Compile Data Set for Download or QSAR
maximum 50k data
Found 47 with Last Name = 'ji' and Initial = 'tf'
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50109277(CHEMBL3601686)
Affinity DataIC50:  3.5nMAssay Description:Modulation of P-gp (unknown origin) transfected in human MDA435/LCC6MDR cells assessed as paclitaxel IC50 for cell growth inhibition at 1 uM after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50109278(CHEMBL3601685)
Affinity DataIC50:  6.5nMAssay Description:Modulation of P-gp (unknown origin) transfected in human MDA435/LCC6MDR cells assessed as paclitaxel IC50 for cell growth inhibition at 1 uM after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50109344(CHEMBL3601682)
Affinity DataIC50:  11nMAssay Description:Modulation of P-gp (unknown origin) transfected in human MDA435/LCC6MDR cells assessed as paclitaxel IC50 for cell growth inhibition at 1 uM after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50109279(CHEMBL3601684)
Affinity DataIC50:  14nMAssay Description:Modulation of P-gp (unknown origin) transfected in human MDA435/LCC6MDR cells assessed as paclitaxel IC50 for cell growth inhibition at 1 uM after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50109314(CHEMBL3601683)
Affinity DataIC50:  25nMAssay Description:Modulation of P-gp (unknown origin) transfected in human MDA435/LCC6MDR cells assessed as paclitaxel IC50 for cell growth inhibition at 1 uM after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50109274(CHEMBL3601689)
Affinity DataIC50:  26nMAssay Description:Modulation of P-gp (unknown origin) transfected in human MDA435/LCC6MDR cells assessed as paclitaxel IC50 for cell growth inhibition at 1 uM after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50109275(CHEMBL3601688)
Affinity DataIC50:  58nMAssay Description:Modulation of P-gp (unknown origin) transfected in human MDA435/LCC6MDR cells assessed as paclitaxel IC50 for cell growth inhibition at 1 uM after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50109276(CHEMBL3601687)
Affinity DataIC50:  126nMAssay Description:Modulation of P-gp (unknown origin) transfected in human MDA435/LCC6MDR cells assessed as paclitaxel IC50 for cell growth inhibition at 1 uM after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50109273(CHEMBL3601690)
Affinity DataIC50:  136nMAssay Description:Modulation of P-gp (unknown origin) transfected in human MDA435/LCC6MDR cells assessed as paclitaxel IC50 for cell growth inhibition at 1 uM after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400427(CHEMBL2178445)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400420(CHEMBL2178452)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50193394(CHEMBL536352)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of serotonin transporter (unknown origin) assessed as suppression of synaptosomal uptake of serotoninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400416(CHEMBL2178456)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50193394(CHEMBL536352)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of dopamine transporter (unknown origin) assessed as suppression of synaptosomal uptake of dopamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400418(CHEMBL2178454)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50193394(CHEMBL536352)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of norepinephrine transporter (unknown origin) assessed as suppression of synaptosomal uptake of norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50193079(CHEBI:5834 | CHEMBL1237210)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of dopamine transporter (unknown origin) assessed as suppression of synaptosomal uptake of dopamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50193079(CHEBI:5834 | CHEMBL1237210)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of norepinephrine transporter (unknown origin) assessed as suppression of synaptosomal uptake of norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Chinese Academy Of Medical Sciences And Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50193079(CHEBI:5834 | CHEMBL1237210)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of serotonin transporter (unknown origin) assessed as suppression of synaptosomal uptake of serotoninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400424(CHEMBL2178448)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400429(CHEMBL2178443)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400428(CHEMBL2178444)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400415(CHEMBL2178457)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400426(CHEMBL2178446)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400425(CHEMBL2178447)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400435(CHEMBL2177806)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400431(CHEMBL2177810)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400423(CHEMBL2178449)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400419(CHEMBL2178453)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400440(CHEMBL2177801)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400430(CHEMBL2177811)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400434(CHEMBL2177807)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400432(CHEMBL2177809)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400433(CHEMBL2177808)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400417(CHEMBL2178455)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400439(CHEMBL2177802)
Affinity DataIC50:  5.60E+4nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400442(CHEMBL2178460)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400421(CHEMBL2178451)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400438(CHEMBL2177803)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400437(CHEMBL2177804)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400444(CHEMBL2178458)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400443(CHEMBL2178459)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400441(CHEMBL2177800)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400436(CHEMBL2177805)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicative DNA helicase(Bacillus anthracis)
Microbiotix

Curated by ChEMBL
LigandPNGBDBM50400422(CHEMBL2178450)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Bacillus anthracis Sterne 34F2 replicative DNA helicase-mediated ATP-dependent dissociation of Hel-5'FAM:Hel-3'BHQ by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50109277(CHEMBL3601686)
Affinity DataEC50:  423nMAssay Description:Modulation of P-gp in human MDA435/LCC6MDR cells assessed as reversal of paclitaxel resistanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)
Affinity DataEC50:  446nMAssay Description:Modulation of P-gp in human MDA435/LCC6MDR cells assessed as reversal of paclitaxel resistanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed