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Found 242 with Last Name = 'shonberg' and Initial = 'j'
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50395587(CHEMBL2165126 | UNC10000006 | US9156822, 2)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50395587(CHEMBL2165126 | UNC10000006 | US9156822, 2)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239412(CHEMBL4072780)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239410(CHEMBL4100183)
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239403(CHEMBL4102628)
Affinity DataKi:  0.810nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239410(CHEMBL4100183)
Affinity DataKi:  0.860nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239412(CHEMBL4072780)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239408(CHEMBL4083239)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239408(CHEMBL4083239)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239412(CHEMBL4072780)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239419(CHEMBL4064186)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  1.60nMAssay Description:Antagonist activity at human adenosine A2A receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239416(CHEMBL4070604)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239403(CHEMBL4102628)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239405(CHEMBL4064742)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239405(CHEMBL4064742)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239403(CHEMBL4102628)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50395587(CHEMBL2165126 | UNC10000006 | US9156822, 2)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239418(CHEMBL4099666)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239405(CHEMBL4064742)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239410(CHEMBL4100183)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50395587(CHEMBL2165126 | UNC10000006 | US9156822, 2)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2AR expressed in HEK293T cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239413(CHEMBL4091933)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239413(CHEMBL4091933)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239411(CHEMBL4068702)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239406(CHEMBL4091507)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239419(CHEMBL4064186)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2AR expressed in HEK293T cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239409(CHEMBL4092441)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239409(CHEMBL4092441)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239410(CHEMBL4100183)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239418(CHEMBL4099666)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  5.80nMAssay Description:Antagonist activity at human adenosine A2A receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50176058(2-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-...)
Affinity DataKi:  6.60nMAssay Description:Antagonist activity at human adenosine A2A receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239418(CHEMBL4099666)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-NPA from dopamine D2L receptor (unknown origin) expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  8.30nMAssay Description:Antagonist activity at human adenosine A1 receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239412(CHEMBL4072780)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]spiperone from human D4R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239409(CHEMBL4092441)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]spiperone from human D2LR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239414(CHEMBL4073330)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50443100(CHEMBL3085820)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2L receptor expressed in CHO cell membranes after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239408(CHEMBL4083239)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]spiperone from human D3R expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  12nMAssay Description:Antagonist activity at human adenosine A2A receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50443101(Cariprazine | RGH-188)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2L receptor expressed in CHO cell membranes after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239414(CHEMBL4073330)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50443102(CHEMBL3085819)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-spiperone from human dopamine D2L receptor expressed in CHO cell membranes after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-Nuernberg

Curated by ChEMBL
LigandPNGBDBM50239417(CHEMBL4061986)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]spiperone from human D2SR expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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