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Found 91 with Last Name = 'royo' and Initial = 'm'
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Landsteiner Genmed

US Patent
LigandPNGBDBM535882(US11242312, Example 3)
Affinity DataIC50:  0.00800nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Landsteiner Genmed

US Patent
LigandPNGBDBM535880(US11242312, Example 1)
Affinity DataIC50:  0.0300nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Landsteiner Genmed

US Patent
LigandPNGBDBM535881(US11242312, Example 2)
Affinity DataIC50:  2.20nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Landsteiner Genmed

US Patent
LigandPNGBDBM535883(US11242312, Example 4)
Affinity DataIC50:  7.10nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50503395(CHEMBL4515776)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at human dopamine D2 receptor expressed in CHO cells co-expressing A2A receptor assessed as reduction in sumanirole-induced respo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Landsteiner Genmed

US Patent
LigandPNGBDBM535885(N-((S)-1-(((S)-4-(cyclopropylamino)-3,4-dioxo-1-ph...)
Affinity DataIC50:  110nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Landsteiner Genmed

US Patent
LigandPNGBDBM535884(N-((S)-1-(((S)-4-(cyclopropylamino)-3,4-dioxo-1-ph...)
Affinity DataIC50:  255nMAssay Description:Activity of Calpain 1 was measured by using Calpain-Glo Protease kit from Promega. Assays were run in 384-well black plates with clear bottom. 5 _...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50503396(CHEMBL4542935)
Affinity DataIC50:  280nMAssay Description:Antagonist activity at human dopamine D2 receptor expressed in CHO cells co-expressing A2A receptor assessed as reduction in sumanirole-induced respo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162761(CHEMBL180302 | [4-Guanidino-1-((S)-4-{(S)-5-[4-((S...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162770(CHEMBL180281 | N-[4-Guanidino-1-((S)-4-{(S)-5-[4-(...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162764(CHEMBL359680 | [1-((S)-4-{(S)-5-[4-((S)-(S)-2-Benz...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162760(4-Guanidino-N-[(S)-4-((S)-5-{4-[2-(2-imino-imidazo...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162758(4-Guanidino-N-(4-{(S)-5-[4-((S)-4-guanidino-butyry...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162762(CHEMBL181327 | [(S)-4-Guanidino-1-((S)-4-{(S)-5-[4...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162763(CHEMBL181685 | N-((S)-4-{5-[4-(3-Guanidino-propion...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162759(CHEMBL178315 | [1-(4-{(S)-5-[((S)-3-Carbamimidoyl-...)
Affinity DataIC50:  9.09E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162765((S)-N-[4-Guanidino-1-((S)-4-{(S)-5-[4-(5-guanidino...)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162769(CHEMBL361835 | N-[(S)-1-(4-{(S)-5-[((S)-3-Carbamim...)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162766(CHEMBL181467 | N-((S)-4-{(S)-5-[(3-Carbamimidoyl-p...)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162771(CHEMBL181234 | N-(3-Carbamimidoyl-phenyl)-2-{(2S,5...)
Affinity DataIC50:  1.99E+4nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162768(CHEMBL178777 | N-((S)-4-{(S)-5-[(3-Carbamimidoyl-p...)
Affinity DataIC50:  2.13E+4nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162767(CHEMBL180850 | N-((S)-4-{(S)-5-[(3-Carbamimidoyl-p...)
Affinity DataIC50:  2.36E+4nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50214408((6aR,9S)-N-((S)-1-((S)-1-((S)-2-carbamoylpyrrolidi...)
Affinity DataKd:  700nMAssay Description:Displacement of [3H]SCH 23390 from dopamine D1 receptor in lamb striatum membrane after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50214409((6aR,9R)-N-((S)-1-((S)-1-((S)-2-carbamoylindolin-1...)
Affinity DataKd:  2.00E+3nMAssay Description:Displacement of [3H]YM 09151-2 from dopamine D2 receptor in lamb striatum membrane after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50214409((6aR,9R)-N-((S)-1-((S)-1-((S)-2-carbamoylindolin-1...)
Affinity DataKd:  100nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor in lamb striatum membrane after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50336701((6aR,9R)-N-((2S)-1-((2S)-1-(3-(6-((S)-6-amino-6-ox...)
Affinity DataKd:  93nMAssay Description:Displacement of [3H]-raclopride from human dopamine D3 receptor low binding affinity site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50336701((6aR,9R)-N-((2S)-1-((2S)-1-(3-(6-((S)-6-amino-6-ox...)
Affinity DataKd:  23nMAssay Description:Displacement of [3H]-raclopride from human dopamine D3 receptor high binding affinity site expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083509(CHEMBL3423402)
Affinity DataKd:  7.00E+3nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as low affinity constant aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083510(CHEMBL3423411)
Affinity DataKd:  400nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083540(CHEMBL3423410)
Affinity DataKd:  200nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083544(CHEMBL3423409)
Affinity DataKd:  2.00E+3nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083546(CHEMBL3423408)
Affinity DataKd:  500nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083550(CHEMBL3423407)
Affinity DataKd:  190nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083551(CHEMBL3423406)
Affinity DataKd:  900nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083554(CHEMBL3423405)
Affinity DataKd:  600nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083555(CHEMBL3423404)
Affinity DataKd:  4.70E+3nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083558(CHEMBL3423403)
Affinity DataKd:  280nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083509(CHEMBL3423402)
Affinity DataKd:  240nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083559(CHEMBL3423401)
Affinity DataKd:  6.30E+3nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Biomaterials And Nanomedicine (Ciber-Bbn)

Curated by ChEMBL
LigandPNGBDBM50083560(CHEMBL3423400)
Affinity DataKd:  5.00E+3nMAssay Description:Displacement of [3H]-YM09151-2 from dopamine D2 receptor (unknown origin) expressed in sheep striatum membranes assessed as high affinity constant af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50083544(CHEMBL3423409)
Affinity DataKd:  3.30E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50083546(CHEMBL3423408)
Affinity DataKd:  4.00E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50083550(CHEMBL3423407)
Affinity DataKd:  1.30E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50083551(CHEMBL3423406)
Affinity DataKd:  1.90E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50083554(CHEMBL3423405)
Affinity DataKd:  3.40E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50083555(CHEMBL3423404)
Affinity DataKd:  1.20E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50083558(CHEMBL3423403)
Affinity DataKd:  1.50E+4nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50083509(CHEMBL3423402)
Affinity DataKd:  2.90E+3nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50083559(CHEMBL3423401)
Affinity DataKd:  3.80E+4nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Institut D'Investigacions BiomèDiques August Pi I

Curated by ChEMBL
LigandPNGBDBM50083560(CHEMBL3423400)
Affinity DataKd:  2.70E+4nMAssay Description:Displacement of [3H]-SCH23390 from dopamine D1 receptor (unknown origin) expressed in sheep striatum membranes after 1.5 hrs by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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