Affinity DataKi: 0.130nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 120 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence ...More data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 30 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 0.620nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 90 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 0.730nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 60 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 60 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 120 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence ...More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 30 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 90 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 90 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 120 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence ...More data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 30 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 60 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataKi: 99nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibitory activity against human renin inhibition (at pH 7.4)More data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Inhibition of human plasma ACEMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60nMAssay Description:Inhibition of Wistar rat plasma ACEMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against human renin inhibition (at pH 7.4)More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against human renin inhibition (at pH 7.4)More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Compound was tested in vitro for binding affinity against human carbonic anhydrase II; (ki*10e-9)More data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibitory activity against human renin inhibition (at pH 7.4)More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibitory activity against human renin inhibition (at pH 7.4)More data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Inhibitory activity against human renin inhibition (at pH 7.4)More data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of ob/ob mouse plasma ACEMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of ob/ob mouse plasma ACEMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of rat kidney NADPH-dependent aldose reductase assessed as DL-glyceraldehyde conversion to glycerol preincubated for 20 mins followed by N...More data for this Ligand-Target Pair
Affinity DataIC50: 102nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 155nMAssay Description:Inhibition of Wistar rat plasma DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human plasma ACEMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 217nMAssay Description:Inhibition of ob/ob mouse plasma DPP4More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of rat kidney NADPH-dependent aldose reductase assessed as DL-glyceraldehyde conversion to glycerol preincubated for 20 mins followed by N...More data for this Ligand-Target Pair
Affinity DataIC50: 255nMAssay Description:Inhibitory activity against human renin inhibition (at pH 7.4)More data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 279nMAssay Description:Inhibition of human plasma ACEMore data for this Ligand-Target Pair
Affinity DataIC50: 319nMAssay Description:Inhibition of Wistar rat plasma DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 334nMAssay Description:Inhibitory activity against human renin inhibition (at pH 7.4)More data for this Ligand-Target Pair
Affinity DataIC50: 488nMAssay Description:Inhibition of ob/ob mouse plasma DPP4More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of rat kidney NADPH-dependent aldose reductase assessed as DL-glyceraldehyde conversion to glycerol preincubated for 20 mins followed by N...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 690nMAssay Description:Inhibition of rat kidney NADPH-dependent aldose reductase assessed as DL-glyceraldehyde conversion to glycerol preincubated for 20 mins followed by N...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inhibition of rat kidney NADPH-dependent aldose reductase assessed as DL-glyceraldehyde conversion to glycerol preincubated for 20 mins followed by N...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Csir-Indian Institute Of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Inhibition of rat kidney NADPH-dependent aldose reductase assessed as DL-glyceraldehyde conversion to glycerol preincubated for 20 mins followed by N...More data for this Ligand-Target Pair
Affinity DataIC50: 893nMAssay Description:Inhibition of Wistar rat plasma ACEMore data for this Ligand-Target Pair