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Found 707 with Last Name = 'hansen' and Initial = 'kb'
TargetGlutamate receptor 3(RAT)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50059672((S)-2-AMINO-3-[3-HYDROXY-5-(2-METHYL-2H-TETRAZOL-5...)
Affinity DataKi:  2.20nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50059672((S)-2-AMINO-3-[3-HYDROXY-5-(2-METHYL-2H-TETRAZOL-5...)
Affinity DataKi:  2.70nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA4 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50059672((S)-2-AMINO-3-[3-HYDROXY-5-(2-METHYL-2H-TETRAZOL-5...)
Affinity DataKi:  3.90nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50059672((S)-2-AMINO-3-[3-HYDROXY-5-(2-METHYL-2H-TETRAZOL-5...)
Affinity DataKi:  5.20nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA1 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512945((S)-AMPA)
Affinity DataKi:  17nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(RAT)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512945((S)-AMPA)
Affinity DataKi:  21nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512945((S)-AMPA)
Affinity DataKi:  22nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA1 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512945((S)-AMPA)
Affinity DataKi:  40nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA4 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50318264((+)-2-Amino-3-(4-hydroxy-1,2,5-oxadiazol-3-yl)prop...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]AMPA from rat iGluR2 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50318264((+)-2-Amino-3-(4-hydroxy-1,2,5-oxadiazol-3-yl)prop...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]AMPA from rat iGluR2 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2A(Rattus norvegicus (Rat))
University of Copenhagen

LigandPNGBDBM213889(5,7-Dichlorokynurenic acid (5,7-DCKA))
Affinity DataKi:  65nM ΔG°:  -41.0kJ/mole IC50:  92nMpH: 7.4 T: 2°CAssay Description:Two-electrode voltage clamp (TEVC) recordings were performed on Xenopus oocytes at room temperature 3-6 days postinjection using an OC-725C TEVC ampl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]SYM2081 from rat iGluR5 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50211399((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Affinity DataKi:  200nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA4 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]AMPA from rat iGluR2 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2D(Rattus norvegicus (Rat))
University of Copenhagen

LigandPNGBDBM213888(1-thioxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]-quinox...)
Affinity DataKi: >300nM ΔG°: >-37.2kJ/mole IC50: >3.00E+3nMpH: 7.4 T: 2°CAssay Description:Two-electrode voltage clamp (TEVC) recordings were performed on Xenopus oocytes at room temperature 3-6 days postinjection using an OC-725C TEVC ampl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512944(CHEMBL4529665)
Affinity DataKi:  320nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2-ABD expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]SYM2081 from rat iGluR6 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50211399((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Affinity DataKi:  390nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  390nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]SYM2081 from rat iGluR7 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2A(Rattus norvegicus (Rat))
University of Copenhagen

LigandPNGBDBM213888(1-thioxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]-quinox...)
Affinity DataKi:  560nM ΔG°:  -35.7kJ/mole IC50:  770nMpH: 7.4 T: 2°CAssay Description:Two-electrode voltage clamp (TEVC) recordings were performed on Xenopus oocytes at room temperature 3-6 days postinjection using an OC-725C TEVC ampl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512944(CHEMBL4529665)
Affinity DataKi:  710nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50211399((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Affinity DataKi:  750nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
University of Copenhagen

LigandPNGBDBM213888(1-thioxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]-quinox...)
Affinity DataKi: >800nM ΔG°: >-34.8kJ/mole IC50: >3.00E+3nMpH: 7.4 T: 2°CAssay Description:Two-electrode voltage clamp (TEVC) recordings were performed on Xenopus oocytes at room temperature 3-6 days postinjection using an OC-725C TEVC ampl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
University of Copenhagen

LigandPNGBDBM213888(1-thioxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]-quinox...)
Affinity DataKi: >1.30E+3nM ΔG°: >-33.6kJ/mole IC50: >3.00E+3nMpH: 7.4 T: 2°CAssay Description:Two-electrode voltage clamp (TEVC) recordings were performed on Xenopus oocytes at room temperature 3-6 days postinjection using an OC-725C TEVC ampl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512939(CHEMBL3742451)
Affinity DataKi:  1.87E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512944(CHEMBL4529665)
Affinity DataKi:  1.91E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512940(CHEMBL3742450)
Affinity DataKi:  1.97E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2-ABD expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  2.80E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2B expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512941(CHEMBL4556711)
Affinity DataKi:  3.25E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512939(CHEMBL3742451)
Affinity DataKi:  4.08E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA4 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512940(CHEMBL3742450)
Affinity DataKi:  4.38E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  4.70E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(RAT)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512940(CHEMBL3742450)
Affinity DataKi:  4.89E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutamate receptor 3(RAT)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512939(CHEMBL3742451)
Affinity DataKi:  4.98E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  5.90E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2C expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50211399((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Affinity DataKi:  7.70E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA1 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318264((+)-2-Amino-3-(4-hydroxy-1,2,5-oxadiazol-3-yl)prop...)
Affinity DataKi:  8.10E+3nMAssay Description:Displacement of [3H]SYM2081 from rat iGluR5 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50318264((+)-2-Amino-3-(4-hydroxy-1,2,5-oxadiazol-3-yl)prop...)
Affinity DataKi:  8.10E+3nMAssay Description:Displacement of [3H]SYM2081 from rat iGluR5 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512944(CHEMBL4529665)
Affinity DataKi:  9.02E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA1 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512944(CHEMBL4529665)
Affinity DataKi:  9.47E+3nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA4 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  1.00E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2B expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50246919(CHEMBL4099104)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512940(CHEMBL3742450)
Affinity DataKi:  1.16E+4nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA4 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGlutamate receptor 3(RAT)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512941(CHEMBL4556711)
Affinity DataKi:  1.19E+4nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50246919(CHEMBL4099104)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50512939(CHEMBL3742451)
Affinity DataKi:  1.57E+4nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA1 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50318266((+)-2-Amino-5-(4-hydroxy-1,2,5-oxadiazol-3-yl)pent...)
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]AMPA from rat iGluR2 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2D(RAT)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  2.10E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2D expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  2.40E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2C expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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