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Found 16 with Last Name = 'sartorelli' and Initial = 'ac'
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50397045(CHEMBL485756)
Affinity DataIC50:  9nMAssay Description:Inhibition of AGT in human HL60 cells assessed as AGT levels using [3H]AGT after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50397044(CHEMBL2171205)
Affinity DataIC50:  25nMAssay Description:Inhibition of AGT in human HL60 cells assessed as AGT levels using [3H]AGT after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM5491(6-(benzyloxy)-9H-purin-2-amine | CHEMBL407874 | O6...)
Affinity DataIC50:  39nMAssay Description:Inhibition of AGT in human HL60 cells assessed as AGT levels using [3H]AGT after 2 hrsMore data for this Ligand-Target Pair
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50397043(CHEMBL2171202)
Affinity DataIC50:  86nMAssay Description:Inhibition of AGT in human HL60 cells assessed as AGT levels using [3H]AGT after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051772((Z)-N'-(5-amino-6-formylpyridin-2-yl)carbamohydraz...)
Affinity DataIC50:  820nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051768((1Z,N'E)-N'-((3-(methylamino)pyridin-2-yl)methylen...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051776((1Z,N'E)-N'-((5-(ethylamino)pyridin-2-yl)methylene...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051769((1Z,N'E)-N'-((5-(methylamino)pyridin-2-yl)methylen...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051767((1Z,N'E)-N'-((5-(propylamino)pyridin-2-yl)methylen...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051775((1Z,N'E)-N'-((5-(allylamino)pyridin-2-yl)methylene...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051774((1Z,N'E)-N'-((3-(allylamino)pyridin-2-yl)methylene...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051766((1Z,N'E)-N'-((5-(butylamino)pyridin-2-yl)methylene...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051777((1Z,N'E)-N'-((5-(aminomethyl)pyridin-2-yl)methylen...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051773((Z)-N'-(3-amino-6-formylpyridin-2-yl)carbamohydraz...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051771((1Z,N'E)-N'-((3,5-diaminopyridin-2-yl)methylene)ca...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051770((1Z,N'E)-N'-((5-amino-4-(morpholinomethyl)pyridin-...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed