Affinity DataIC50: 0.00800nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human dopamine D2 receptor expressed in CHO cells co-expressing A2A receptor assessed as reduction in sumanirole-induced respo...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
Affinity DataIC50: 255nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Antagonist activity at human dopamine D2 receptor expressed in CHO cells co-expressing A2A receptor assessed as reduction in sumanirole-induced respo...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9.09E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.13E+4nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.36E+4nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 700nMAssay Description:Displacement of [3H]SCH 23390 from dopamine D1 receptor in lamb striatum membrane after 1 hrMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Displacement of [3H]YM 09151-2 from dopamine D2 receptor in lamb striatum membrane after 2 hrsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 100nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor in lamb striatum membrane after 1 hrMore data for this Ligand-Target Pair
Affinity DataKd: 93nMAssay Description:Displacement of [3H]-raclopride from human dopamine D3 receptor low binding affinity site expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 23nMAssay Description:Displacement of [3H]-raclopride from human dopamine D3 receptor high binding affinity site expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 7.00E+3nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as low affinity constant aft...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 200nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 500nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 900nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 600nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 4.70E+3nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 280nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 240nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 6.30E+3nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Biomaterials And Nanomedicine (Ciber-Bbn)
Curated by ChEMBL
Affinity DataKd: 5.00E+3nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 3.30E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 4.00E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 1.30E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 1.90E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 3.40E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 1.20E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 1.50E+4nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 2.90E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 3.80E+4nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Institut D'Investigacions BiomèDiques August Pi I
Curated by ChEMBL
Affinity DataKd: 2.70E+4nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair