Affinity DataKi: 1.76E+3nMAssay Description:Binding affinity towards GluR4 receptor from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 2.09E+3nMAssay Description:Displacement of (R,S)-[5-methyl-3H]AMPA from rat recombinant flop iGluR4 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.43E+4nMAssay Description:Agonist activity at cyclothiazide-desensitized rat recombinant flop iGluR4c expressed in Xenopus laevis oocytes by two electrode voltage-clamp electr...More data for this Ligand-Target Pair
Affinity DataEC50: 3.43E+4nMAssay Description:The potency at recombinant rat AMPA-R was measured on GluR4 receptor expressed in Xenopus Laevis oocytesMore data for this Ligand-Target Pair