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Found 85 with Last Name = 'saghir' and Initial = 'n'
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Piramed Pharma

LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataKi:  580nM ΔG°:  -35.6kJ/molepH: 7.5 T: 2°CAssay Description:Mammalian target of rapamycin (mTOR) was assayed by monitoring phosphorylation of GFP-4EBP using a homogeneous time-resolved fluorescence resonance e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25021(3-{6-[(dimethylamino)methyl]-4-(morpholin-4-yl)thi...)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  3nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25022(3-(6-{[(2-methoxyethyl)(methyl)amino]methyl}-4-(mo...)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25019(3-[6-methyl-4-(morpholin-4-yl)thieno[3,2-d]pyrimid...)
Affinity DataIC50:  6nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25024(3-(6-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-4-...)
Affinity DataIC50:  7nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25018(3-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phe...)
Affinity DataIC50:  8nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25023(3-{6-[(4-methylpiperazin-1-yl)methyl]-4-(morpholin...)
Affinity DataIC50:  10nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25020(3-[7-methyl-4-(morpholin-4-yl)thieno[3,2-d]pyrimid...)
Affinity DataIC50:  21nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  33nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
LigandPNGBDBM25027(4-[2-(1H-indazol-4-yl)-6-[(4-methylpiperazin-1-yl)...)
Affinity DataIC50:  44nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333813(3-(4-Morpholino-6-(pyridin-2-yl)pyrimidin-2-yl)phe...)
Affinity DataIC50:  44nMAssay Description:Inhibition of human recombinant PI3K p110gamma after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333813(3-(4-Morpholino-6-(pyridin-2-yl)pyrimidin-2-yl)phe...)
Affinity DataIC50:  62nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  75nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333813(3-(4-Morpholino-6-(pyridin-2-yl)pyrimidin-2-yl)phe...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant PI3K p110beta after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25025(4-[2-(1H-indazol-4-yl)thieno[3,2-d]pyrimidin-4-yl]...)
Affinity DataIC50:  102nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333821(3-(2-Morpholino-6-(pyridin-2-ylmethoxy)pyrimidin-4...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333815(3-(4-Morpholino-6-(pyridin-4-yl)pyrimidin-2-yl)phe...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333819(3-(2-Morpholino-6-(2-(pyridin-4-yl)ethylamino)pyri...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333815(3-(4-Morpholino-6-(pyridin-4-yl)pyrimidin-2-yl)phe...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human recombinant PI3K p110gamma after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333820(3-(6-Morpholino-2-(2-(pyridin-2-yl)ethylamino)pyri...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333815(3-(4-Morpholino-6-(pyridin-4-yl)pyrimidin-2-yl)phe...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant PI3K p110beta after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333828(3-(4-(3,4-Dichlorophenyl)-6-morpholinopyrimidin-2-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333834(3-(6-Morpholino-2-(2-(pyridin-4-yl)ethylamino)pyri...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333817(3-(2-Morpholino-6-(2-(pyridin-2-yl)ethylamino)pyri...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333833(3-(6-Morpholino-2-(2-(pyridin-3-yl)ethylamino)pyri...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333814(3-(4-Morpholino-6-(pyridin-3-yl)pyrimidin-2-yl)phe...)
Affinity DataIC50:  260nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333818(3-(2-Morpholino-6-(2-(pyridin-3-yl)ethylamino)pyri...)
Affinity DataIC50:  260nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333814(3-(4-Morpholino-6-(pyridin-3-yl)pyrimidin-2-yl)phe...)
Affinity DataIC50:  340nMAssay Description:Inhibition of human recombinant PI3K p110gamma after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333821(3-(2-Morpholino-6-(pyridin-2-ylmethoxy)pyrimidin-4...)
Affinity DataIC50:  370nMAssay Description:Inhibition of human recombinant PI3K p110beta after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333820(3-(6-Morpholino-2-(2-(pyridin-2-yl)ethylamino)pyri...)
Affinity DataIC50:  380nMAssay Description:Inhibition of human recombinant PI3K p110gamma after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333814(3-(4-Morpholino-6-(pyridin-3-yl)pyrimidin-2-yl)phe...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human recombinant PI3K p110beta after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333809(4-(1H-indazol-4-yl)-6-morpholino-N-(2-(pyridin-4-y...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333800(4-(4-(1H-indazol-4-yl)-6-(pyridin-2-ylmethoxy)pyri...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333796(6-(1H-indazol-4-yl)-2-morpholino-N-(2-(pyridin-3-y...)
Affinity DataIC50:  660nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataIC50:  670nMpH: 7.5 T: 2°CAssay Description:Test compounds were added to reaction buffer containing yttrium silicate (Ysi) polylysine SPA beads (Amersham), and the enzyme was added to the assay...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333827(3-(4-(4-Chlorophenyl)-6-morpholinopyrimidin-2-yl)p...)
Affinity DataIC50:  690nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50331594(3-(2-morpholino-6-(pyridin-3-ylmethylamino)pyrimid...)
Affinity DataIC50:  720nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333821(3-(2-Morpholino-6-(pyridin-2-ylmethoxy)pyrimidin-4...)
Affinity DataIC50:  730nMAssay Description:Inhibition of human recombinant PI3K p110gamma after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333819(3-(2-Morpholino-6-(2-(pyridin-4-yl)ethylamino)pyri...)
Affinity DataIC50:  740nMAssay Description:Inhibition of human recombinant PI3K p110gamma after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333797(6-(1H-indazol-4-yl)-2-morpholino-N-(2-(pyridin-4-y...)
Affinity DataIC50:  770nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333808(4-(1H-indazol-4-yl)-6-morpholino-N-(2-(pyridin-3-y...)
Affinity DataIC50:  820nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333817(3-(2-Morpholino-6-(2-(pyridin-2-yl)ethylamino)pyri...)
Affinity DataIC50:  830nMAssay Description:Inhibition of human recombinant PI3K p110gamma after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333832(3-(6-Morpholino-2-(pyridin-4-ylmethylamino)pyrimid...)
Affinity DataIC50:  860nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333835(3-(6-Morpholino-2-(pyridin-2-ylmethoxy)pyrimidin-4...)
Affinity DataIC50:  860nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333831(3-(6-Morpholino-2-(pyridin-3-ylmethylamino)pyrimid...)
Affinity DataIC50:  880nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50333816(3-(2-Morpholino-6-(pyridin-2-ylmethylamino)pyrimid...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human recombinant PI3K p110alpha after 1 hr by radiometric scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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