Affinity DataKi: 1nMAssay Description:Displacement of [3H]-DAMGO (2 nM ) from opioid receptor mu 1 in human brainMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]-DAMGO (2 nM ) from opioid receptor mu 1 in human brainMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A/B(Homo sapiens (Human))
Instituto De QuíMica MéDica
Curated by ChEMBL
Instituto De QuíMica MéDica
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]-2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]-DAMGO (2 nM ) from opioid receptor mu 1 in human brainMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A/B(Homo sapiens (Human))
Instituto De QuíMica MéDica
Curated by ChEMBL
Instituto De QuíMica MéDica
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Displacement of [3H]-2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of [3H]-DAMGO (2 nM ) from opioid receptor mu 1 in human brainMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A/B(Homo sapiens (Human))
Instituto De QuíMica MéDica
Curated by ChEMBL
Instituto De QuíMica MéDica
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Displacement of [3H]-2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 360nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A/B(Homo sapiens (Human))
Instituto De QuíMica MéDica
Curated by ChEMBL
Instituto De QuíMica MéDica
Curated by ChEMBL
Affinity DataKi: 409nMAssay Description:Displacement of [3H]-2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
Affinity DataKi: 433nMAssay Description:Displacement of [3H]-DAMGO (2 nM ) from opioid receptor mu 1 in human brainMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A/B(Homo sapiens (Human))
Instituto De QuíMica MéDica
Curated by ChEMBL
Instituto De QuíMica MéDica
Curated by ChEMBL
Affinity DataKi: 437nMAssay Description:Displacement of [3H]-2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
Affinity DataKi: 477nMAssay Description:Displacement of [3H]-DAMGO (2 nM ) from opioid receptor mu 1 in human brainMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 1.52E+3nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A/B(Homo sapiens (Human))
Instituto De QuíMica MéDica
Curated by ChEMBL
Instituto De QuíMica MéDica
Curated by ChEMBL
Affinity DataKi: 1.92E+3nMAssay Description:Displacement of [3H]-2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 2.54E+3nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Binding affinity to recombinant Trypanosoma brucei brucei 427 alternative oxidase expressed in Escherichia coli BL21 cells using ubiquinol-1 as subst...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A/B(Homo sapiens (Human))
Instituto De QuíMica MéDica
Curated by ChEMBL
Instituto De QuíMica MéDica
Curated by ChEMBL
Affinity DataKi: 5.46E+3nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 1.07E+4nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 3.92E+4nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 4.00E+4nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 1.09E+5nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 1.92E+5nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 1.98E+5nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 5.88E+5nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 6.25E+5nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 7.14E+5nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 7.70E+5nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University
Curated by ChEMBL
Cardiff University
Curated by ChEMBL
Affinity DataKi: 7.84E+5nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol as substrate preincubated for 2 mins followed by substrate ad...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol-1 as substrate incubated for 2 mins followed by substrate add...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol-1 as substrate incubated for 2 mins followed by substrate add...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol-1 as substrate incubated for 2 mins followed by substrate add...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 9.10nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol-1 as substrate incubated for 2 mins followed by substrate add...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol-1 as substrate incubated for 2 mins followed by substrate add...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol-1 as substrate incubated for 2 mins followed by substrate add...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol as substrate preincubated for 2 mins followed by substrate ad...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol-1 as substrate incubated for 2 mins followed by substrate add...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 145nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol as substrate preincubated for 2 mins followed by substrate ad...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol-1 as substrate incubated for 2 mins followed by substrate add...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol as substrate preincubated for 2 mins followed by substrate ad...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol as substrate preincubated for 2 mins followed by substrate ad...More data for this Ligand-Target Pair
TargetAlternative oxidase, mitochondrial(Trypanosoma brucei brucei)
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Instituto De Qu£Mica M£Dica
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of recombinant Trypanosoma brucei brucei alternative oxidase using ubiquinol-1 as substrate incubated for 2 mins followed by substrate add...More data for this Ligand-Target Pair