Compile Data Set for Download or QSAR
maximum 50k data
Found 61 with Last Name = 'figueroa' and Initial = 'm'
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50266275(CHEMBL456494 | Tajixanthone hydrate)
Affinity DataKi:  1.39E+4nMAssay Description:Inhibition of recombinant calmodulin (unknown origin) mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release using v...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  1.93E+4nMAssay Description:Inhibition of recombinant calmodulin (unknown origin) mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release using v...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50266274(14-methoxytajixanthone | CHEMBL515370)
Affinity DataKi:  2.54E+4nMAssay Description:Inhibition of recombinant calmodulin (unknown origin) mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release using v...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020375(CHEMBL3289785)
Affinity DataIC50:  12nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human PDE4B2More data for this Ligand-Target Pair
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50081950(6-Hydroxy-2-phenyl-chromen-4-one | 6-Hydroxyflavon...)
Affinity DataIC50:  5.17E+3nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50266274(14-methoxytajixanthone | CHEMBL515370)
Affinity DataIC50:  5.54E+3nMAssay Description:Inhibition of recombinant calmodulin (unknown origin) mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release by spec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50266275(CHEMBL456494 | Tajixanthone hydrate)
Affinity DataIC50:  5.62E+3nMAssay Description:Inhibition of recombinant calmodulin (unknown origin) mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release by spec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50601437(CHEMBL5207648)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50601435(CHEMBL5204172)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataIC50:  7.26E+3nMAssay Description:Inhibition of recombinant calmodulin (unknown origin) mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release by spec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020376(CHEBI:81348 | CHEMBL290932)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020377(CHEMBL3289786)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346822(CHEMBL66917)
Affinity DataIC50:  9.38E+3nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50266273(15-chlorotajixanthone hydrate | CHEMBL458017)
Affinity DataIC50:  9.59E+3nMAssay Description:Inhibition of recombinant calmodulin (unknown origin) mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release by spec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50601436(CHEMBL5186891)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50540270(CHEMBL4646089)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of human PTP1B expressed in Escherichia coli BL21 (DE3) cells using PNPP as substate preincubated for 5 mins followed by substrate additon...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50601433(CHEMBL2152644)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human recombinant PTP1B (1 to 322 residues) expressed in Escherichia coli using pNPP as substrate incubated for 10 mins followed by sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50540269(CHEMBL4647463)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of human PTP1B expressed in Escherichia coli BL21 (DE3) cells using PNPP as substate preincubated for 5 mins followed by substrate additon...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50540272((+)-Malbrancheamide | CHEMBL508749)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of human PTP1B expressed in Escherichia coli BL21 (DE3) cells using PNPP as substate preincubated for 5 mins followed by substrate additon...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346811(CHEMBL1796022)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50540271(CHEMBL4638865)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of human PTP1B expressed in Escherichia coli BL21 (DE3) cells using PNPP as substate preincubated for 5 mins followed by substrate additon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50601434(CHEBI:4041 | CYPERIN | Cyperin)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human recombinant PTP1B (1 to 322 residues) expressed in Escherichia coli using pNPP as substrate incubated for 10 mins followed by sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50428912(Betulinan C | CHEMBL2331809)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human PDE4B2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346820(CHEMBL1796013)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020378(CHEMBL3289787)
Affinity DataIC50:  1.98E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM23419((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dihydro...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346810(CHEMBL268559)
Affinity DataIC50:  2.25E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346806(CHEMBL1796026)
Affinity DataIC50:  2.29E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020379(CHEMBL3289788)
Affinity DataIC50:  2.65E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Jordan University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  2.78E+4nMAssay Description:Inhibition of human PTP1B expressed in Escherichia coli BL21 (DE3) cells using PNPP as substate preincubated for 5 mins followed by substrate additon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50242273(CHEMBL469860 | shamixanthone)
Affinity DataIC50:  2.92E+4nMAssay Description:Inhibition of recombinant calmodulin (unknown origin) mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release by spec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50020380(CHEMBL3289789)
Affinity DataIC50:  3.01E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346819(CHEMBL1796014)
Affinity DataIC50:  3.01E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM115127(4,5,7-trihydroxy-9,10-diketo-anthracene-2-carboxyl...)
Affinity DataIC50:  3.06E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50428913(CHEMBL2331810)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of human PDE4B2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346821(CHEMBL1796012)
Affinity DataIC50:  3.13E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346805(CHEMBL1796027)
Affinity DataIC50:  3.25E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM7461(5,7-dihydroxy-2-phenyl-4H-chromen-4-one | 5,7-dihy...)
Affinity DataIC50:  3.34E+4nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346818(CHEMBL1796015)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM26664(7-Hydroxy-flavone, 5a | 7-Hydroxyflavone, 11 | 7-h...)
Affinity DataIC50:  3.71E+4nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346809(CHEMBL1796023)
Affinity DataIC50:  3.77E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50312649(6-chloro-4,5,7-trihydroxy-9,10-dioxo-9,10-dihydroa...)
Affinity DataIC50:  3.78E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
University Of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50428914(BETULINAN A)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of human PDE4B2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346815(CHEMBL1796017)
Affinity DataIC50:  4.61E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346814(CHEMBL1796018)
Affinity DataIC50:  5.47E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalmodulin-1(Human)
Universidad Nacional AutóNoma De MéXico

Curated by ChEMBL
LigandPNGBDBM50346812(CHEMBL1796021)
Affinity DataIC50:  5.47E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 61 total ) | Next | Last >>
Jump to: