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Found 155 with Last Name = 'cui' and Initial = 'r'
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504104(CHEMBL4446835)
Affinity DataKi:  1.90nMAssay Description:Irreversible inhibition of human FGFR1 using poly (Glu, Tyr)4:1 as substrate measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504106(CHEMBL4462946)
Affinity DataKi:  10nMAssay Description:Irreversible inhibition of human FGFR1 using poly (Glu, Tyr)4:1 as substrate measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50470518(CHEMBL4294523)
Affinity DataKi:  740nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50470513(CHEMBL4290712)
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50470517(CHEMBL4294114)
Affinity DataKi:  1.18E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50470512(CHEMBL1416382)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50470515(CHEMBL4291509)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50470514(CHEMBL4283640)
Affinity DataKi:  3.92E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50470516(CHEMBL4282824)
Affinity DataKi:  8.87E+3nMAssay Description:Inhibition of Cy5-labeled double-strand DNA probe binding to STAT3 (unknown origin) expressed in H1299 cell lysates assessed as decrease in DNA bindi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259656(CHEMBL4089402)
Affinity DataIC50:  0.000200nMAssay Description:Dissociation constant against galectin-3 using competitive fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259645(CHEMBL4070336)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human HL60 cells using Suc-LLVYaminoluciferin as substrate after 2 hrs by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504107(CHEMBL4448252)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human FGFR1 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50065454(CHEBI:63453 | CHEMBL3348846)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human FGFR2 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50065454(CHEBI:63453 | CHEMBL3348846)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human FGFR1 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504108(CHEMBL4467025)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human FGFR1 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504108(CHEMBL4467025)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human FGFR2 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504104(CHEMBL4446835)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human FGFR1 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504104(CHEMBL4446835)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human FGFR2 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504103(CHEMBL4463714)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human FGFR2 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504107(CHEMBL4448252)
Affinity DataIC50:  2nMAssay Description:Inhibition of human FGFR2 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259647(CHEMBL4100727)
Affinity DataIC50:  2nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human HL60 cells using Suc-LLVYaminoluciferin as substrate after 2 hrs by fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259657(CHEMBL4068221)
Affinity DataIC50:  2nMAssay Description:Dissociation constant against galectin-3 using competitive fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504103(CHEMBL4463714)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human FGFR1 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259659(CHEMBL4076838)
Affinity DataIC50:  3nMAssay Description:Dissociation constant against galectin-3 using competitive fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50065454(CHEBI:63453 | CHEMBL3348846)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human FGFR3 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  4nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human HL60 cells using Suc-LLVYaminoluciferin as substrate after 2 hrs by fluorescence ...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259642(CHEMBL4077037)
Affinity DataIC50:  4nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human HL60 cells using Suc-LLVYaminoluciferin as substrate after 2 hrs by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504102(CHEMBL4541330)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human FGFR2 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504106(CHEMBL4462946)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of human FGFR2 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504109(CHEMBL4447110)
Affinity DataIC50:  8nMAssay Description:Inhibition of human FGFR2 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582160(CHEMBL5072982)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259641(CHEMBL484701)
Affinity DataIC50:  10nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human HL60 cells using Suc-LLVYaminoluciferin as substrate after 2 hrs by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259655(CHEMBL4080306)
Affinity DataIC50:  10nMAssay Description:Dissociation constant against galectin-3 using competitive fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582161(CHEMBL5076889)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504105(CHEMBL4586512)
Affinity DataIC50:  11nMAssay Description:Inhibition of human FGFR1 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259646(CHEMBL4075225)
Affinity DataIC50:  12nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human HL60 cells using Suc-LLVYaminoluciferin as substrate after 2 hrs by fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504102(CHEMBL4541330)
Affinity DataIC50:  13nMAssay Description:Inhibition of human FGFR3 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504104(CHEMBL4446835)
Affinity DataIC50:  15nMAssay Description:Inhibition of human FGFR3 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504102(CHEMBL4541330)
Affinity DataIC50:  16nMAssay Description:Inhibition of human FGFR1 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504106(CHEMBL4462946)
Affinity DataIC50:  20nMAssay Description:Inhibition of human FGFR1 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259656(CHEMBL4089402)
Affinity DataIC50:  20nMAssay Description:Inhibition of caspase-like activity of 20S proteasome in human HL60 cells using Z-nLPnLDaminoluciferin as substrate after 2 hrs by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259649(CHEMBL4077282)
Affinity DataIC50:  20nMAssay Description:Dissociation constant against galectin-3 using competitive fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50259658(CHEMBL4096371)
Affinity DataIC50:  20nMAssay Description:Dissociation constant against galectin-3 using competitive fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504104(CHEMBL4446835)
Affinity DataIC50:  23nMAssay Description:Inhibition of human FGFR4 using poly (Glu, Tyr)4:1 as substrate measured after 60 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetInactive serine/threonine-protein kinase 19(Homo sapiens (Human))
Trustees of Boston University

US Patent
LigandPNGBDBM588065(US11542240, Formula number IV)
Affinity DataIC50:  24nMAssay Description:The optimal amount of STK19 is the minimal amount that produces luminescence within the linear portion of the kinase titration curve and generates an...More data for this Ligand-Target Pair
Ligand InfoPurchase
In DepthDetails US Patent
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Bytedance Ai Lab

Curated by ChEMBL
LigandPNGBDBM50582159(CHEMBL5082740)
Affinity DataIC50:  28nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInactive serine/threonine-protein kinase 19(Homo sapiens (Human))
Trustees of Boston University

US Patent
LigandPNGBDBM588081(US11542240, Formula number XLVI)
Affinity DataIC50:  29.3nMAssay Description:The optimal amount of STK19 is the minimal amount that produces luminescence within the linear portion of the kinase titration curve and generates an...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504110(CHEMBL4577458)
Affinity DataIC50:  30nMAssay Description:Inhibition of human ERG by patch-clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  30nMAssay Description:Inhibition of caspase-like activity of 20S proteasome in human HL60 cells using Z-nLPnLDaminoluciferin as substrate after 2 hrs by fluorescence analy...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50504113(CHEMBL4537540)
Affinity DataIC50:  30nMAssay Description:Inhibition of human ERG by patch-clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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