Affinity DataKi: 5.10nMAssay Description:TP_TRANSPORTER: inhibition of Dopamine uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:TP_TRANSPORTER: inhibition of Adrenaline uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:TP_TRANSPORTER: inhibition of Noradrenaline uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:TP_TRANSPORTER: inhibition of Serotonin uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg
Curated by ChEMBL
University Of Heidelberg
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg
Curated by ChEMBL
University Of Heidelberg
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:TP_TRANSPORTER: inhibition of Dopamine uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:TP_TRANSPORTER: inhibition of Adrenaline uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:TP_TRANSPORTER: inhibition of Noradrenaline uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 605nMAssay Description:TP_TRANSPORTER: inhibition of Serotonin uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 670nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 930nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg
Curated by ChEMBL
University Of Heidelberg
Curated by ChEMBL
Affinity DataKi: 1.40E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.90E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+6nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+6nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+6nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.60E+6nMAssay Description:TP_TRANSPORTER: inhibition of uptake of 0.1 uM MPP+ in OCT1-expressing 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+7nMAssay Description:TP_TRANSPORTER: inhibition of uptake of 0.1 uM MPP+ in OCT1-expressing 293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg
Curated by ChEMBL
University Of Heidelberg
Curated by ChEMBL
Affinity DataIC50: 1.76E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.2 uM) in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg
Curated by ChEMBL
University Of Heidelberg
Curated by ChEMBL
Affinity DataIC50: 7.93E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.2 uM) in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg
Curated by ChEMBL
University Of Heidelberg
Curated by ChEMBL
Affinity DataIC50: 1.03E+7nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.2 uM) in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair