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Found 81 with Last Name = 'soualmia' and Initial = 'f'
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588058(US11541023, Compound 6)
Affinity DataKi:  670nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588055(US11541023, Compound 3)
Affinity DataKi:  790nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574434(CHEMBL4861066)
Affinity DataKi:  800nMAssay Description:Non-competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588057(US11541023, Compound 5)
Affinity DataKi:  1.00E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574435(CHEMBL4862261)
Affinity DataKi:  1.00E+3nMAssay Description:Competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574434(CHEMBL4861066)
Affinity DataKi:  1.30E+3nMAssay Description:Competitive inhibition of plasmin (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588055(US11541023, Compound 3)
Affinity DataKi:  1.32E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574432(CHEMBL4863108)
Affinity DataKi:  1.50E+3nMAssay Description:Competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574433(CHEMBL4852575)
Affinity DataKi:  1.50E+3nMAssay Description:Competitive inhibition of plasmin (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588054(US11541023, Compound 2)
Affinity DataKi:  1.51E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588058(US11541023, Compound 6)
Affinity DataKi:  1.75E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588056(US11541023, Compound 4)
Affinity DataKi:  1.92E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574431(CHEMBL4847066)
Affinity DataKi:  2.00E+3nMAssay Description:Competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588057(US11541023, Compound 5)
Affinity DataKi:  2.16E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588054(US11541023, Compound 2)
Affinity DataKi:  2.26E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-1(Homo sapiens (Human))
Sorbonne Universit£

Curated by ChEMBL
LigandPNGBDBM50574434(CHEMBL4861066)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of KLK1 (unknown origin) assessed as release of AMC fluorescent product using H-PFR-AMC as substrate incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574433(CHEMBL4852575)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574430(CHEMBL4853943)
Affinity DataKi:  4.30E+3nMAssay Description:Competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588053(US11541023, Compound 1)
Affinity DataKi:  4.44E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588056(US11541023, Compound 4)
Affinity DataKi:  4.66E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588053(US11541023, Compound 1)
Affinity DataKi:  1.44E+4nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574430(CHEMBL4853943)
Affinity DataKi:  1.45E+4nMAssay Description:Competitive inhibition of plasmin (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073221(CHEMBL3408420)
Affinity DataKi:  2.70E+4nMAssay Description:Competitive inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50073222(CHEMBL3125572)
Affinity DataKi:  5.06E+4nMAssay Description:Competitive inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588055(US11541023, Compound 3)
Affinity DataIC50:  1.17E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588055(US11541023, Compound 3)
Affinity DataIC50:  1.23E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (PAR2) and 1 μl o...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588054(US11541023, Compound 2)
Affinity DataIC50:  1.50E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588054(US11541023, Compound 2)
Affinity DataIC50:  1.50E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588058(US11541023, Compound 6)
Affinity DataIC50:  1.56E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574434(CHEMBL4861066)
Affinity DataIC50:  1.57E+3nMAssay Description:Inhibition of KLK6 (unknown origin) assessed as release of AMC fluorescent product using Boc-QAR-AMC as substrate incubated for 30 mins by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574431(CHEMBL4847066)
Affinity DataIC50:  2.37E+3nMAssay Description:Inhibition of KLK6 (unknown origin) assessed as release of AMC fluorescent product using Boc-QAR-AMC as substrate incubated for 30 mins by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588055(US11541023, Compound 3)
Affinity DataIC50:  2.38E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (MBP3) and 1 μl o...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588054(US11541023, Compound 2)
Affinity DataIC50:  2.63E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (PAR2) and 1 μl o...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588057(US11541023, Compound 5)
Affinity DataIC50:  2.72E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588055(US11541023, Compound 3)
Affinity DataIC50:  3.25E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (PAR4) and 1 μl o...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574435(CHEMBL4862261)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of plasmin (unknown origin) assessed as release of AMC fluorescent product using Boc-QAR-AMC as substrate incubated for 30 mins by micropl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574432(CHEMBL4863108)
Affinity DataIC50:  3.63E+3nMAssay Description:Inhibition of KLK6 (unknown origin) assessed as release of AMC fluorescent product using Boc-QAR-AMC as substrate incubated for 30 mins by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588057(US11541023, Compound 5)
Affinity DataIC50:  3.74E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588055(US11541023, Compound 3)
Affinity DataIC50:  3.75E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588058(US11541023, Compound 6)
Affinity DataIC50:  4.78E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574432(CHEMBL4863108)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of plasmin (unknown origin) assessed as release of AMC fluorescent product using Boc-QAR-AMC as substrate incubated for 30 mins by micropl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588054(US11541023, Compound 2)
Affinity DataIC50:  4.92E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (PAR4) and 1 μl o...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588056(US11541023, Compound 4)
Affinity DataIC50:  5.06E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (PAR2) and 1 μl o...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-1(Homo sapiens (Human))
Sorbonne Universit£

Curated by ChEMBL
LigandPNGBDBM50574434(CHEMBL4861066)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of KLK1 (unknown origin) assessed as release of AMC fluorescent product using H-PFR-AMC as substrate incubated for 30 mins by microplate r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM588056(US11541023, Compound 4)
Affinity DataIC50:  5.42E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetKallikrein-1(Homo sapiens (Human))
Sorbonne Universit£

Curated by ChEMBL
LigandPNGBDBM588055(US11541023, Compound 3)
Affinity DataIC50:  5.90E+3nMAssay Description:Table 4: The molecules were tested in order to evaluate their possible inhibitory effect on the enzymatic activity of KLK1. The % inhibitions were de...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574436(CHEMBL4852387)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of plasmin (unknown origin) assessed as release of AMC fluorescent product using Boc-QAR-AMC as substrate incubated for 30 mins by micropl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574433(CHEMBL4852575)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of KLK6 (unknown origin) assessed as release of AMC fluorescent product using Boc-QAR-AMC as substrate incubated for 30 mins by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574435(CHEMBL4862261)
Affinity DataIC50:  7.18E+3nMAssay Description:Inhibition of KLK6 (unknown origin) assessed as release of AMC fluorescent product using Boc-QAR-AMC as substrate incubated for 30 mins by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Sarbonne Universite

US Patent
LigandPNGBDBM50574434(CHEMBL4861066)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of plasmin (unknown origin) assessed as release of AMC fluorescent product using Boc-QAR-AMC as substrate incubated for 30 mins by micropl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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