Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nM ΔG°: -54.0kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 0.450nM ΔG°: -53.3kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nM ΔG°: -51.8kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 0.910nM ΔG°: -51.6kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 1.5nM ΔG°: -50.4kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 9.30nM ΔG°: -45.8kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12.8nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 16.4nM ΔG°: -44.4kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 17.6nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 21.4nM ΔG°: -43.8kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 39.3nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 41.7nM ΔG°: -42.1kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 47.2nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 78.8nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of [3H]-APS-314d binding to prostacyclin receptors (IP) of human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Inhibition of [3H]-SQ-29,548 binding to thromboxane A2 receptors (TP) of human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair