Affinity DataKi: 109nMAssay Description:Binding affinity towards GluR1 receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 218nMAssay Description:Binding affinity towards Ionotropic glutamate receptor AMPA 2 from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in absence of L-glutamic acid.More data for this Ligand-Target Pair
Affinity DataKi: 1.76E+3nMAssay Description:Binding affinity towards GluR4 receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 2.14E+3nMAssay Description:Binding affinity towards Ionotropic glutamate receptor AMPA 3 from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in presence of 20 uM L-glutamic acidMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in absence of L-glutamic acid in mammalian cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.20E+4nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in presence of 20 uM L-glutamic acid in mammalian cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.50E+4nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in absence of L-glutamic acid.More data for this Ligand-Target Pair
Affinity DataKi: 5.30E+5nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in presence of 20 uM L-glutamic acid.More data for this Ligand-Target Pair
Affinity DataEC50: 3.43E+4nMAssay Description:The potency at recombinant rat AMPA-R was measured on GluR4 receptor expressed in Xenopus Laevis oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.39E+4nMAssay Description:The potency at recombinant rat AMPA-R was measured on receptor Ionotropic glutamate receptor AMPA 2 expressed in Xenopus Laevis oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.49E+4nMAssay Description:The potency at recombinant rat AMPA-R was measured on GluR1 receptor expressed in Xenopus Laevis oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.24E+5nMAssay Description:The potency at recombinant rat AMPA-R was measured on Ionotropic glutamate receptor AMPA 3 expressed in Xenopus Laevis oocytesMore data for this Ligand-Target Pair