TargetProtein M2-1(Human respiratory syncytial virus A (strain A2))
Sygnature Discovery
Curated by ChEMBL
Sygnature Discovery
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Respiratory syncytial virus A2 M2-1 by luciferase reporter-based RSV minigenome assayMore data for this Ligand-Target Pair
TargetPhosphoprotein(Human respiratory syncytial virus A (strain A2))
Sygnature Discovery
Curated by ChEMBL
Sygnature Discovery
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Respiratory syncytial virus A2 protein P by luciferase reporter-based RSV minigenome assayMore data for this Ligand-Target Pair
TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Sygnature Discovery
Curated by ChEMBL
Sygnature Discovery
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Respiratory syncytial virus A2 protein N by luciferase reporter-based RSV minigenome assayMore data for this Ligand-Target Pair
Affinity DataEC50: 31.6nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 50.1nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.31E+3nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 25.1nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.51E+3nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.94E+3nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 31.6nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.31E+3nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 25.1nMAssay Description:Agonist activity at human PAR2 expressed in HEK293T cells assessed as effect on intracellular calcium mobilization by R-SAT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Transcriptional activity against RARbeta1More data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Transcriptional activity against RARbeta2More data for this Ligand-Target Pair
Affinity DataEC50: 117nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 871nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 6.46E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 275nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.12E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.41E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.09E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.12E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.02E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.07E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.19E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.29E+3nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 288nMAssay Description:Activity against human urotensin-2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair