Affinity DataKi: 1nMAssay Description:Evaluated for the Non competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 51nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 530nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 610nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 870nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
University of Dundee
Curated by PDSP Ki Database
University of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 3.20E+3nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair