BindingDB PrimarySearch_ki

Found 369 with Last Name = 'ratia' and Initial = 'k'

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539801(CHEMBL4648912 | US11840533, Compound 70)

IC50: 1.70nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 2 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539801(CHEMBL4648912 | US11840533, Compound 70)

IC50: 5.90nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539804(CHEMBL4640025 | US11840533, Compound 71)

IC50: 8.30nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539802(CHEMBL4647718)

IC50: 9.40nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539800(CHEMBL4632358)

IC50: 13nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 2 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539803(CHEMBL4633289)

IC50: 13nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539800(CHEMBL4632358)

IC50: 13nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50031720((Dofetilide) N-[4-(2-{[2-(4-Methanesulfonylamino-p...)

IC50: 15nMAssay Description:Inhibition of human ERG stably expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539804(CHEMBL4640025 | US11840533, Compound 71)

IC50: 22nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 2 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539805(CHEMBL4644032 | US11840533, Compound 72)

IC50: 40nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539786(CHEMBL4640133)

IC50: 48nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539792(CHEMBL4646027)

IC50: 54nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM50537622(CHEMBL4634168)

IC50: 55nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539803(CHEMBL4633289)

IC50: 63nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 2 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM561983(BDBM50369389 | US11396496, Compound A1)

IC50: 63nMAssay Description:Concentration required to inhibit the phosphorylation of a 14-residue fragment of phospholipase C gamma 1 by Epidermal growth factor receptor from A4...More data for this Ligand-Target Pair

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Kelch-like ECH-associated protein 1(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50519234(CHEMBL4440989)

IC50: 63nMAssay Description:Inhibition of FITC-9mer Nrf2 peptide binding to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) b...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM561992(BDBM50537618 | US11396496, Compound B0)

IC50: 73nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair

PDB KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539799(CHEMBL4638621)

IC50: 83nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539791(CHEMBL4637378)

IC50: 89nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539785(CHEMBL4646327)

IC50: 96nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Replicase polyprotein 1ab(2019-nCoV)
University of Illinois At Chicago

PNG

BDBM496864(SARS-CoV-2 PLpro Inhibitor, 94)

IC50: 113nMAssay Description:The PLpro primary assay, which measures protease activity with the short peptide substrate Z-RLRGG-AMC (Bachem), was performed in black flat-bottom 3...More data for this Ligand-Target Pair

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3D Structure (crystal)

Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM50537620(CHEMBL4641049)

IC50: 120nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair

PDB KEGG
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Kelch-like ECH-associated protein 1(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50538489(CHEMBL4632368)

IC50: 126nMAssay Description:Inhibition of FITC-9mer Nrf2 peptide binding to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) b...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 126nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 2 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM50537619(CHEMBL4648321)

IC50: 130nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Details Article PubMed

Kelch-like ECH-associated protein 1(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50190617(CHEMBL3827626)

IC50: 140nMAssay Description:Inhibition of FITC-9mer Nrf2 peptide binding to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) b...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Kelch-like ECH-associated protein 1(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50538490(CHEMBL4632722)

IC50: 151nMAssay Description:Inhibition of FITC-9mer Nrf2 peptide binding to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) b...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539793(CHEMBL4644443)

IC50: 158nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539798(CHEMBL4649774)

IC50: 161nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Replicase polyprotein 1ab(2019-nCoV)
University of Illinois At Chicago

PNG

BDBM496858(SARS-CoV-2 PLpro Inhibitor, 88)

IC50: 170nMAssay Description:The PLpro primary assay, which measures protease activity with the short peptide substrate Z-RLRGG-AMC (Bachem), was performed in black flat-bottom 3...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539796(CHEMBL4632925)

IC50: 174nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539794(CHEMBL4647786)

IC50: 175nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539797(CHEMBL4635722)

IC50: 180nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Kelch-like ECH-associated protein 1(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM561995(BDBM50538487 | US11396496, Compound C3)

IC50: 189nMAssay Description:Inhibition of FITC-9mer Nrf2 peptide binding to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) b...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)

IC50: 199nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM50537623(CHEMBL4640762)

IC50: 210nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Details Article PubMed

Replicase polyprotein 1ab(2019-nCoV)
University of Illinois At Chicago

PNG

BDBM496862(SARS-CoV-2 PLpro Inhibitor, 92)

IC50: 210nMAssay Description:The PLpro primary assay, which measures protease activity with the short peptide substrate Z-RLRGG-AMC (Bachem), was performed in black flat-bottom 3...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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3D Structure (crystal)

Bromodomain-containing protein 4(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50539805(CHEMBL4644032 | US11840533, Compound 72)

IC50: 220nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 2 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM561988(BDBM50537615 | US11396496, Compound A6)

IC50: 230nMAssay Description:Concentration required to inhibit the phosphorylation of a 14-residue fragment of phospholipase C gamma 1 by Epidermal growth factor receptor from A4...More data for this Ligand-Target Pair

PDB KEGG
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Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM50537613(CHEMBL4637137)

IC50: 240nMAssay Description:Concentration required to inhibit the phosphorylation of a 14-residue fragment of phospholipase C gamma 1 by Epidermal growth factor receptor from A4...More data for this Ligand-Target Pair

PDB KEGG
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Kelch-like ECH-associated protein 1(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL

PNG

BDBM50538491(CHEMBL4647946)

IC50: 241nMAssay Description:Inhibition of FITC-9mer Nrf2 peptide binding to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) b...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Replicase polyprotein 1ab(2019-nCoV)
University of Illinois At Chicago

