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Found 417 with Last Name = 'malmberg' and Initial = 'a'
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]-quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054342(8-{4-[((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  0.246nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054342(8-{4-[((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50005118((S)-3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)...)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.660nMAssay Description:Inhibition of [3H]-raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50005118((S)-3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  2.74nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054338(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  4.42nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054333(8-[4-((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2...)
Affinity DataKi:  4.94nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054342(8-{4-[((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  4.94nMAssay Description:Displacement of [3H]-quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080053(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054333(8-[4-((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2...)
Affinity DataKi:  6.46nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50053670(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  8.62nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  13.2nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054342(8-{4-[((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H]-raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080047((4-Methoxy-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahyd...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054337(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  23.8nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50053670(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50053670(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054337(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  28.8nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50053670(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  30.2nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50349984(CHEMBL1813048)
Affinity DataKi:  35nMAssay Description:Binding affinity to inactivated human sodium channel Nav1.7 expressed in human HEK293 cells by patch-clamp electrophysiological assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054336(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  35.8nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054333(8-[4-((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080048((4-Fluoro-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahydr...)
Affinity DataKi:  43.8nMAssay Description:Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054338(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  44.5nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080053(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054338(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080050(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080047((4-Methoxy-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahyd...)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080051(Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthale...)
Affinity DataKi:  65.6nMAssay Description:Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054333(8-[4-((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2...)
Affinity DataKi:  68nMAssay Description:Inhibition of [3H]-raclopride binding to Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080048((4-Fluoro-benzyl)-((R)-5-methoxy-1,2,3,4-tetrahydr...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080051(Benzyl-((R)-5-methoxy-1,2,3,4-tetrahydro-naphthale...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080055(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  82.3nMAssay Description:Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054336(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  108nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080055(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080052(CHEMBL303502 | Furan-2-ylmethyl-((R)-5-methoxy-1,2...)
Affinity DataKi:  118nMAssay Description:Displacement of [3H]-quinpirole from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080052(CHEMBL303502 | Furan-2-ylmethyl-((R)-5-methoxy-1,2...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054334((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-ylami...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50080049(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  152nMAssay Description:Displacement of [3H]-raclopride from human dopamine D2A receptors expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054341(Butyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054336(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  167nMAssay Description:Displacement of [3H]-quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054337(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  179nMAssay Description:Displacement of [3H]-quinpirole from Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054337(Benzyl-((R)-5-fluoro-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataKi:  179nMAssay Description:Inhibition of [3H]-quinpirole binding to human dopamine D2A receptor expressed in LtK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50054335(((R)-5-Fluoro-1,2,3,4-tetrahydro-naphthalen-2-yl)-...)
Affinity DataKi:  199nMAssay Description:Displacement of [3H]-raclopride from Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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