Affinity DataKi: 0.282nMAssay Description:Adenosine A1 receptor binding using [3H]DPCPX in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Adenosine A1 receptor binding using [3H]DPCOX in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Adenosine A1 receptor binding using [3H]DPCPX in human cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Adenosine A1 receptor using [3H]DPCOX in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 151nMAssay Description:Adenosine A2 receptor binding using [3H]CGS-21680 in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Adenosine A2 receptor binding using [3H]CGS-21680 in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+3nMAssay Description:Adenosine A2 receptor binding using [3H]CGS-21680 in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Inhibition of adenosine induced negative inotropic activity against guinea-pig atria (Adenosine A1 receptor)More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of adenosine induced negative inotropic activity against guinea-pig atria (Adenosine A1 receptor)More data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of [3H]-CHA binding against Adenosine A1 receptors of rat cortical membranes; Not testedMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of [3H]-CHA binding against Adenosine A1 receptors of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:Inhibition of adenosine induced negative inotropic activity against guinea-pig atria (Adenosine A1 receptor) at 10 nMMore data for this Ligand-Target Pair
Affinity DataIC50: 656nMAssay Description:Compound was evaluated for inhibition of adenosine induced relaxation against guinea-pig aorta (Adenosine A2 receptor).More data for this Ligand-Target Pair
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of [3H]NECA specific binding against Adenosine A2 receptors of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of adenosine induced negative inotropic activity against guinea-pig atria (Adenosine A1 receptor)More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Compound was evaluated for inhibition of adenosine induced relaxation against guinea-pig aorta (Adenosine A2 receptor).More data for this Ligand-Target Pair
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of [3H]-CHA binding against Adenosine A1 receptors of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of [3H]NECA specific binding against Adenosine A2 receptors of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Compound was evaluated for inhibition of adenosine induced relaxation against guinea-pig aorta (Adenosine A2 receptor).More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of [3H]NECA specific binding against Adenosine A2 receptors of rat striatal membranesMore data for this Ligand-Target Pair