PNG

BDBM496865(SARS-CoV-2 PLpro Inhibitor, 95)

IC50: 250nMAssay Description:The PLpro primary assay, which measures protease activity with the short peptide substrate Z-RLRGG-AMC (Bachem), was performed in black flat-bottom 3...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM50537612(CHEMBL4640093)

IC50: 280nMAssay Description:Concentration required to inhibit the phosphorylation of a 14-residue fragment of phospholipase C gamma 1 by Epidermal growth factor receptor from A4...More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Replicase polyprotein 1ab(2019-nCoV)
University of Illinois At Chicago

PNG

BDBM496856(SARS-CoV-2 PLpro Inhibitor, 86)

IC50: 330nMAssay Description:The PLpro primary assay, which measures protease activity with the short peptide substrate Z-RLRGG-AMC (Bachem), was performed in black flat-bottom 3...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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3D Structure (crystal)

Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM561986(BDBM50537611 | US11396496, Compound A4)

IC50: 350nMAssay Description:Concentration required to inhibit the phosphorylation of a 14-residue fragment of phospholipase C gamma 1 by Epidermal growth factor receptor from A4...More data for this Ligand-Target Pair

PDB KEGG
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Replicase polyprotein 1ab(2019-nCoV)
University of Illinois At Chicago

PNG

BDBM496859(SARS-CoV-2 PLpro Inhibitor, 89)

IC50: 370nMAssay Description:The PLpro primary assay, which measures protease activity with the short peptide substrate Z-RLRGG-AMC (Bachem), was performed in black flat-bottom 3...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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3D Structure (crystal)

Replicase polyprotein 1ab(2019-nCoV)
University of Illinois At Chicago

PNG

BDBM496842(SARS-CoV-2 PLpro Inhibitor, 72)

IC50: 390nMAssay Description:The PLpro primary assay, which measures protease activity with the short peptide substrate Z-RLRGG-AMC (Bachem), was performed in black flat-bottom 3...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Replicase polyprotein 1ab(2019-nCoV)
University of Illinois At Chicago

PNG

BDBM496861(SARS-CoV-2 PLpro Inhibitor, 91)

IC50: 410nMAssay Description:The PLpro primary assay, which measures protease activity with the short peptide substrate Z-RLRGG-AMC (Bachem), was performed in black flat-bottom 3...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM50537621(CHEMBL4645359)

IC50: 420nMAssay Description:Inhibitory potency against isolated epidermal growth factor receptor (EGFR) from human A431 carcinoma cellsMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Details Article PubMed

Nuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL

PNG

BDBM561987(BDBM50537610 | US11396496, Compound A5)

IC50: 430nMAssay Description:Concentration required to inhibit the phosphorylation of a 14-residue fragment of phospholipase C gamma 1 by Epidermal growth factor receptor from A4...More data for this Ligand-Target Pair

PDB KEGG
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Displayed 1 to 50 (of 369 total ) | Next | Last >>

Filter my 369 hits

Targets 36▿
- Replicase polyprotein 1ab 193
- Cystathionine gamma-lyase 47
- Bromodomain-containing protein 4 32
- Replicase polyprotein 1ab [1541-1855] 24
- Kelch-like ECH-associated protein 1 15
- Nuclear factor erythroid 2-related factor 2 15
- Bromodomain-containing protein 3 3
- Angiotensin-converting enzyme 2 3
- Bromodomain-containing protein 2 3
- Bromodomain testis-specific protein 3
- Protein polybromo-1 2
- Replicase polyprotein 1a 2
- Bromodomain-containing protein 8 2
- Potassium voltage-gated channel subfamily H member 2 2
- Transcription intermediary factor 1-alpha 2
- ATPase family AAA domain-containing protein 2B 1
- Transcription initiation factor TFIID subunit 1-like 1
- Bromodomain and WD repeat-containing protein 1 1
- Bromodomain adjacent to zinc finger domain protein 2A 1
- Peregrin 1
- Bromodomain adjacent to zinc finger domain protein 2B 1
- Nucleosome-remodeling factor subunit BPTF 1
- Bromodomain and PHD finger-containing protein 3 1
- Bromodomain-containing protein 1 1
- E3 ubiquitin-protein ligase TRIM33 1
- Histone acetyltransferase p300 1
- Transcription activator BRG1 1
- ATPase family AAA domain-containing protein 2 1
- Chromatin remodeling regulator CECR2 1
- CREB-binding protein 1
- Histone acetyltransferase KAT2B 1
- Histone acetyltransferase KAT2A 1
- Transcription initiation factor TFIID subunit 1 1
- Bromodomain-containing protein 7 1
- Probable global transcription activator SNF2L2 1
- Bromodomain-containing protein 9 1
- ...
Publications 8▿
- J Med Chem (2021) 189
- J Med Chem 63: 7186-7210 (2020) 70
- ACS Med Chem Lett 8: 1241-1245 (2017) 47
- J Med Chem 52: 5228-40 (2009) 24
- J Med Chem 63: 6547-6560 (2020) 15
- ACS Med Chem Lett 11: 521-527 (2020) 15
- Bioorg Med Chem Lett 17: 5876-80 (2007) 7
- J Med Chem 48: 6767-71 (2005) 2
Institutions 4▿
- University of Illinois At Chicago 189
- University Of Illinois At Chicago 132
- Purdue University 33
- TBA 15
Affinity: 1 to 1.0E+6 nM▿
- IC50 227
- Kd 130
- EC50 3
- Affinity ≤ nM
Xtal structures: 9
Docked structures: 13
Catalog Cmpds: 21