was performed in 96-well...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of EGF-R or PDGFR-beta kinase autophosphorylation activity. The assay was performed in 96-well...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Southern California
Curated by ChEMBL
University Of Southern California
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of MAO-A (unknown origin) expressed in mouse GL26 cells using 14C 5-hydroxytryptamine as substrate pre-incubated for 20 mins followed by s...More data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human recombinant HDAC6 expressed in baculovirus infected insect cells using [RHKK(Ac)] fluorogenic substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of EGF-R or PDGFR-beta kinase autophosphorylation activity. The assay was performed in 96-well...More data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Inhibition of human recombinant HDAC6 expressed in baculovirus infected insect cells using [RHKK(Ac)] fluorogenic substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human HDAC6 (379 to 382 residues) using RHKKAc fluorogenic peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:Inhibition of human recombinant HDAC1 expressed in baculovirus infected insect cells using [RHKK(Ac)] fluorogenic substrateMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human HDAC6 (379 to 382 residues) using RHKKAc fluorogenic peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human HDAC6 (379 to 382 residues) using RHKKAc fluorogenic peptide as substrate by fluorescence assayMore data for this Ligand-Target Pair