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Found 71 with Last Name = 'lockman' and Initial = 'pr'
TargetHigh affinity choline transporter 1(Rattus norvegicus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50323515(CHEMBL1209714 | Hemicholinium)
Affinity DataKi:  10nMAssay Description:Binding affinity to rat choline transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416502(CHEMBL1209654)
Affinity DataKi:  20.0nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416489(CHEMBL1209507)
Affinity DataKi:  50nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416490(CHEMBL1209508)
Affinity DataKi:  90.0nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416491(CHEMBL1209577)
Affinity DataKi:  180nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416508(CHEMBL1209578)
Affinity DataKi:  200nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416504(CHEMBL1209579)
Affinity DataKi:  230nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416506(CHEMBL1209581)
Affinity DataKi:  521nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416503(CHEMBL1209713)
Affinity DataKi:  640nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50026220(2-hydroxy-N,N,N-trimethylethanaminium | CHEMBL2824...)
Affinity DataKi:  681nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416501(CHEMBL1209653)
Affinity DataKi:  701nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416488(CHEMBL1209506)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50143301((2-Hydroxy-ethyl)-dimethyl-octyl-ammonium | CHEMBL...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of [3H]choline brain uptake through choline transporter was determined in situ brain perfusion studies in Male Fischer-344 ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50147119((3-Hydroxy-propyl)-trimethyl-ammonium | CHEMBL1209...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50143312(CHEMBL53882 | Hexyl-(2-hydroxy-ethyl)-dimethyl-amm...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50204415(1-methyl-1-azonia-bicyclo[2.2.2]octane | CHEMBL120...)
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50060526(2-Dimethylamino-ethanol | 2-hydroxy-N,N-dimethylet...)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of [3H]choline brain uptake through choline transporter was determined in situ brain perfusion studies in Male Fischer-344 ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50079455(CHEMBL46486 | tetramethylammonium)
Affinity DataKi:  3.01E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147117(1-Octyl-piperidine | CHEMBL105218)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM80992(1-cetylpyridin-1-ium;bromide | 1-hexadecylpyridin-...)
Affinity DataKi:  3.21E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147114(Butyl-(2-hydroxy-ethyl)-dimethyl-ammonium | CHEMBL...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416495(CHEMBL1209648)
Affinity DataKi:  4.01E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026220(2-hydroxy-N,N,N-trimethylethanaminium | CHEMBL2824...)
Affinity DataKi:  4.20E+4nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147104(3-(1-Methyl-pyrrolidin-2-yl)-1-octyl-piperidine | ...)
Affinity DataKi:  4.50E+4nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50060526(2-Dimethylamino-ethanol | 2-hydroxy-N,N-dimethylet...)
Affinity DataKi:  5.57E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416507(CHEMBL1209649)
Affinity DataKi:  7.21E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM80386(CHEMBL1209421 | MLS000069658 | PHENYLTRIMETHYLAMMO...)
Affinity DataKi:  7.52E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147116(CHEMBL105536 | Ethyl-(2-hydroxy-ethyl)-dimethyl-am...)
Affinity DataKi:  9.40E+4nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416505(CHEMBL1209580)
Affinity DataKi:  1.07E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147122(2-(Dimethyl-lambda*4*-sulfanyl)-ethanol | CHEMBL54...)
Affinity DataKi:  1.17E+5nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147120(2-Methylamino-ethanol | 2-hydroxy-N-methylethanami...)
Affinity DataKi:  1.27E+5nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147119((3-Hydroxy-propyl)-trimethyl-ammonium | CHEMBL1209...)
Affinity DataKi:  1.62E+5nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147103((2-Hydroxy-ethyl)-dimethyl-propyl-ammonium | CHEMB...)
Affinity DataKi:  1.90E+5nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416484(CHEMBL1209503)
Affinity DataKi:  1.90E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50047005(1-Aza-bicyclo[2.2.2]octan-3-ol | 1-Aza-bicyclo[2.2...)
Affinity DataKi:  2.00E+5nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147112(2-hydroxy-N,N,N-trimethylpropanaminium | 2-methylc...)
Affinity DataKi:  2.00E+5nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50047005(1-Aza-bicyclo[2.2.2]octan-3-ol | 1-Aza-bicyclo[2.2...)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416496(CHEMBL1209650)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416485(CHEMBL1209504)
Affinity DataKi:  2.70E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416483(CHEMBL1209424)
Affinity DataKi:  2.90E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50147105((4-Hydroxy-butyl)-trimethyl-ammonium | CHEMBL10228...)
Affinity DataKi:  3.10E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416499(TRIMETHYLAMMONIUM)
Affinity DataKi:  3.40E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416486(CHEMBL1209505)
Affinity DataKi:  3.40E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50416500(CHEMBL1209652)
Affinity DataKi:  3.61E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147108(2-Hydroxy-4,4-dimethyl-2-phenyl-morpholin-4-ium | ...)
Affinity DataKi:  3.84E+5nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM10458(4-AP | 4-Aminopyridine 10 | CHEMBL284348 | DALFAMP...)
Affinity DataKi:  4.81E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147124(1-(4-Phenethyl-cyclohex-1-enyl)-ethanone | CHEMBL1...)
Affinity DataKi:  4.95E+5nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
Affinity DataKi:  5.20E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50147118((2-Hydroxy-cyclohexyl)-trimethyl-ammonium | CHEMBL...)
Affinity DataKi:  5.74E+5nMAssay Description:Inhibition of [3H]-choline brain uptake was determined by in situ brain perfusion studies in male ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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