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Found 94 with Last Name = 'sherbukhin' and Initial = 'v'
TargetProtein M2-1(Human respiratory syncytial virus A (strain A2))
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50256886(CHEMBL4091425)
Affinity DataIC50:  2nMAssay Description:Inhibition of Respiratory syncytial virus A2 M2-1 by luciferase reporter-based RSV minigenome assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoprotein(Human respiratory syncytial virus A (strain A2))
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50256886(CHEMBL4091425)
Affinity DataIC50:  2nMAssay Description:Inhibition of Respiratory syncytial virus A2 protein P by luciferase reporter-based RSV minigenome assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Sygnature Discovery

Curated by ChEMBL
LigandPNGBDBM50256886(CHEMBL4091425)
Affinity DataIC50:  2nMAssay Description:Inhibition of Respiratory syncytial virus A2 protein N by luciferase reporter-based RSV minigenome assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412708(AC-264613 | CHEMBL494502)
Affinity DataEC50:  31.6nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412708(AC-264613 | CHEMBL494502)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM85517(CAS_171436-38-7 | SL-NH2 | SLIGRL-NH2)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412709(CHEMBL461639)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412710(CHEMBL459724)
Affinity DataEC50:  6.31E+3nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412711(CHEMBL459723)
Affinity DataEC50:  25.1nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412712(CHEMBL459509)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412713(CHEMBL493704)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412714(CHEMBL493494)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412715(CHEMBL494503)
Affinity DataEC50:  7.94E+3nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412708(AC-264613 | CHEMBL494502)
Affinity DataEC50:  31.6nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412716(AC-98170 | CHEMBL494303)
Affinity DataEC50:  6.31E+3nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412717(AC-55541 | CHEMBL493076)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50412718(CHEMBL509819)
Affinity DataEC50:  25.1nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413260(CHEMBL198794)
Affinity DataEC50:  16nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413267(CHEMBL371684)
Affinity DataEC50:  25nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)
Affinity DataEC50:  20nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413260(CHEMBL198794)
Affinity DataEC50:  316nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413272(AC-261066 | CHEMBL198997)
Affinity DataEC50:  10nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50:  25nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475526(CHEMBL198467)
Affinity DataEC50:  50nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)
Affinity DataEC50:  50nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50:  6.30nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475527(CHEMBL197292)
Affinity DataEC50:  16nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413261(AC-55649 | CHEMBL425027)
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413261(AC-55649 | CHEMBL425027)
Affinity DataEC50:  126nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475526(CHEMBL198467)
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475527(CHEMBL197292)
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475528(CHEMBL365798)
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413267(CHEMBL371684)
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Acadia Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50475528(CHEMBL365798)
Affinity DataEC50:  63nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475708(CHEMBL425592)
Affinity DataEC50:  117nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50414759(CHEMBL574304)
Affinity DataEC50:  871nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475709(CHEMBL377938)
Affinity DataEC50:  6.46E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475710(CHEMBL205681)
Affinity DataEC50:  275nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50164424(3-(4-Chloro-phenyl)-3-(2-dimethylamino-ethyl)-isoc...)
Affinity DataEC50:  1.12E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475711(CHEMBL203337)
Affinity DataEC50:  1.41E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475712(CHEMBL382477)
Affinity DataEC50:  2.00E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475713(CHEMBL206661)
Affinity DataEC50:  2.09E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475714(CHEMBL208536)
Affinity DataEC50:  1.12E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475715(CHEMBL203051)
Affinity DataEC50:  251nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475716(CHEMBL205157)
Affinity DataEC50:  1.02E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475717(CHEMBL208436)
Affinity DataEC50:  1.07E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475718(CHEMBL208886)
Affinity DataEC50:  2.19E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475719(CHEMBL205735)
Affinity DataEC50:  2.00E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475720(CHEMBL206719)
Affinity DataEC50:  2.29E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475721(CHEMBL206551)
Affinity DataEC50:  288nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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