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Found 176 with Last Name = 'smiljanic' and Initial = 'e'
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467114(CHEMBL4285682)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467117(CHEMBL4288816)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467123(CHEMBL4288103)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467126(CHEMBL4286880)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467122(CHEMBL4279865)
Affinity DataIC50:  1nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Lifearc

Curated by ChEMBL
LigandPNGBDBM50507968(CHEMBL4444153)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401907(CHEMBL2207181)
Affinity DataIC50:  2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401928(CHEMBL2207195)
Affinity DataIC50:  2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401913(CHEMBL2207214)
Affinity DataIC50:  2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401915(CHEMBL2207212)
Affinity DataIC50:  2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467128(CHEMBL4286841)
Affinity DataIC50:  2nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401903(CHEMBL2207194)
Affinity DataIC50:  3nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50182362(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401927(CHEMBL2207199)
Affinity DataIC50:  3nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401914(CHEMBL2207213)
Affinity DataIC50:  4nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Lifearc

Curated by ChEMBL
LigandPNGBDBM105071(US8569281, 39)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401918(CHEMBL2207209)
Affinity DataIC50:  4nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467124(CHEMBL4283774)
Affinity DataIC50:  6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467127(CHEMBL4284547)
Affinity DataIC50:  6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401902(CHEMBL2207196)
Affinity DataIC50:  6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401910(CHEMBL2207217)
Affinity DataIC50:  6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401900(CHEMBL2207198)
Affinity DataIC50:  6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50168171(4-(2-(4-fluorophenyl)-5-(1-methylpiperidin-4-yl)-1...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401911(CHEMBL2207216)
Affinity DataIC50:  7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401920(CHEMBL2207206)
Affinity DataIC50:  7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401917(CHEMBL2207210)
Affinity DataIC50:  7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401922(CHEMBL2207204)
Affinity DataIC50:  7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401901(CHEMBL2207197)
Affinity DataIC50:  8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401908(CHEMBL2207180)
Affinity DataIC50:  8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401899(CHEMBL2207208)
Affinity DataIC50:  8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401906(CHEMBL2207187)
Affinity DataIC50:  8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401909(CHEMBL2207218)
Affinity DataIC50:  9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467116(CHEMBL4287934)
Affinity DataIC50:  9nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401912(CHEMBL2207215)
Affinity DataIC50:  9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401924(CHEMBL2207202)
Affinity DataIC50:  9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401916(CHEMBL2207211)
Affinity DataIC50:  10nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401905(CHEMBL2207192)
Affinity DataIC50:  11nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Lifearc

Curated by ChEMBL
LigandPNGBDBM50507979(CHEMBL4589022)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Lifearc

Curated by ChEMBL
LigandPNGBDBM50507672(CHEMBL4460272)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401900(CHEMBL2207198)
Affinity DataIC50:  12nMAssay Description:Inhibition of MARK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401926(CHEMBL2207200)
Affinity DataIC50:  13nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Lifearc

Curated by ChEMBL
LigandPNGBDBM50507981(CHEMBL4561299)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467121(CHEMBL4282026)
Affinity DataIC50:  15nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401925(CHEMBL2207201)
Affinity DataIC50:  15nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401921(CHEMBL2207205)
Affinity DataIC50:  16nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467119(CHEMBL4281827)
Affinity DataIC50:  17nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Plasmodium falciparum)
Lifearc

Curated by ChEMBL
LigandPNGBDBM50467118(CHEMBL4295199)
Affinity DataIC50:  17nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401899(CHEMBL2207208)
Affinity DataIC50:  20nMAssay Description:Inhibition of MARK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401939(CHEMBL2207178)
Affinity DataIC50:  22nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401910(CHEMBL2207217)
Affinity DataIC50:  26nMAssay Description:Inhibition of PDK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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