Affinity DataKi: 127nMAssay Description:Binding affinity to Bcl-xL after 2 hrs by fluorescein-labeled Bak-BH3 peptide competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity to Bcl-xL after 2 hrs by fluorescein-labeled Bak-BH3 peptide competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Binding affinity to Bcl-xL after 2 hrs by fluorescein-labeled Bak-BH3 peptide competition binding assayMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataIC50: 6.69E+3nMAssay Description:Inhibition of human FLT3 using gamma-33P-ATP as substrate by scintillation countingMore data for this Ligand-Target Pair
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Louisana
Curated by ChEMBL
University Of Louisana
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 activation in human T47D cells by cell based reporter gene assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human KIT using gamma-33P-ATP as substrate by scintillation countingMore data for this Ligand-Target Pair
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Louisana
Curated by ChEMBL
University Of Louisana
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of 1,10-phenanthroline-induced HIF1 activation in human T47D cells by cell based reporter gene assayMore data for this Ligand-Target Pair
TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
University Of Louisana
Curated by ChEMBL
University Of Louisana
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of hypoxia-induced HIF1 activation in human T47D cells by cell based reporter gene assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 7.80E+3nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 260nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 240nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 0.620nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 31nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 2.70nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 200nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 2nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 14nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 170nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 5.40nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 3.70nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 2.80nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 7.5nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 17nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 0.680nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 0.370nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 5.10nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 460nMAssay Description:Binding affinity to human FLT3 incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 2.20E+3nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 19nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 27.2nMAssay Description:Binding affinity to human unphosphorylated c-METMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 8nMAssay Description:Binding affinity to PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Binding affinity to KIT (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 14nMAssay Description:Binding affinity to PDGFRalpha (unknown origin)More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of The Pacific
Curated by ChEMBL
University Of The Pacific
Curated by ChEMBL
Affinity DataKd: 0.400nMAssay Description:Binding affinity to KIT D816V mutant (unknown origin)More data for this Ligand-Target Pair