Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 135nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 165nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 194nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 215nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 266nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 447nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 505nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 523nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 554nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 603nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 741nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid
Curated by ChEMBL
Universidad Complutense De Madrid
Curated by ChEMBL
Affinity DataKi: 747nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 913nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
Affinity DataKi: 1.01E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
Affinity DataKi: 1.05E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
Affinity DataKi: 2.09E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
TargetPhospholipase C(Bacillus cereus)
Institute Of Advance Chemistry Of Catalonia (Iqac-Csic)
Curated by ChEMBL
Institute Of Advance Chemistry Of Catalonia (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Mixed-type inhibition of Bacillus cereus phosphatidylcholine preferred phospholipase C by Dixon plot analysisMore data for this Ligand-Target Pair
TargetPhospholipase C(Bacillus cereus)
Institute Of Advance Chemistry Of Catalonia (Iqac-Csic)
Curated by ChEMBL
Institute Of Advance Chemistry Of Catalonia (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Non-competitive inhibition of Bacillus cereus phosphatidylcholine preferred phospholipase C by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.41E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
TargetPhospholipase C(Bacillus cereus)
Institute Of Advance Chemistry Of Catalonia (Iqac-Csic)
Curated by ChEMBL
Institute Of Advance Chemistry Of Catalonia (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Uncompetitive inhibition of Bacillus cereus phosphatidylcholine preferred phospholipase C by Dixon plot analysisMore data for this Ligand-Target Pair
TargetPhospholipase C(Bacillus cereus)
Institute Of Advance Chemistry Of Catalonia (Iqac-Csic)
Curated by ChEMBL
Institute Of Advance Chemistry Of Catalonia (Iqac-Csic)
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Mixed-type inhibition of Bacillus cereus phosphatidylcholine preferred phospholipase C by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.33E+4nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 7.80nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter
Curated by ChEMBL
Alter
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Ex vivo inhibitory concentration against human choline kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against human choline kinase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Ex vivo inhibitory concentration against human choline kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Ex vivo inhibitory concentration against human choline kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of human DNA topoisomerase 1More data for this Ligand-Target Pair